CN101193869B - 糖皮质激素模拟物、其制备方法、药物组合物及其用途 - Google Patents

糖皮质激素模拟物、其制备方法、药物组合物及其用途 Download PDF

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CN101193869B
CN101193869B CN2006800205382A CN200680020538A CN101193869B CN 101193869 B CN101193869 B CN 101193869B CN 2006800205382 A CN2006800205382 A CN 2006800205382A CN 200680020538 A CN200680020538 A CN 200680020538A CN 101193869 B CN101193869 B CN 101193869B
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trifluoro
indazol
phenyl
fluorophenyl
ethanol
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CN101193869A (zh
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英戈·A·马格
迈克尔·J·伯克
马克·S·拉尔夫
戴维·S·汤姆森
阿卜杜拉金·哈马克
詹妮弗·A·科瓦尔斯基
乔尔格·M·本齐恩
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Boehringer Ingelheim International GmbH
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  • Diabetes (AREA)
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  • Ophthalmology & Optometry (AREA)
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  • Cardiology (AREA)
  • Dermatology (AREA)
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  • Urology & Nephrology (AREA)
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  • Obesity (AREA)
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  • Child & Adolescent Psychology (AREA)
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CN2006800205382A 2005-06-10 2006-06-08 糖皮质激素模拟物、其制备方法、药物组合物及其用途 Expired - Fee Related CN101193869B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US68941205P 2005-06-10 2005-06-10
US60/689,412 2005-06-10
PCT/US2006/022651 WO2006135826A1 (en) 2005-06-10 2006-06-08 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof

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CN101193869A CN101193869A (zh) 2008-06-04
CN101193869B true CN101193869B (zh) 2011-03-02

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US (1) US7622594B2 (cg-RX-API-DMAC10.html)
EP (1) EP1893588A1 (cg-RX-API-DMAC10.html)
JP (1) JP2008543780A (cg-RX-API-DMAC10.html)
KR (1) KR20080027828A (cg-RX-API-DMAC10.html)
CN (1) CN101193869B (cg-RX-API-DMAC10.html)
AR (1) AR058006A1 (cg-RX-API-DMAC10.html)
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NZ538932A (en) * 2002-08-29 2007-04-27 Boehringer Ingelheim Pharma 3-(sulfonamidoethyl)-indole derivatives for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative disease
UY28526A1 (es) 2003-09-24 2005-04-29 Boehringer Ingelheim Pharma Miméticos de glucocorticoides, métodos de preparación composiciones farmacéuticas y usos de los mismos
US7795272B2 (en) 2004-03-13 2010-09-14 Boehringer Ingelheim Pharmaceutical, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof
PE20060776A1 (es) 2004-12-27 2006-09-26 Boehringer Ingelheim Pharma Mimeticos de glucocorticoides, metodos para prepararlos y composiciones farmaceuticas
JP2010500300A (ja) 2006-08-08 2010-01-07 サノフィ−アベンティス アリールアミノアリール−アルキル−置換イミダゾリジン−２，４−ジオン、それらの製造法、それらの化合物を含有する薬剤、およびそれらの使用
JP2010508358A (ja) * 2006-11-01 2010-03-18 ブリストル−マイヤーズ スクイブ カンパニー グルココルチコイド受容体、ＡＰ−１、および／またはＮＦ−κＢ活性の調節剤、並びにその使用
TW200829578A (en) 2006-11-23 2008-07-16 Astrazeneca Ab Chemical compounds 537
MX2009005264A (es) 2006-12-06 2009-05-28 Boehringer Ingelheim Int Mimeticos de glucocorticoides, metodos para su fabricacion, composiciones farmaceuticas y usos de los mismos.
JO2754B1 (en) 2006-12-21 2014-03-15 استرازينكا ايه بي Amylendazoleil derivatives for the treatment of glucocorticoid-mediated disorders
WO2008079073A1 (en) * 2006-12-22 2008-07-03 Astrazeneca Ab Indazolyl sulphonamide derivatives for the treatment of glucocorticoid receptor mediated disorders
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CN101193869A (zh) 2008-06-04
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US20070060633A1 (en) 2007-03-15
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