CN101812056A - 作为单胺神经递质再摄取抑制剂的新颖烷基取代的哌啶衍生物 - Google Patents
作为单胺神经递质再摄取抑制剂的新颖烷基取代的哌啶衍生物 Download PDFInfo
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- CN101812056A CN101812056A CN201010178208A CN201010178208A CN101812056A CN 101812056 A CN101812056 A CN 101812056A CN 201010178208 A CN201010178208 A CN 201010178208A CN 201010178208 A CN201010178208 A CN 201010178208A CN 101812056 A CN101812056 A CN 101812056A
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- 150000004685 tetrahydrates Chemical class 0.000 description 1
- 125000000383 tetramethylene group Chemical group [H]C([H])([*:1])C([H])([H])C([H])([H])C([H])([H])[*:2] 0.000 description 1
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Classifications
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
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- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Child & Adolescent Psychology (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| DKPA200400960 | 2004-06-18 | ||
| DKPA200400960 | 2004-06-18 |
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| CNA2005800172613A Division CN1960985A (zh) | 2004-06-18 | 2005-06-14 | 作为单胺神经递质再摄取抑制剂的新颖烷基取代的哌啶衍生物 |
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| CNA2005800172613A Pending CN1960985A (zh) | 2004-06-18 | 2005-06-14 | 作为单胺神经递质再摄取抑制剂的新颖烷基取代的哌啶衍生物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
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| CNA2005800172613A Pending CN1960985A (zh) | 2004-06-18 | 2005-06-14 | 作为单胺神经递质再摄取抑制剂的新颖烷基取代的哌啶衍生物 |
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| JP (1) | JP2008502653A (https=) |
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| CA (1) | CA2570065A1 (https=) |
| MX (1) | MXPA06013918A (https=) |
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| WO (1) | WO2005123715A1 (https=) |
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| JP2010527915A (ja) * | 2007-04-26 | 2010-08-19 | アバロン ファーマシューティカルズ，インコーポレイテッド | 多重環化合物及びその用途 |
| AU2009264334A1 (en) * | 2008-06-27 | 2009-12-30 | Neurosearch A/S | Novel tetramethyl substituted piperidine derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| US20110263651A1 (en) * | 2008-11-26 | 2011-10-27 | Neurosearch A/S | Novel piperidine-butyramide derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
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| CA284097A (en) * | 1928-10-16 | Schonhofer Fritz | Pharmaceutical product | |
| US718124A (en) * | 1902-05-19 | 1903-01-13 | John B Heydt | Loaf-forming device. |
| US1760781A (en) * | 1926-12-20 | 1930-05-27 | Winthrop Chem Co Inc | Manufacture of new pharmaceutical products |
| DE490275C (de) * | 1926-12-20 | 1930-02-05 | I G Farbenindustrie Akt Ges | Verfahren zur Darstellung N-substituierter Amine der carbo- und heterocyclischen Reihen |
| NL21937C (https=) * | 1926-12-20 | |||
| GB1393551A (en) * | 1972-04-21 | 1975-05-07 | Ciba Geigy Ag | Piperidine derivatives |
| JP3087763B2 (ja) * | 1990-11-30 | 2000-09-11 | 三井化学株式会社 | 新規な複素環式化合物およびそれを含有する医薬組成物 |
| DE4228792A1 (de) * | 1992-08-29 | 1994-03-03 | Hoechst Ag | Pyridylaminopiperidine, Verfahren zu ihrer Herstellung, sie enthaltende Mittel und deren Verwendung als Fungizide |
