CN104981240B - 通过控制血糖水平用于治疗糖尿病及相关病症的组合物、方法以及用途 - Google Patents

通过控制血糖水平用于治疗糖尿病及相关病症的组合物、方法以及用途 Download PDF

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Publication number
CN104981240B
CN104981240B CN201380069483.4A CN201380069483A CN104981240B CN 104981240 B CN104981240 B CN 104981240B CN 201380069483 A CN201380069483 A CN 201380069483A CN 104981240 B CN104981240 B CN 104981240B
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ifenprodil
composition
glucose
diabetes
compound
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CN104981240A (zh
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丹尼尔·科恩
伊利亚·丘马克威
赛尔格·纳比洛克基恩
鲁道夫·哈吉
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Pharnext SA
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
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    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • Organic Chemistry (AREA)
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  • Molecular Biology (AREA)
  • Hematology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
CN201380069483.4A 2012-10-30 2013-10-30 通过控制血糖水平用于治疗糖尿病及相关病症的组合物、方法以及用途 Expired - Fee Related CN104981240B (zh)

Priority Applications (1)

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CN201910123083.6A CN110141663A (zh) 2012-10-30 2013-10-30 通过控制血糖水平用于治疗糖尿病及相关病症的组合物、方法以及用途

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Application Number Priority Date Filing Date Title
US201261720156P 2012-10-30 2012-10-30
EP12306354.7A EP2727587A1 (en) 2012-10-30 2012-10-30 Compositions, methods and uses for the treatment of diabetes and related conditions by controlling blood glucose level
US61/720,156 2012-10-30
EP12306354.7 2012-10-30
PCT/EP2013/072728 WO2014068007A1 (en) 2012-10-30 2013-10-30 Compositions, methods and uses for the treatment of diabetes and related conditions by controlling blood glucose level

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CN104981240A CN104981240A (zh) 2015-10-14
CN104981240B true CN104981240B (zh) 2019-03-15

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CN201380069483.4A Expired - Fee Related CN104981240B (zh) 2012-10-30 2013-10-30 通过控制血糖水平用于治疗糖尿病及相关病症的组合物、方法以及用途

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US (2) US10092554B2 (enExample)
EP (3) EP2727587A1 (enExample)
JP (2) JP6387010B2 (enExample)
KR (1) KR20150081323A (enExample)
CN (2) CN110141663A (enExample)
AU (2) AU2013340826B2 (enExample)
BR (1) BR112015009702A2 (enExample)
CA (1) CA2888576C (enExample)
EA (1) EA031798B1 (enExample)
ES (2) ES2757846T3 (enExample)
HK (1) HK1214168A1 (enExample)
IL (1) IL238283A0 (enExample)
MX (1) MX2015005368A (enExample)
NZ (1) NZ707139A (enExample)
SG (2) SG11201503225UA (enExample)
WO (1) WO2014068007A1 (enExample)
ZA (1) ZA201503110B (enExample)

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