CN102875430A - 莫达非尼多晶型 - Google Patents
莫达非尼多晶型 Download PDFInfo
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- CN102875430A CN102875430A CN2012103955547A CN201210395554A CN102875430A CN 102875430 A CN102875430 A CN 102875430A CN 2012103955547 A CN2012103955547 A CN 2012103955547A CN 201210395554 A CN201210395554 A CN 201210395554A CN 102875430 A CN102875430 A CN 102875430A
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- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A61P25/20—Hypnotics; Sedatives
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Psychology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
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| US40206402P | 2002-08-09 | 2002-08-09 | |
| US60/402,064 | 2002-08-09 | ||
| US10/635,445 | 2003-08-07 | ||
| US10/635,445 US6992219B2 (en) | 2002-08-09 | 2003-08-07 | Modafinil polymorphic forms |
Related Parent Applications (1)
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| CNB038190850A Division CN100506790C (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
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| CN102875430A true CN102875430A (zh) | 2013-01-16 |
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| CNB038190850A Expired - Fee Related CN100506790C (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
| CN201210395545.8A Expired - Fee Related CN102875429B (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
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| CNB038190850A Expired - Fee Related CN100506790C (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
| CN201210395545.8A Expired - Fee Related CN102875429B (zh) | 2002-08-09 | 2003-08-08 | 莫达非尼多晶型 |
Country Status (11)
| Country | Link |
|---|---|
| US (3) | US6992219B2 (https=) |
| EP (2) | EP1575915A1 (https=) |
| JP (2) | JP4718177B2 (https=) |
| CN (3) | CN102875430A (https=) |
| AU (1) | AU2003253128B2 (https=) |
| CA (4) | CA2494010C (https=) |
| IL (3) | IL166301A (https=) |
| MX (1) | MXPA05001506A (https=) |
| NZ (1) | NZ537840A (https=) |
| WO (1) | WO2004014846A1 (https=) |
| ZA (1) | ZA200500411B (https=) |
Families Citing this family (40)
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|---|---|---|---|---|
| ES2277937T3 (es) | 2000-07-27 | 2007-08-01 | Teva Pharmaceutical Industries Ltd. | Modafinilo puro y cristalino y su procedimiento de preparacion. |
| WO2002092094A1 (en) * | 2001-03-27 | 2002-11-21 | Sumitomo Pharmaceuticals Co., Ltd. | Crystalline isoxazole derivative and medical preparation thereof |
| US6992219B2 (en) * | 2002-08-09 | 2006-01-31 | Cephalon France | Modafinil polymorphic forms |
| FR2849029B1 (fr) * | 2002-12-20 | 2005-03-18 | Lafon Labor | Procede de preparation et formes cristallines des enantiomeres optiques du modafinil. |
| MXPA05008088A (es) * | 2003-02-24 | 2005-09-21 | Mallinckrodt Inc | Proceso mejorado para preparar benzhidril tioacetamida. |
| WO2004083183A1 (en) * | 2003-03-21 | 2004-09-30 | Hetero Drugs Limited | Novel crystalline forms of aripiprazole |
| WO2004085416A1 (en) * | 2003-03-24 | 2004-10-07 | Hetero Drugs Limited | Novel crystalline forms of (s)-citalopram oxalate |
| WO2004085426A1 (en) * | 2003-03-27 | 2004-10-07 | Hetero Drugs Limited | Novel crystalline forms of candesartan cilexetil |
| WO2004087660A1 (en) * | 2003-04-02 | 2004-10-14 | Hetero Drugs Limited | A novel process for amorphous form of donepezil hydrochloride |
