CN101254172A - 一种呱西替柳干混悬剂及其制备方法 - Google Patents
一种呱西替柳干混悬剂及其制备方法 Download PDFInfo
- Publication number
- CN101254172A CN101254172A CNA2008100011941A CN200810001194A CN101254172A CN 101254172 A CN101254172 A CN 101254172A CN A2008100011941 A CNA2008100011941 A CN A2008100011941A CN 200810001194 A CN200810001194 A CN 200810001194A CN 101254172 A CN101254172 A CN 101254172A
- Authority
- CN
- China
- Prior art keywords
- guacetisal
- dry suspension
- weight portion
- dry
- suspension
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Images
Landscapes
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Description
实施例2 | 实施例3 | 实施例4 | 实施例5 | 实施例6 | 实施例7 | |
呱西替柳(g) | 160 | 170 | 163 | 162 | 168 | 125 |
羟丙甲纤维素(g) | 5 | 5 | 8 | 9 | 7 | 6 |
十二烷基硫酸钠(g) | 8 | 6 | 7 | 9 | 5 | 4 |
蔗糖(g) | 815 | 818 | 819 | 816 | 815 | 817 |
鲜奶香精(g) | 12 | 1 | 3 | 4 | 5 | 适量 |
200410068927.5 | 本发明 | |
沉降体积比 | 0.93 | 0.97 |
项目 | 本发明呱西替柳干混悬剂 | 200410068927.5的呱西替柳干混悬剂 | 本发明呱西替柳干混悬剂放置6个月后 | 200410068927.5的呱西替柳干混悬剂放置6个月后 |
沉降体积比 | 0.968 | 0.931 | 0.962 | 0.890 |
降解产物(%) | 0.6 | 0.7 | 0.63 | 1.3 |
含量(%) | 103.8 | 102.5 | 103.2 | 100.1 |
200410068927.5 | 本发明 | |
Cmax | 16.70±3.45 | 18.50±5.46 |
Tmax | 2.4±1.0 | 2.3±2.0 |
T1/2 | 2.56±0.85 | 3.56±0.88 |
AUC0-t | 93.2±21.7 | 96.2±23.7 |
AUC0-∞ | 97.4±24.3 | 98.8±26.3 |
Claims (7)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CNB2008100011941A CN100484515C (zh) | 2007-08-14 | 2008-01-18 | 一种呱西替柳干混悬剂及其制备方法 |
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN200710016385.0 | 2007-08-14 | ||
CN200710016385 | 2007-08-14 | ||
CNB2008100011941A CN100484515C (zh) | 2007-08-14 | 2008-01-18 | 一种呱西替柳干混悬剂及其制备方法 |
Publications (2)
Publication Number | Publication Date |
---|---|
CN101254172A true CN101254172A (zh) | 2008-09-03 |
CN100484515C CN100484515C (zh) | 2009-05-06 |
Family
ID=39889500
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CNB2008100011941A Active CN100484515C (zh) | 2007-08-14 | 2008-01-18 | 一种呱西替柳干混悬剂及其制备方法 |
Country Status (1)
Country | Link |
---|---|
CN (1) | CN100484515C (zh) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103102271A (zh) * | 2012-02-29 | 2013-05-15 | 大连名森制药有限公司 | 一种呱西替柳的工业化制备方法及干混悬剂的医药用途 |
-
2008
- 2008-01-18 CN CNB2008100011941A patent/CN100484515C/zh active Active
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103102271A (zh) * | 2012-02-29 | 2013-05-15 | 大连名森制药有限公司 | 一种呱西替柳的工业化制备方法及干混悬剂的医药用途 |
CN103102271B (zh) * | 2012-02-29 | 2014-09-03 | 大连名森制药有限公司 | 一种呱西替柳的工业化制备方法及干混悬剂的医药用途 |
Also Published As
Publication number | Publication date |
---|---|
CN100484515C (zh) | 2009-05-06 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CN1377270A (zh) | β-咔啉药物产品 | |
CN106539768B (zh) | 一种盐酸鲁拉西酮口腔崩解片及其制备方法 | |
CN109662950B (zh) | 一种含有盐酸达泊西汀的药物组合物 | |
