CL2016000787A1 - Composición farmacéutica en forma de comprimido que comprende atazanavir y cobicistat; procedimiento de preparación; y uso de la composición para preparar un medicamento útil para tratar la infección por el virus de inmunodeficiencia humana (vih). - Google Patents

Composición farmacéutica en forma de comprimido que comprende atazanavir y cobicistat; procedimiento de preparación; y uso de la composición para preparar un medicamento útil para tratar la infección por el virus de inmunodeficiencia humana (vih).

Info

Publication number
CL2016000787A1
CL2016000787A1 CL2016000787A CL2016000787A CL2016000787A1 CL 2016000787 A1 CL2016000787 A1 CL 2016000787A1 CL 2016000787 A CL2016000787 A CL 2016000787A CL 2016000787 A CL2016000787 A CL 2016000787A CL 2016000787 A1 CL2016000787 A1 CL 2016000787A1
Authority
CL
Chile
Prior art keywords
composition
cobicistat
tablet
atazanavir
hiv
Prior art date
Application number
CL2016000787A
Other languages
English (en)
Inventor
Otilia May Yue Koo
Faranak Nikfar
Jing Tao
Niranjan Kumar Kottala
Sailesh A Varia
Original Assignee
Bristol Myers Squibb Holdings Ireland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=51743576&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2016000787(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Holdings Ireland filed Critical Bristol Myers Squibb Holdings Ireland
Publication of CL2016000787A1 publication Critical patent/CL2016000787A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418—Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente solicitud describe a una composición farmacéutica en forma de comprimido que comprende atazanavir y cobicistat en forma de cobicistat en dióxido de silicio; un procedimiento de preparación de la composición en forma de comprimido; y su uso para preparar un medicamento para tratar la infección por el virus de inmunodeficiencia humana (VIH).
CL2016000787A 2013-10-07 2016-04-05 Composición farmacéutica en forma de comprimido que comprende atazanavir y cobicistat; procedimiento de preparación; y uso de la composición para preparar un medicamento útil para tratar la infección por el virus de inmunodeficiencia humana (vih). CL2016000787A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201361887574P 2013-10-07 2013-10-07

Publications (1)

Publication Number Publication Date
CL2016000787A1 true CL2016000787A1 (es) 2016-11-25

Family

ID=51743576

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2016000787A CL2016000787A1 (es) 2013-10-07 2016-04-05 Composición farmacéutica en forma de comprimido que comprende atazanavir y cobicistat; procedimiento de preparación; y uso de la composición para preparar un medicamento útil para tratar la infección por el virus de inmunodeficiencia humana (vih).

Country Status (27)

Country Link
US (2) US20160038502A1 (es)
EP (2) EP3054926B1 (es)
JP (2) JP6574415B2 (es)
KR (1) KR102286386B1 (es)
CN (1) CN106029058A (es)
AU (1) AU2014332200B2 (es)
BR (1) BR112016007526A8 (es)
CA (1) CA2926650A1 (es)
CL (1) CL2016000787A1 (es)
CY (1) CY1121105T1 (es)
DK (2) DK3054926T3 (es)
EA (1) EA031172B1 (es)
ES (2) ES2693580T3 (es)
HR (2) HRP20221126T1 (es)
HU (1) HUE059757T2 (es)
IL (1) IL244881B (es)
LT (2) LT3054926T (es)
MX (1) MX368268B (es)
MY (1) MY178960A (es)
PE (1) PE20160596A1 (es)
PL (2) PL3054926T3 (es)
PT (2) PT3421033T (es)
RS (2) RS63570B1 (es)
SA (1) SA516370891B1 (es)
SG (1) SG11201602501VA (es)
SI (2) SI3054926T1 (es)
WO (1) WO2015054133A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20130203759A1 (en) * 2010-04-09 2013-08-08 Faranak Nikfar ATAZANAVIR SULFATE FORMULATIONS WITH IMPROVED pH EFFECT
MA43114A (fr) 2015-10-30 2018-09-05 Cancer Prevention Pharmaceuticals Inc Formulation combinée à dose fixe d'éflornithine et sulindac
CA2937365C (en) 2016-03-29 2018-09-18 F. Hoffmann-La Roche Ag Granulate formulation of 5-methyl-1-phenyl-2-(1h)-pyridone and method of making the same
BR112019002120A2 (pt) * 2016-08-08 2019-05-14 Hetero Labs Limited composição anti-retroviral de várias classes
US11045423B2 (en) 2016-08-08 2021-06-29 Hetero Labs Limited Anti-retroviral compositions