| AU2003245029A1 (en) * | 2003-04-16 | 2004-11-04 | Hetero Drugs Limited | Novel crystalline forms of donepezil hydrochloride |
| US20040253308A1 (en) * | 2003-04-29 | 2004-12-16 | Barr Laboratories, Inc. | Surface-treated modafinil particles |
| ES2330321T3 (es) | 2003-05-16 | 2009-12-09 | Cephalon France | Procedimiento de sintesis de modafinilo. |
| US7368591B2 (en) | 2003-09-19 | 2008-05-06 | Cephalon France | Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation |
| PT1673370E (pt) | 2003-10-16 | 2009-11-05 | Symed Labs Ltd | Forma cristalina de linezolida |
| US20090018202A1 (en) * | 2004-02-06 | 2009-01-15 | Cephalon, Inc. | Modafinil compositions |
| EP2292213A1 (en) * | 2004-02-06 | 2011-03-09 | Cephalon, Inc. | Compositions comprising a polymorphic form of armodafinil |
| WO2005099822A2 (en) * | 2004-04-13 | 2005-10-27 | Cephalon, Inc. | Reduction of drug / drug interactions with modafinil |
| WO2005099353A2 (en) * | 2004-04-19 | 2005-10-27 | Symed Labs Limited | A novel process for the preparation of linezolid and related compounds |
| EP1755388B1 (en) * | 2004-05-28 | 2010-10-06 | Transform Pharmaceuticals, Inc. | Mixed co-crystals and pharmaceutical compositions comprising the same |
| JP2008506764A (ja) | 2004-07-20 | 2008-03-06 | ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー | ［Ｒ−（Ｒ＊，Ｒ＊）］−２−（４−フルオロフェニル）−β、δ−ジヒドロキシ−５−（１−メチルエチル）−３−フェニル−４−［（フェニルアミノ）カルボニル］−１Ｈ−ピロール−１−ヘプタン酸カルシウム塩（２：１）の新規形態 |
| WO2006018853A2 (en) | 2004-08-19 | 2006-02-23 | Hetero Drugs Limited | Novel polymorphs of efavirenz |
| AU2006272874B2 (en) * | 2005-07-21 | 2010-03-11 | Neurohealing Pharmaceuticals, Inc. | Rapid onset and short term modafinil compositions and methods of use thereof |
| US7518019B2 (en) * | 2006-06-01 | 2009-04-14 | Hetero Drugs Limited | Processes for preparing sertraline hydrochloride crystalline forms |
| AU2007272501A1 (en) * | 2006-07-12 | 2008-01-17 | Elan Pharma International Limited | Nanoparticulate formulations of modafinil |
| WO2008021341A2 (en) * | 2006-08-14 | 2008-02-21 | Neurohealing Pharmaceuticals, Inc. | Modafinil-based treatment for premature ejaculation |
| UA110598C2 (uk) | 2006-11-10 | 2016-01-25 | Басф Се | Спосіб одержання кристалічної модифікації фіпронілу |
| NZ576524A (en) | 2006-11-10 | 2012-01-12 | Basf Se | Crystalline modification of fipronil |
| AU2007316640B2 (en) | 2006-11-10 | 2012-11-29 | Basf Se | Crystalline modification of fipronil |
| WO2008068767A2 (en) * | 2006-12-07 | 2008-06-12 | Hetero Drugs Limited | A novel crystalline form of lansoprazole |
| US20100010092A1 (en) * | 2006-12-19 | 2010-01-14 | Arless Ltd. | Use of modafinil to treat restless leg syndrome |
| US20100234468A1 (en) * | 2007-06-04 | 2010-09-16 | Abhay Gaitonde | Novel process |
| FR2923482B1 (fr) * | 2007-11-09 | 2010-01-29 | Servier Lab | Nouvelle forme cristalline vi de l'agomelatine, son procede de preparation et les compositions pharmaceutiques qui la contiennent |
| TW200930343A (en) * | 2007-09-21 | 2009-07-16 | Organon Nv | Drug delivery system |
| WO2009045488A2 (en) * | 2007-10-02 | 2009-04-09 | Teva Pharmaceutical Industries Ltd. | Novel crystalline forms of armodafinil and preparation thereof |
| US9265458B2 (en) | 2012-12-04 | 2016-02-23 | Sync-Think, Inc. | Application of smooth pursuit cognitive testing paradigms to clinical drug development |
| US9380976B2 (en) | 2013-03-11 | 2016-07-05 | Sync-Think, Inc. | Optical neuroinformatics |
| WO2015086489A1 (en) | 2013-12-11 | 2015-06-18 | Merck Sharp & Dohme B.V. | Drug delivery system for delivery of anti-virals |