| PL167185B1 (pl) * | 1992-09-09 | 1995-08-31 | Univ Lodzki | Sposób równoczesnego otrzymywania izomerycznych pochodnych 3-pirydynokarbonitrylu |
| US5494908A (en) * | 1992-11-23 | 1996-02-27 | Hoechst-Roussel Pharmaceutical Incorporated | Substituted 3-(aminoalkylamino)-1,2-benzisoxazoles and related compounds |
| US5852037A (en) * | 1995-11-13 | 1998-12-22 | Eli Lilly And Company | Method for treating anxiety |
| US5804622A (en) * | 1996-03-22 | 1998-09-08 | Ciba Specialty Chemicals Corporation | Monomeric N-piperidinylmelamines as stabilizers for chlorine-containing polymers |
| ES2128978B1 (es) * | 1996-04-01 | 2000-03-01 | Ciba Sc Holding Ag | Derivados de politriazina que contienen grupos de polialquilpiperidiniloxilo o polialquilpiperidinilamino. |
| ATE247104T1 (de) * | 1997-11-05 | 2003-08-15 | Neurosearch As | Azaring-ether-derivate und ihre verwendung als nicotinic-ach-rezeptormodulatoren |
| JP3589160B2 (ja) * | 2000-07-07 | 2004-11-17 | 日本電気株式会社 | レジスト用材料、化学増幅型レジスト及びそれを用いたパターン形成方法 |
| JPWO2002100833A1 (ja) * | 2001-06-12 | 2004-09-24 | 住友製薬株式会社 | Ｒｈｏキナーゼ阻害剤 |
| WO2003062224A1 (en) * | 2002-01-17 | 2003-07-31 | Eli Lilly And Company | Aza-cyclic compounds as modulators of acetylcholine receptors |
| GB0308466D0 (en) * | 2003-04-11 | 2003-05-21 | Novartis Ag | Organic compounds |
| MXPA05011223A (es) * | 2003-04-18 | 2006-01-26 | Lilly Co Eli | Compuestos de (piperidiniloxi)fenilo, (piperidiniloxi)piridinilo, (piperidinilsulfanil)fenilo y (piperidinilsulfanil)piridinilo como agonistas 5-htif. |
| EP1638939A2 (en) * | 2003-06-24 | 2006-03-29 | Neurosearch A/S | Aza-ring derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| RU2344136C2 (ru) * | 2003-06-24 | 2009-01-20 | НьюроСёрч А/С | Новые производные 8-аза-бицикло[3.2.1]октана и их применение в качестве ингибиторов обратного захвата моноаминовых нейротрансмиттеров |
| BRPI0413018B8 (pt) * | 2003-07-30 | 2021-05-25 | Rigel Pharmaceuticals Inc | composto, e, uso de um composto |
-
2005
- 2005-06-14 EP EP05752808A patent/EP1761518A1/en not_active Withdrawn
- 2005-06-14 CA CA002570065A patent/CA2570065A1/en not_active Abandoned
- 2005-06-14 CN CN201010178208A patent/CN101812056A/zh active Pending
- 2005-06-14 CN CNA2005800172613A patent/CN1960985A/zh active Pending
- 2005-06-14 MX MXPA06013918A patent/MXPA06013918A/es not_active Application Discontinuation
- 2005-06-14 US US11/579,059 patent/US20070232659A1/en not_active Abandoned
- 2005-06-14 WO PCT/EP2005/052733 patent/WO2005123715A1/en not_active Ceased
- 2005-06-14 JP JP2007515946A patent/JP2008502653A/ja not_active Abandoned
- 2005-06-17 AR ARP050102509A patent/AR049923A1/es unknown
- 2005-06-17 TW TW094120096A patent/TW200603803A/zh unknown
-
2009
- 2009-11-09 US US12/614,857 patent/US20100056567A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| AR049923A1 (es) | 2006-09-13 |
| US20070232659A1 (en) | 2007-10-04 |
| TW200603803A (en) | 2006-02-01 |
| JP2008502653A (ja) | 2008-01-31 |
| CA2570065A1 (en) | 2005-12-29 |
| CN1960985A (zh) | 2007-05-09 |
| EP1761518A1 (en) | 2007-03-14 |
| MXPA06013918A (es) | 2007-03-07 |
| US20100056567A1 (en) | 2010-03-04 |
| WO2005123715A1 (en) | 2005-12-29 |
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