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5558071A (en) * 1994-03-07 1996-09-24 Combustion Electromagnetics, Inc. Ignition system power converter and controller
US5849911A (en) 1996-04-22 1998-12-15 Novartis Finance Corporation Antivirally active heterocyclic azahexane derivatives
IL134830A0 (en) * 2000-03-01 2001-05-20 Chay 13 Medical Res Group N V Peptides and immunostimulatory and anti-bacterial pharmaceutical compositions containing them
EP1267912A2 (en) * 2000-03-14 2003-01-02 Burkhard Göke Effects of glucagon-like peptide-1 (7-36) on antro-pyloro-duodenal motility
KR101329658B1 (ko) * 2006-09-25 2013-11-14 아처 다니엘 미드랜드 캄파니 초흡수성 표면처리된 카르복시알킬화 다당류 및 그 제조방법
AR065439A1 (es) 2007-02-23 2009-06-10 Gilead Sciences Inc Derivados de tiazoles 1,3 no condensados,composiciones farmaceuticas que los contienen y usos como agentes antivirales, en particular anti hiv.
ES2360336T3 (es) * 2007-06-22 2011-06-03 Bristol-Myers Squibb Company Composiciones en comprimidos que contienen atazanavir.
US20130084243A1 (en) * 2010-01-27 2013-04-04 Liliane Goetsch Igf-1r specific antibodies useful in the detection and diagnosis of cellular proliferative disorders
WO2009084036A2 (en) * 2007-12-20 2009-07-09 Matrix Laboratories Limited Composition for treatment of viral infections
EP2889029A1 (en) * 2008-09-25 2015-07-01 Cephalon, Inc. Liquid formulations of bendamustine
US20110028412A1 (en) * 2009-08-03 2011-02-03 Cappellos, Inc. Herbal enhanced analgesic formulations
US20130203759A1 (en) * 2010-04-09 2013-08-08 Faranak Nikfar ATAZANAVIR SULFATE FORMULATIONS WITH IMPROVED pH EFFECT

Also Published As

Publication number Publication date
MY178960A (en) 2020-10-26
LT3421033T (lt) 2022-11-10
EP3054926B1 (en) 2018-07-25
JP6574415B2 (ja) 2019-09-11
EP3421033A1 (en) 2019-01-02
EA031172B1 (ru) 2018-11-30
PT3054926T (pt) 2018-10-26
ES2693580T3 (es) 2018-12-12
SA516370891B1 (ar) 2018-08-08
ES2927484T3 (es) 2022-11-07
IL244881B (en) 2021-12-01
RS63570B1 (sr) 2022-10-31
AU2014332200B2 (en) 2018-10-04
WO2015054133A1 (en) 2015-04-16
MX2016004078A (es) 2016-06-06
AU2014332200A1 (en) 2016-05-19
EP3054926A1 (en) 2016-08-17
SI3421033T1 (sl) 2022-11-30
LT3054926T (lt) 2018-11-12
IL244881A0 (en) 2016-05-31
US20160038502A1 (en) 2016-02-11
EA201690594A1 (ru) 2016-09-30
CN106029058A (zh) 2016-10-12
HRP20181582T1 (hr) 2018-11-30
DK3421033T3 (da) 2022-10-10
JP2019011334A (ja) 2019-01-24
BR112016007526A8 (pt) 2020-03-03
CA2926650A1 (en) 2015-04-16
HRP20221126T1 (hr) 2022-11-25
MX368268B (es) 2019-09-26
PL3054926T3 (pl) 2018-12-31
PT3421033T (pt) 2022-09-23
RS57882B1 (sr) 2019-01-31
HUE059757T2 (hu) 2023-01-28
DK3054926T3 (en) 2018-10-29
SG11201602501VA (en) 2016-04-28
US20190358240A1 (en) 2019-11-28
KR102286386B1 (ko) 2021-08-05
CY1121105T1 (el) 2019-12-11
PL3421033T3 (pl) 2022-10-03
PE20160596A1 (es) 2016-06-15
BR112016007526A2 (pt) 2017-08-01
EP3421033B1 (en) 2022-07-27
SI3054926T1 (sl) 2018-10-30
JP2016532649A (ja) 2016-10-20
KR20160060764A (ko) 2016-05-30

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