PT1673370E - Forma cristalina de linezolida - Google Patents
Forma cristalina de linezolida Download PDFInfo
- Publication number
- PT1673370E PT1673370E PT03769887T PT03769887T PT1673370E PT 1673370 E PT1673370 E PT 1673370E PT 03769887 T PT03769887 T PT 03769887T PT 03769887 T PT03769887 T PT 03769887T PT 1673370 E PT1673370 E PT 1673370E
- Authority
- PT
- Portugal
- Prior art keywords
- linezolid
- crystalline form
- preparation
- relates
- present
- Prior art date
Links
- TYZROVQLWOKYKF-ZDUSSCGKSA-N linezolid Chemical compound O=C1O[C@@H](CNC(=O)C)CN1C(C=C1F)=CC=C1N1CCOCC1 TYZROVQLWOKYKF-ZDUSSCGKSA-N 0.000 title abstract 2
- 229960003907 linezolid Drugs 0.000 title abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/IN2003/000336 WO2005035530A1 (en) | 2003-10-16 | 2003-10-16 | A novel crystalline form of linezolid |
Publications (1)
Publication Number | Publication Date |
---|---|
PT1673370E true PT1673370E (pt) | 2009-11-05 |
Family
ID=34430675
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT03769887T PT1673370E (pt) | 2003-10-16 | 2003-10-16 | Forma cristalina de linezolida |
Country Status (10)
Country | Link |
---|---|
US (4) | US7714128B2 (pt) |
EP (3) | EP2100884A1 (pt) |
AT (1) | ATE442364T1 (pt) |
AU (1) | AU2003278592A1 (pt) |
DE (2) | DE09163348T1 (pt) |
DK (1) | DK1673370T3 (pt) |
ES (3) | ES2331001T3 (pt) |
HU (1) | HUE051230T2 (pt) |
PT (1) | PT1673370E (pt) |
WO (1) | WO2005035530A1 (pt) |
Families Citing this family (36)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2100884A1 (en) | 2003-10-16 | 2009-09-16 | Symed Labs Limited | Crystalline form of linezolid |
WO2005099353A2 (en) | 2004-04-19 | 2005-10-27 | Symed Labs Limited | A novel process for the preparation of linezolid and related compounds |
EP1745028A2 (en) * | 2004-06-29 | 2007-01-24 | Teva Pharmaceutical Industries Ltd | Solid forms of linezolid and processes for preparation thereof |
CA2572054A1 (en) * | 2004-06-29 | 2006-01-12 | Teva Pharmaceutical Industries Ltd. | Crystalline form iv of linezolid |
JP2008530028A (ja) * | 2005-02-24 | 2008-08-07 | テバ ファーマシューティカル インダストリーズ リミティド | リネゾリッド中間体の調製方法 |
WO2007018588A1 (en) * | 2005-07-20 | 2007-02-15 | Teva Pharmaceutical Industries Ltd. | Stable pharmaceutical composition comprising linezolid form iv |
IT1390957B1 (it) * | 2008-07-07 | 2011-10-27 | Dipharma Francis Srl | Sali di linezolid e loro uso nella preparazione di forme cristalline di linezolid |
EP2033960A3 (en) | 2007-09-04 | 2009-04-29 | Dipharma Francis S.r.l. | Linezolid crystalline hydrate form and linezolid salts |
US20090093631A1 (en) * | 2007-09-06 | 2009-04-09 | Ben-Zion Dolitzky | Processes for the preparation of a linezolid intermediate, linezolid hydroxide |
WO2009140466A2 (en) * | 2008-05-14 | 2009-11-19 | Dr. Reddy's Laboratories Ltd. | Linezolid co-crystals |
EP2493867A1 (en) | 2009-10-28 | 2012-09-05 | Synthon BV | Process for making crystalline form a of linezolid |
WO2011050826A1 (en) | 2009-10-28 | 2011-05-05 | Synthon B.V. | Process for making crystalline form a of linezolid |
US20130137864A1 (en) | 2009-12-26 | 2013-05-30 | Jayaraman Venkat Raman | Process for the preparation of linezolid |
CN103140487A (zh) | 2010-08-11 | 2013-06-05 | 斯索恩有限公司 | 制备利奈唑胺的方法 |
EP2690100A1 (en) | 2010-08-11 | 2014-01-29 | Synhton B.V. | Process for making linezolid |
WO2012029074A2 (en) | 2010-09-02 | 2012-03-08 | Hetero Research Foundation | Pharmaceutical compositions of linezolid |
CN102070548B (zh) * | 2011-01-13 | 2012-12-26 | 浙江新东港药业股份有限公司 | 一种晶型ⅰ型利奈唑胺的蒸发结晶工艺 |
EP2593440A1 (en) | 2011-02-24 | 2013-05-22 | Lee Pharma Limited | Anhydrous linezolid crystalline form-ii |
EP2683696A1 (en) | 2011-03-09 | 2014-01-15 | Synthon BV | Process for making crystalline form a of linezolid |
