CN105793247B - 咪唑甲酰胺类及其作为faah抑制剂的用途 - Google Patents

咪唑甲酰胺类及其作为faah抑制剂的用途 Download PDF

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Publication number
CN105793247B
CN105793247B CN201480041611.9A CN201480041611A CN105793247B CN 105793247 B CN105793247 B CN 105793247B CN 201480041611 A CN201480041611 A CN 201480041611A CN 105793247 B CN105793247 B CN 105793247B
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compound
purposes
pharmaceutical composition
imidazole
mmol
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Expired - Fee Related
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CN105793247A (zh
Inventor
卡拉·帕特里夏·达科斯塔·佩特拉·罗莎
丽塔·古斯芒·德诺朗尼亚
拉斯洛·艾尔诺·基斯
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Bial Portela and Cia SA
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Bial Portela and Cia SA
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Priority claimed from GB201313202A external-priority patent/GB201313202D0/en
Priority claimed from GB201313204A external-priority patent/GB201313204D0/en
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CN201480041611.9A 2013-07-24 2014-07-24 咪唑甲酰胺类及其作为faah抑制剂的用途 Expired - Fee Related CN105793247B (zh)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
GB1313202.2 2013-07-24
GB201313202A GB201313202D0 (en) 2013-07-24 2013-07-24 Urea Compound And Its Use As An Enzyme Inhibitor
GB1313203.0 2013-07-24
GB201313204A GB201313204D0 (en) 2013-07-24 2013-07-24 Urea compound and its use as an enzyme inhibitor
GB1313204.8 2013-07-24
GB201313203A GB201313203D0 (en) 2013-07-24 2013-07-24 Urea compound and its use as an enzyme inhibitor
PCT/PT2014/000049 WO2015012708A1 (en) 2013-07-24 2014-07-24 Imidazolecarboxamides and their use as faah inhibitors

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CN105793247A CN105793247A (zh) 2016-07-20
CN105793247B true CN105793247B (zh) 2018-03-16

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SG10201802129QA (en) 2017-07-05 2019-02-27 Frimline Private Ltd A pharmaceutical composition for neuropathic pain
US10702487B2 (en) 2017-08-19 2020-07-07 Frimline Private Limited Pharmaceutical composition for prevention of diet induced obesity
SG10201807034XA (en) 2017-09-05 2019-04-29 Frimline Private Ltd A pharmaceutical composition for improving or preventing progression of Chronic Kidney Disease

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EP0014810A3 (en) 1979-01-18 1980-11-26 Fbc Limited Pesticidal pyrazoles, their production, compositions and uses, as well as intermediates and their preparation
JPH01203366A (ja) 1988-02-10 1989-08-16 Mitsui Petrochem Ind Ltd N−置換イミダゾール誘導体
AU674358B2 (en) 1992-10-28 1996-12-19 Toyama Chemical Co. Ltd. Novel 1,2-benzoisoxazole derivative or its salt and brain -protecting agent comprising the same
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DK1836179T3 (en) * 2004-12-30 2015-05-26 Janssen Pharmaceutica Nv PIPERIDINE AND PIPERAZINE-1-CARBOXYLIC ACID AMIDE DERIVATIVES AND RELATED COMPOUNDS AS MODULATORS OF FAT ACID AMIDE HYDRALASE (FAAH) FOR THE TREATMENT OF ANCIENT, PAIN AND OTHER CONDITIONS
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WO2009126624A1 (en) 2008-04-11 2009-10-15 Bristol-Myers Squibb Company Triazolo compounds useful as dgat1 inhibitors
CA2806701A1 (en) 2010-07-29 2012-02-02 Bial - Portela & Ca, S.A. Process for the synthesis of substituted urea compounds
FR2965262A1 (fr) 2010-09-24 2012-03-30 Sanofi Aventis Derives de nicotinamide, leur preparation et leur application en therapeutique
HRP20180543T1 (hr) 2012-07-24 2018-06-29 Bial-Portela & Ca, S.A. Spojevi uree i njihova upotreba kao inhibitora enzima

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CN105793247A (zh) 2016-07-20
EP3024825B1 (en) 2017-06-21
ES2640800T3 (es) 2017-11-06
KR20160034359A (ko) 2016-03-29
US10501447B2 (en) 2019-12-10
JP6449277B2 (ja) 2019-01-09
HUE033615T2 (hu) 2017-12-28
US20200255412A1 (en) 2020-08-13
CY1119482T1 (el) 2018-03-07
PT3024825T (pt) 2017-09-28
PL3024825T3 (pl) 2017-12-29
LT3024825T (lt) 2017-12-11
MX2016000797A (es) 2016-09-08
AU2014293731B2 (en) 2018-03-08
WO2015012708A1 (en) 2015-01-29
CA2918993A1 (en) 2015-01-29
JP2016525543A (ja) 2016-08-25
US20160176854A1 (en) 2016-06-23
MX362315B (es) 2019-01-11
RU2671404C2 (ru) 2018-10-31
CA2918993C (en) 2021-08-24
EP3024825A1 (en) 2016-06-01
DK3024825T3 (en) 2017-10-02
RU2016104221A (ru) 2017-08-29
AU2014293731A1 (en) 2016-02-11
SI3024825T1 (sl) 2017-11-30
RS56297B1 (sr) 2017-12-29
HRP20171378T1 (hr) 2017-12-15

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