| US10413504B2 (en) | 2013-12-11 | 2019-09-17 | Merck Sharp & Dohme Corp. | Intravaginal ring drug delivery system |
| US9616068B2 (en) | 2014-10-27 | 2017-04-11 | Pohela LLC | Animal training using cognitive enhancement |
| PT4210709T (pt) | 2020-09-14 | 2026-02-04 | Pharma Cinq Llc | 2¿,3¿‐diacetiluridina substituída com acetoacetilo na posição 5¿ |
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-
2003
- 2003-08-07 US US10/635,445 patent/US6992219B2/en not_active Expired - Fee Related
- 2003-08-08 WO PCT/IB2003/003215 patent/WO2004014846A1/en not_active Ceased
- 2003-08-08 JP JP2004527153A patent/JP4718177B2/ja not_active Expired - Fee Related
- 2003-08-08 AU AU2003253128A patent/AU2003253128B2/en not_active Ceased
- 2003-08-08 CN CN2012103955547A patent/CN102875430A/zh active Pending
- 2003-08-08 CN CNB038190850A patent/CN100506790C/zh not_active Expired - Fee Related
- 2003-08-08 NZ NZ537840A patent/NZ537840A/en not_active IP Right Cessation
- 2003-08-08 MX MXPA05001506A patent/MXPA05001506A/es active IP Right Grant
- 2003-08-08 CN CN201210395545.8A patent/CN102875429B/zh not_active Expired - Fee Related
- 2003-08-08 CA CA2494010A patent/CA2494010C/en not_active Expired - Fee Related
- 2003-08-08 CA CA2746788A patent/CA2746788C/en not_active Expired - Fee Related
- 2003-08-08 EP EP03784340A patent/EP1575915A1/en not_active Withdrawn
- 2003-08-08 CA CA2840721A patent/CA2840721C/en not_active Expired - Fee Related
- 2003-08-08 CA CA2804385A patent/CA2804385A1/en not_active Abandoned
- 2003-08-08 EP EP11171058A patent/EP2402311A1/en not_active Withdrawn
-
2005
- 2005-01-13 IL IL166301A patent/IL166301A/en not_active IP Right Cessation
- 2005-01-17 ZA ZA2005/00411A patent/ZA200500411B/en unknown
- 2005-10-12 US US11/248,442 patent/US7405323B2/en not_active Expired - Fee Related
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2007
- 2007-12-14 US US11/956,877 patent/US7649020B2/en not_active Expired - Fee Related
-
2010
- 2010-10-20 JP JP2010235766A patent/JP5307106B2/ja not_active Expired - Fee Related
- 2010-12-13 IL IL209965A patent/IL209965A0/en unknown
- 2010-12-13 IL IL209966A patent/IL209966A/en not_active IP Right Cessation
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| US5180745A (en) * | 1990-06-14 | 1993-01-19 | Laboratoire L. Lafon | Method for providing a neuroprotective effect |
| US5391576A (en) * | 1991-12-13 | 1995-02-21 | Laboratoire L. Lafon | Method for treating and protecting the cerebral tissue against repercussions of cerebral ischaemia and cerebral infarctions |
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| US5612379A (en) * | 1993-06-22 | 1997-03-18 | Laboratoire L. Lafon | Modafinil for the treatment of sleep apneas and ventilatory disorders of central origin |
| WO1999025329A1 (fr) * | 1997-11-19 | 1999-05-27 | Institut Curie | Utilisation de derives de benzhydryl sulfinyle pour traiter la somnolence d'origine medicamenteuse |
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Effective date of registration: 20151110 Address after: Paris France Applicant after: Teva Sante Address before: French Maisons Alfort Applicant before: Saifulun European Co. Effective date of registration: 20151110 Address after: French Maisons Alfort Applicant after: Saifulun European Co. Address before: French Maisons Alfort Applicant before: Cephalon France |
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