CN105461648B (zh) * | 2011-05-03 | 2018-01-12 | 江苏豪森药业集团有限公司 | 利奈唑胺的晶型及其制备方法 |
ITMI20111311A1 (it) * | 2011-07-14 | 2013-01-15 | Dipharma Francis Srl | Sali di linezolid e loro uso nella preparazione di forme cristalline di linezolid |
WO2013072923A1 (en) * | 2011-09-19 | 2013-05-23 | Cadila Healthcare Limited | Process for the preparation of crystalline linezolid |
WO2013093751A1 (en) * | 2011-12-24 | 2013-06-27 | Alembic Pharmaceuticals Limited | Packaging for linezolid |
WO2013111048A1 (en) * | 2012-01-24 | 2013-08-01 | Jubilant Life Sciences Limited | Improved process for the preparation of stable crystalline form-i of linezolid, substantially free of residual solvent |
WO2013120496A1 (en) | 2012-02-14 | 2013-08-22 | Pharmathen S.A. | Process for the preparation of linezolid in crystalline form and salts thereof |
WO2013190559A1 (en) * | 2012-06-19 | 2013-12-27 | Symed Labs Limited | Improved processes for the preparation of linezolid crystalline form iii |
US9492459B2 (en) * | 2012-08-10 | 2016-11-15 | Indoco Remedies Limited | Pharmaceutical composition of linezolid |
EP2917189B1 (en) | 2012-11-09 | 2016-08-17 | Synthon BV | Process for making linezolid |
WO2014118809A1 (en) | 2013-01-29 | 2014-08-07 | Actavis Group Ptc Ehf. | Pharmaceutical composition with linezolid |
IN2013MU03508A (pt) | 2013-11-06 | 2015-07-24 | Unimark Remedies Ltd | |
CN105254580B (zh) * | 2014-04-22 | 2018-01-02 | 江苏豪森药业集团有限公司 | 利奈唑胺晶型的制备方法 |
WO2016113751A1 (en) * | 2015-01-13 | 2016-07-21 | Nosch Labs Private Limited | Process for preparing crystalline linezolid form-iii |
WO2018051360A1 (en) * | 2016-09-16 | 2018-03-22 | Lee Pharma Limited | A novel process for the preparation of crystalline linezolid form-iii |
US11517574B2 (en) | 2017-11-16 | 2022-12-06 | Persica Pharmaceuticals Ltd. | Linezolid formulations |
CN110194750A (zh) * | 2019-06-19 | 2019-09-03 | 四川美大康华康药业有限公司 | 一种利奈唑胺的制备方法及精制方法 |
WO2023062080A1 (en) | 2021-10-12 | 2023-04-20 | Persica Pharmaceuticals Ltd. | Low back pain treatment |
Family Cites Families (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US583870A (en) * | 1897-06-01 | Wrench | ||
DE2810349A1 (de) | 1978-03-10 | 1979-09-20 | Kali Chemie Pharma Gmbh | Verfahren zur herstellung von 3-hydroxy-6-phenyl-1,2,3,4-tetrahydro- 1,5-benzodiazocinen |
FR2506769A2 (fr) | 1978-06-09 | 1982-12-03 | Delalande Sa | Para-((cyano-5 n pentyl-1) phenyl)-3 methoxymethyl-5 oxazolidinone-2, son procede de preparation et ses applications en therapeutique |
US4340606A (en) | 1980-10-23 | 1982-07-20 | E. I. Du Pont De Nemours And Company | 3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents |
FR2608604B1 (fr) | 1986-12-19 | 1989-04-28 | Delalande Sa | Derives 5-hydroxyethyles de l'oxazolidinone-2, leurs procedes de preparation et leurs applications en therapeutique |
US5006528A (en) * | 1988-10-31 | 1991-04-09 | Otsuka Pharmaceutical Co., Ltd. | Carbostyril derivatives |
DE9310451U1 (de) | 1993-03-05 | 1994-06-30 | Landis & Gyr Business Support | Steuer- bzw. Regeleinrichtung für Gas-Feuerungsautomaten von Heizungsanlagen |
EP0615095B1 (de) | 1993-03-11 | 1997-05-07 | Landis & Gyr Technology Innovation AG | Brennerregler |
MY115155A (en) | 1993-09-09 | 2003-04-30 | Upjohn Co | Substituted oxazine and thiazine oxazolidinone antimicrobials. |
US5688792A (en) | 1994-08-16 | 1997-11-18 | Pharmacia & Upjohn Company | Substituted oxazine and thiazine oxazolidinone antimicrobials |
ATE209193T1 (de) | 1996-04-11 | 2001-12-15 | Upjohn Co | Verfahren zur herstellung von oxazolidinonen |
EP0890791A1 (de) | 1997-07-11 | 1999-01-13 | Electrowatt Technology Innovation AG | Steuer- und Regelgerät für einen Brenner |
