CN101356179A - 脂肪酶抑制剂 - Google Patents
脂肪酶抑制剂 Download PDFInfo
- Publication number
- CN101356179A CN101356179A CNA2005800464039A CN200580046403A CN101356179A CN 101356179 A CN101356179 A CN 101356179A CN A2005800464039 A CNA2005800464039 A CN A2005800464039A CN 200580046403 A CN200580046403 A CN 200580046403A CN 101356179 A CN101356179 A CN 101356179A
- Authority
- CN
- China
- Prior art keywords
- compound
- alkyl
- inhibitor
- lipase
- thiazolinyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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| US62747604P | 2004-11-12 | 2004-11-12 | |
| US60/627,476 | 2004-11-12 |
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| CN101356179A true CN101356179A (zh) | 2009-01-28 |
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| JO3598B1 (ar) | 2006-10-10 | 2020-07-05 | Infinity Discovery Inc | الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني |
| US8653258B2 (en) * | 2007-06-08 | 2014-02-18 | Georgia State University Research Foundation, Inc. | Compositions for regulating or modulating quorum sensing in bacteria, methods of using the compounds, and methods of regulating or modulating quorum sensing in bacteria |
| PE20091838A1 (es) | 2008-04-09 | 2009-12-18 | Infinity Pharmaceuticals Inc | Inhibidores de amida hidrolasa de acido graso |
| JP5605844B2 (ja) | 2008-10-17 | 2014-10-15 | 塩野義製薬株式会社 | 血管内皮リパーゼ阻害活性を有する酢酸アミド誘導体 |
| ES2493916T3 (es) | 2009-04-07 | 2014-09-12 | Infinity Pharmaceuticals, Inc. | Inhibidores de hidrolasa de amida de ácidos grasos |
| US8541581B2 (en) | 2009-04-07 | 2013-09-24 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
| EP2243423B1 (de) * | 2009-04-23 | 2012-05-02 | Roche Diagnostics GmbH | Verfahren und Gerät zur Ermittlung von Empfehlungen für Wirkstoffdosierungen anhand von Messserien zumindest eines physiologischen Parameters eines Patienten |
| US8754113B2 (en) | 2009-12-15 | 2014-06-17 | Shionogi & Co., Ltd. | Oxadiazole derivative having endothelial lipase inhibitory activity |
| MX336742B (es) | 2010-02-03 | 2016-01-29 | Infinity Pharmaceuticals Inc | Inhibidores de amida hidrolasa de acido graso. |
| EP2575823A1 (en) * | 2010-05-31 | 2013-04-10 | Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. | 3-substituted vinylboronates and uses thereof |
| CN105806967B (zh) * | 2014-12-31 | 2018-02-06 | 广州朗圣药业有限公司 | 依折麦布关键中间体4‑[[(4‑氟苯基)亚胺]甲基]‑苯酚的分析方法 |
| CN105572252A (zh) * | 2015-12-18 | 2016-05-11 | 武汉武药科技有限公司 | 一种分析/分离依折麦布(r,r,s)型的光学异构体的方法 |
| EP3765006A4 (en) * | 2018-03-13 | 2022-02-23 | Merck Sharp & Dohme Corp. | ARGINASE INHIBITORS AND METHODS OF USE |
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| UA58494C2 (uk) | 1995-06-07 | 2003-08-15 | Зенека Лімітед | Похідні n-гетероарилпіридинсульфонаміду, фармацевтична композиція, спосіб одержання та спосіб протидії впливам ендотеліну |
| JP3456511B2 (ja) * | 1997-01-27 | 2003-10-14 | 昭和電工株式会社 | 陰イオンの分析法及び陰イオン分析セット |
| JPH10210999A (ja) * | 1997-01-29 | 1998-08-11 | Eiken Chem Co Ltd | エステル加水分解酵素活性の阻害方法 |
| TW458977B (en) | 1997-04-16 | 2001-10-11 | Abbott Lab | 6,7-disubstituted-4-aminopyrido[2,3-D] pyrimidine compounds |
| US6858592B2 (en) * | 2001-06-29 | 2005-02-22 | Genzyme Corporation | Aryl boronic acids for treating obesity |
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2005
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- 2005-11-14 US US11/719,159 patent/US20090209492A1/en not_active Abandoned
- 2005-11-14 KR KR1020077013216A patent/KR20070086076A/ko not_active Application Discontinuation
- 2005-11-14 CN CNA2005800464039A patent/CN101356179A/zh active Pending
- 2005-11-14 BR BRPI0517840-1A patent/BRPI0517840A/pt not_active IP Right Cessation
- 2005-11-14 EP EP05851568A patent/EP1824861A2/en not_active Withdrawn
- 2005-11-14 CA CA002586479A patent/CA2586479A1/en not_active Abandoned
- 2005-11-14 WO PCT/US2005/041022 patent/WO2006053250A2/en active Application Filing
- 2005-11-14 AU AU2005304318A patent/AU2005304318A1/en not_active Abandoned
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2007
- 2007-05-10 IL IL183129A patent/IL183129A0/en unknown
- 2007-06-12 NO NO20073011A patent/NO20073011L/no not_active Application Discontinuation
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2011
- 2011-10-28 US US13/284,230 patent/US20120101062A1/en not_active Abandoned
Also Published As
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|---|---|
| NO20073011L (no) | 2007-08-08 |
| EP1824861A2 (en) | 2007-08-29 |
| WO2006053250A3 (en) | 2008-07-10 |
| BRPI0517840A (pt) | 2008-10-21 |
| CA2586479A1 (en) | 2006-05-18 |
| AU2005304318A1 (en) | 2006-05-18 |
| WO2006053250A2 (en) | 2006-05-18 |
| JP2008519853A (ja) | 2008-06-12 |
| US20120101062A1 (en) | 2012-04-26 |
| KR20070086076A (ko) | 2007-08-27 |
| US20090209492A1 (en) | 2009-08-20 |
| IL183129A0 (en) | 2008-04-13 |
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