CN101618038B - 化合物在制备治疗抗生素耐药性细菌感染的药物中的用途 - Google Patents
化合物在制备治疗抗生素耐药性细菌感染的药物中的用途 Download PDFInfo
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- CN101618038B CN101618038B CN2008101700068A CN200810170006A CN101618038B CN 101618038 B CN101618038 B CN 101618038B CN 2008101700068 A CN2008101700068 A CN 2008101700068A CN 200810170006 A CN200810170006 A CN 200810170006A CN 101618038 B CN101618038 B CN 101618038B
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
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| KR101392808B1 (ko) * | 2011-12-30 | 2014-05-12 | 순천대학교 산학협력단 | 식물 추출물 또는 이의 분획물을 포함하는 항균용 조성물 |
| CN103145615B (zh) * | 2013-03-20 | 2015-07-29 | 浙江医药股份有限公司 | 一种奈诺沙星螯合物的后处理方法 |
| KR101392810B1 (ko) * | 2013-09-25 | 2014-05-12 | 순천대학교 산학협력단 | 된장풀 추출물 또는 이의 분획물을 포함하는 항균용 조성물 |
| US9492374B2 (en) | 2015-03-25 | 2016-11-15 | Jose Rafael Salinas Andrade | Composition and method for treatment of ulcers |
| CN105368825B (zh) * | 2015-10-14 | 2019-09-10 | 华东医院 | 幽门螺杆菌抗生素耐药性分析试剂盒及耐药性检测方法 |
| US12358902B2 (en) * | 2017-12-11 | 2025-07-15 | Denovamed Inc. | 5-(2,5-bis(4-chloro-2-isopropylphenyl)thiophen-3-yl)-1H-tetrazole for the topical treatment of bacterial infections |
| CN111979292B (zh) * | 2020-07-27 | 2022-08-05 | 广东省微生物研究所（广东省微生物分析检测中心） | 一种同时携带多重耐药基因cfr和lsa(E)的MRSA的用途 |
| CN114437026A (zh) * | 2021-10-26 | 2022-05-06 | 浙江医药股份有限公司新昌制药厂 | 一种低组合物杂质的苹果酸奈诺沙星原料药及其制备方法 |
| CN118852222B (zh) * | 2024-06-27 | 2025-09-05 | 南京桦冠生物技术有限公司 | 一种奈诺沙星中间体及其制备方法和应用 |
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| US100800A (en) | 1870-03-15 | Improvement in riding attachments for plows | ||
| US3989816A (en) | 1975-06-19 | 1976-11-02 | Nelson Research & Development Company | Vehicle composition containing 1-substituted azacycloheptan-2-ones |
| US4444762A (en) | 1980-04-04 | 1984-04-24 | Nelson Research & Development Company | Vehicle composition containing 1-substituted azacyclopentan-2-ones |
| US6387928B1 (en) * | 1997-09-15 | 2002-05-14 | The Procter & Gamble Co. | Antimicrobial quinolones, their compositions and uses |
| US6348624B1 (en) | 1998-01-09 | 2002-02-19 | The Procter & Gamble Co. | Process for making certain benzoic acid compounds |
| DK1343766T3 (da) | 2000-12-14 | 2005-10-31 | Procter & Gamble | Procestrin med cyklisering ved fremstilling af quinoloner og naphthyridiner |
| US6900224B2 (en) * | 2002-07-31 | 2005-05-31 | The Procter & Gamble Company | Antimicrobial quinolones, their compositions and uses |
| US6803469B2 (en) | 2002-08-05 | 2004-10-12 | The Procter & Gamble Company | Process for preparing quinolone antibiotic intermediates |
| WO2005026145A2 (en) * | 2003-09-12 | 2005-03-24 | Warner-Lambert Company Llc | Quinolone antibacterial agents |
| DK2001862T3 (da) | 2006-03-28 | 2011-08-08 | Warner Chilcott Co Llc | Malatsalte og polymorfe af (3S,5S)-7-[3-amino-5-methyl-piperidinyl]-1-cyklopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolincarboxylsyre |
| JP4876165B2 (ja) | 2006-03-28 | 2012-02-15 | ザ プロクター アンド ギャンブル カンパニー | キノロン中間体を調製するための水素化物還元法 |
| BRPI0709220A2 (pt) * | 2006-03-28 | 2011-07-12 | Procter & Gamble | processo de acoplamento para preparo de intermediários de quinolona |
| US8658183B2 (en) | 2007-08-09 | 2014-02-25 | Taigen Biotechnology Company, Ltd. | Antimicrobial parenteral formulation |
| US20120157492A1 (en) | 2008-07-15 | 2012-06-21 | Taigen Biotechnology Co., Ltd. | Antibiotic drug |
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| EP2303271B1 (en) | 2018-11-07 |
| ZA201100616B (en) | 2011-10-26 |
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| JP2011526887A (ja) | 2011-10-20 |
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| TWI375558B (en) | 2012-11-01 |
| EP2303271A1 (en) | 2011-04-06 |
| CN101618038A (zh) | 2010-01-06 |
| EA018653B1 (ru) | 2013-09-30 |
| NZ588898A (en) | 2012-09-28 |
| TR201820964T4 (tr) | 2019-01-21 |
| EP2303271A4 (en) | 2012-01-25 |
| TW201002322A (en) | 2010-01-16 |
| CA2728328C (en) | 2015-02-24 |
| WO2010002415A1 (en) | 2010-01-07 |
| US20100004282A1 (en) | 2010-01-07 |
| AU2008358909B2 (en) | 2012-12-13 |
| KR20110044168A (ko) | 2011-04-28 |
| CA2728328A1 (en) | 2010-01-07 |
| KR20150006080A (ko) | 2015-01-15 |
| AU2008358909A1 (en) | 2010-01-07 |
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