CN1019492B - 制备苯并-和噻唑并-咪唑并二氮杂衍生物的方法 - Google Patents

制备苯并-和噻唑并-咪唑并二氮杂衍生物的方法

Info

Publication number
CN1019492B
CN1019492B CN85101490A CN85101490A CN1019492B CN 1019492 B CN1019492 B CN 1019492B CN 85101490 A CN85101490 A CN 85101490A CN 85101490 A CN85101490 A CN 85101490A CN 1019492 B CN1019492 B CN 1019492B
Authority
CN
China
Prior art keywords
imidazo
benzodiazepine
chloro
mmol
mixture
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CN85101490A
Other languages
English (en)
Chinese (zh)
Other versions
CN85101490A (zh
Inventor
瓦尔特·亨克勒
凯伯茨
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Jean Jakes Ogrey
F Hoffmann La Roche AG
Original Assignee
Jean Jakes Ogrey
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jean Jakes Ogrey, F Hoffmann La Roche AG filed Critical Jean Jakes Ogrey
Priority to CN85101490A priority Critical patent/CN1019492B/zh
Publication of CN85101490A publication Critical patent/CN85101490A/zh
Publication of CN1019492B publication Critical patent/CN1019492B/zh
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CN85101490A 1984-01-19 1985-04-01 制备苯并-和噻唑并-咪唑并二氮杂衍生物的方法 Expired CN1019492B (zh)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN85101490A CN1019492B (zh) 1984-01-19 1985-04-01 制备苯并-和噻唑并-咪唑并二氮杂衍生物的方法

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH22584 1984-01-19
CN85101490A CN1019492B (zh) 1984-01-19 1985-04-01 制备苯并-和噻唑并-咪唑并二氮杂衍生物的方法

Publications (2)

Publication Number Publication Date
CN85101490A CN85101490A (zh) 1987-01-24
CN1019492B true CN1019492B (zh) 1992-12-16

Family

ID=4182136

Family Applications (1)

Application Number Title Priority Date Filing Date
CN85101490A Expired CN1019492B (zh) 1984-01-19 1985-04-01 制备苯并-和噻唑并-咪唑并二氮杂衍生物的方法

Country Status (5)

Country Link
KR (1) KR850005443A (cg-RX-API-DMAC10.html)
CN (1) CN1019492B (cg-RX-API-DMAC10.html)
BR (1) BR8500228A (cg-RX-API-DMAC10.html)
GR (1) GR850137B (cg-RX-API-DMAC10.html)
ZA (1) ZA85362B (cg-RX-API-DMAC10.html)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA110640C2 (uk) * 2011-05-05 2016-01-25 Янссен Фармацевтика Нв ПРОТИГРИБКОВІ 5,6-ДИГІДРО-4Н-ПІРОЛО[1,2-a][1,4]БЕНЗОДІАЗЕПІНИ ТА 6Н-ПІРОЛО[1,2-a][1,4]БЕНЗОДІАЗЕПІНИ, ЯКІ ЗАМІЩЕНІ ГЕТЕРОЦИКЛІЧНИМИ ПОХІДНИМИ
CN107325101B (zh) * 2017-06-29 2019-03-26 上海合全药物研发有限公司 6-羟甲基-6,7-二氢-5h,9h-咪唑并二氮杂卓-8-羧酸叔丁酯的合成方法
CN111606926B (zh) * 2020-05-13 2021-10-15 大连理工大学 一种苯并咪唑[1,3]氮硫杂卓类化合物的制备方法

Also Published As

Publication number Publication date
GR850137B (cg-RX-API-DMAC10.html) 1985-05-20
KR850005443A (ko) 1985-08-26
CN85101490A (zh) 1987-01-24
ZA85362B (en) 1985-09-25
BR8500228A (pt) 1985-08-27

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