CN104546851A (zh) | 一种颗粒组合物及其制备方法、制剂 | |
CN101926840B (zh) | 一种紫锥菊的超微粉散剂及其制备方法和应用 | |
CN106511348B (zh) | 石杉碱甲骨架微粒、口崩片及其制备方法 | |
CN101766578B (zh) | 一种含瑞舒伐他汀钙的片剂及其制备工艺 | |
CN109893503A (zh) | 一种艾曲泊帕口服混悬液及其制备方法 | |
CN100484515C (zh) | 一种呱西替柳干混悬剂及其制备方法 | |
CN102462675A (zh) | 一种苯扎贝特缓释片及其制备方法 | |
CN103007286B (zh) | 一种托伐普坦的固体药物组合物 | |
CN114652692B (zh) | 一种治疗肝病的药物缓释片及其制备方法和用途 | |
Rekha et al. | Formulation and development of Bilastine tablets 20 mg | |
CN114601803B (zh) | 一种巴洛沙韦酯干混悬剂及其制备方法和应用 | |
CN109381431B (zh) | 石杉碱甲缓释微丸及其制备方法 | |
CN104415034A (zh) | 一种咪达那新药物组合物及其制备方法 | |
CN102240282B (zh) | 穿琥宁口服药物组合物及其制备方法 | |
CN102600149A (zh) | 一种治疗糖尿病的药物组合物 | |
CN102641253B (zh) | 缬沙坦缓释片及其制备方法 | |
CN107449844B (zh) | 一种测定二巯丁二酸制剂溶出度的方法 | |
CN104257618B (zh) | 一种含有法罗培南钠的口腔崩解片及其制备方法 | |
CN101081213B (zh) | 丁二酸(5-雄甾烯-17-酮-3β-羟基)二酯固体分散体及其制备方法与应用 | |
CN104644558A (zh) | 一种西尼地平的固体分散体及其制备方法 | |
CN113368066B (zh) | 一种淫羊藿苷元片剂及其制备方法 | |
CN113750051B (zh) | 一种供口服给药的固体化穿心莲内酯溶液及其制备方法 |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
C06 | Publication | ||
PB01 | Publication | ||
C10 | Entry into substantive examination | ||
SE01 | Entry into force of request for substantive examination | ||
C14 | Grant of patent or utility model | ||
GR01 | Patent grant | ||
C56 | Change in the name or address of the patentee |
Owner name: SHANDONG LUOXIN PHARMACY GROUP CO., LTD. Free format text: FORMER NAME: SHANDONG LUOXIN PHARMACY STOCK CO., LTD. |
|
CP01 | Change in the name or title of a patent holder |
Address after: Seven of 276017 Shandong province Linyi city Luozhuang District Patentee after: Shandong Luo Xin Pharmaceutical Group Plc Address before: Seven of 276017 Shandong province Linyi city Luozhuang District Patentee before: SHANDONG LUOXIN PHARMACY STOCK Co., LTD. |
|
C41 | Transfer of patent application or patent right or utility model | ||
TR01 | Transfer of patent right |
Effective date of registration: 20160726 Address after: Seven of 276017 Shandong province Linyi city Luozhuang District Patentee after: Shandong Luo Xin Pharmaceutical Group Plc Patentee after: Luo Xin Biotechnology (Shanghai) Co., Ltd. Address before: Seven of 276017 Shandong province Linyi city Luozhuang District Patentee before: Shandong Luo Xin Pharmaceutical Group Plc |
|
CP03 | Change of name, title or address |
Address after: 276017 18 Luo Qi Road, Luozhuang District, Linyi, Shandong Co-patentee after: Luoxin Pharmaceutical (Shanghai) Co., Ltd. Patentee after: Shandong Luo Xin Pharmaceutical Group Plc Address before: 276017 Luoqi Road, Luozhuang District, Linyi City, Shandong Province Co-patentee before: Luo Xin Biotechnology (Shanghai) Co., Ltd. Patentee before: Shandong Luo Xin Pharmaceutical Group Plc |
|
CP03 | Change of name, title or address |