CN101578275A - 苯胺基哌嗪衍生物及其使用方法 - Google Patents

苯胺基哌嗪衍生物及其使用方法 Download PDF

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Publication number
CN101578275A
CN101578275A CNA2007800490776A CN200780049077A CN101578275A CN 101578275 A CN101578275 A CN 101578275A CN A2007800490776 A CNA2007800490776 A CN A2007800490776A CN 200780049077 A CN200780049077 A CN 200780049077A CN 101578275 A CN101578275 A CN 101578275A
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China
Prior art keywords
compound
alkyl
alkylidene group
preparation
cancer
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CNA2007800490776A
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Chinese (zh)
Inventor
G·W·小席普
C·C·程
X·黄
T·O·菲斯柯曼
J·S·杜卡
M·里察斯
H·曾
B·孙
P·A·兰迪
T·T·王
P·K·塔迪肯德
M·A·西迪昆
M·M·拉伯里
C·波克
T·J·古奇
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Merck Sharp and Dohme LLC
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Schering Corp
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Publication of CN101578275A publication Critical patent/CN101578275A/zh
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CNA2007800490776A 2006-10-31 2007-10-29 苯胺基哌嗪衍生物及其使用方法 Pending CN101578275A (zh)

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US85565406P 2006-10-31 2006-10-31
US60/855,654 2006-10-31

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CN101578275A true CN101578275A (zh) 2009-11-11

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US (1) US9206142B2 (de)
EP (1) EP2078003B1 (de)
JP (1) JP5063700B2 (de)
KR (1) KR20090075873A (de)
CN (1) CN101578275A (de)
AR (1) AR063721A1 (de)
AU (1) AU2007314342B2 (de)
CA (1) CA2668210C (de)
IL (1) IL198397A0 (de)
MX (1) MX2009004786A (de)
TW (1) TW200829583A (de)
WO (1) WO2008054702A1 (de)

Cited By (8)

* Cited by examiner, † Cited by third party
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CN102603667A (zh) * 2012-02-10 2012-07-25 合肥工业大学 一种n-(2-氯-6-甲基苯基)-2-(苯丙烯酰胺)噻唑-5-甲酰胺衍生物、其制备方法及其用途
CN102993124A (zh) * 2012-11-25 2013-03-27 大理学院 取代哌嗪类化合物及其制备方法和药物用途
WO2014194667A1 (zh) * 2013-06-05 2014-12-11 中国科学院上海药物研究所 一类炔基杂环类化合物及其应用
CN105555785A (zh) * 2013-06-18 2016-05-04 4Sc新发现股份有限公司 作为dyrk激酶抑制剂的2，3-二氢苯并呋喃-5-基化合物
CN105829293A (zh) * 2013-12-20 2016-08-03 中国人民解放军军事医学科学院毒物药物研究所 新型哌啶氨甲酰类化合物、制备方法及其用途
CN112204017A (zh) * 2018-04-27 2021-01-08 国立大学法人大阪大学 苯并异噁唑化合物
CN113620863A (zh) * 2015-09-14 2021-11-09 内盖夫国家生物技术研究所 新的哌嗪和哌啶衍生物、它们的合成及其用途
CN115590854A (zh) * 2019-12-25 2023-01-13 安斯泰来制药株式会社（Jp） 哒嗪基噻唑甲酰胺类化合物

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CA2649043C (en) * 2006-04-19 2013-09-17 Astellas Pharma Inc. Azolecarboxamide derivative
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