CZ20001613A3 (cs) | 1997-11-07 | 2001-12-12 | Pharmacia & Upjohn Company | Způsob výroby oxazolidinonů |
US6444813B2 (en) | 2000-02-02 | 2002-09-03 | Pharmacia & Upjohn Company | Linezolid-crystal form II |
AR027261A1 (es) | 2000-02-02 | 2003-03-19 | Upjohn Co | Linezolid forma cristalina ii |
MY127336A (en) * | 2000-03-22 | 2006-11-30 | Upjohn Co | Container for linezolid iv solution |
DE10037585A1 (de) * | 2000-08-02 | 2002-02-14 | Valeo Schalter & Sensoren Gmbh | Rückstellvorrichtung für einen Blinkerschalter in Kraftfahrzeugen |
HUP0302874A2 (hu) | 2000-08-14 | 2003-12-29 | Teva Pharmaceutical Industries Ltd. | Eljárás risperidon előállítására |
EP1365739A1 (en) * | 2001-02-05 | 2003-12-03 | Pharmacia & Upjohn Company | Composition for rectal delivery of an oxazolidinone antibacterial drug |
NZ528996A (en) * | 2001-04-20 | 2006-01-27 | Upjohn Co | Process to prepare oxazolidinones |
CN1155585C (zh) | 2001-12-19 | 2004-06-30 | 中国医学科学院医药生物技术研究所 | 3,5-取代噁唑烷酮衍生物及其制备方法和应用 |
US6992219B2 (en) | 2002-08-09 | 2006-01-31 | Cephalon France | Modafinil polymorphic forms |
EP2100884A1 (en) | 2003-10-16 | 2009-09-16 | Symed Labs Limited | Crystalline form of linezolid |
WO2005099353A2 (en) | 2004-04-19 | 2005-10-27 | Symed Labs Limited | A novel process for the preparation of linezolid and related compounds |
CA2572054A1 (en) | 2004-06-29 | 2006-01-12 | Teva Pharmaceutical Industries Ltd. | Crystalline form iv of linezolid |
PL1768967T3 (pl) | 2004-07-20 | 2009-09-30 | Symed Labs Ltd | Nowe związki pośrednie do wytwarzania linezolidu oraz związki pokrewne |
-
2003
- 2003-10-16 EP EP20090163348 patent/EP2100884A1/en not_active Withdrawn
- 2003-10-16 WO PCT/IN2003/000336 patent/WO2005035530A1/en active Application Filing
- 2003-10-16 DK DK03769887T patent/DK1673370T3/da active
- 2003-10-16 DE DE2009163348 patent/DE09163348T1/de active Pending
- 2003-10-16 AU AU2003278592A patent/AU2003278592A1/en not_active Abandoned
- 2003-10-16 AT AT03769887T patent/ATE442364T1/de active
- 2003-10-16 EP EP15155714.7A patent/EP2902386B1/en not_active Expired - Lifetime
- 2003-10-16 EP EP03769887A patent/EP1673370B1/en not_active Revoked
- 2003-10-16 US US10/524,478 patent/US7714128B2/en active Active
- 2003-10-16 PT PT03769887T patent/PT1673370E/pt unknown
- 2003-10-16 DE DE60329237T patent/DE60329237D1/de not_active Expired - Lifetime
- 2003-10-16 ES ES03769887T patent/ES2331001T3/es not_active Expired - Lifetime
- 2003-10-16 ES ES15155714T patent/ES2803516T3/es not_active Expired - Lifetime
- 2003-10-16 ES ES09163348T patent/ES2331454T1/es active Pending
- 2003-10-16 HU HUE15155714A patent/HUE051230T2/hu unknown
-
2007
- 2007-09-26 US US11/861,340 patent/US7718799B2/en not_active Expired - Fee Related
- 2007-09-26 US US11/861,406 patent/US7732597B2/en not_active Expired - Fee Related
- 2007-09-26 US US11/861,433 patent/US7718800B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US7718800B2 (en) | 2010-05-18 |
EP1673370B1 (en) | 2009-09-09 |
US20060128703A1 (en) | 2006-06-15 |
EP2902386B1 (en) | 2020-04-08 |
ATE442364T1 (de) | 2009-09-15 |
US20080090824A1 (en) | 2008-04-17 |
DE09163348T1 (de) | 2010-01-07 |
ES2331454T1 (es) | 2010-01-05 |
US20080090820A1 (en) | 2008-04-17 |
EP2100884A1 (en) | 2009-09-16 |
WO2005035530A1 (en) | 2005-04-21 |
AU2003278592A1 (en) | 2005-04-27 |
HUE051230T2 (hu) | 2021-03-01 |
DE60329237D1 (de) | 2009-10-22 |
EP1673370A1 (en) | 2006-06-28 |
DK1673370T3 (da) | 2009-12-07 |
US7732597B2 (en) | 2010-06-08 |
ES2331001T3 (es) | 2009-12-18 |
US7714128B2 (en) | 2010-05-11 |
US20080091011A1 (en) | 2008-04-17 |
US7718799B2 (en) | 2010-05-18 |
EP2902386A1 (en) | 2015-08-05 |
ES2803516T3 (es) | 2021-01-27 |
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