CL2013003556A1 - Compuestos derivados de ftalazinona-pirrolo[3,2-d]pirimidin-carboxamida, inhibidoers de fosfodiesterasa tipo 4 y tipo 5; composcin farmaceutica que o comprende, combinacion fija, no fija y kit, uso del compuesto en la preparacion de un medicamento para trata enfermedaes de las vias respiratorias - Google Patents
Compuestos derivados de ftalazinona-pirrolo[3,2-d]pirimidin-carboxamida, inhibidoers de fosfodiesterasa tipo 4 y tipo 5; composcin farmaceutica que o comprende, combinacion fija, no fija y kit, uso del compuesto en la preparacion de un medicamento para trata enfermedaes de las vias respiratoriasInfo
- Publication number
- CL2013003556A1 CL2013003556A1 CL2013003556A CL2013003556A CL2013003556A1 CL 2013003556 A1 CL2013003556 A1 CL 2013003556A1 CL 2013003556 A CL2013003556 A CL 2013003556A CL 2013003556 A CL2013003556 A CL 2013003556A CL 2013003556 A1 CL2013003556 A1 CL 2013003556A1
- Authority
- CL
- Chile
- Prior art keywords
- type
- fixed
- phthalazinone
- pyrrolo
- pyrimidine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP11170440 | 2011-06-17 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2013003556A1 true CL2013003556A1 (es) | 2014-06-13 |
Family
ID=44764312
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2013003556A CL2013003556A1 (es) | 2011-06-17 | 2013-12-11 | Compuestos derivados de ftalazinona-pirrolo[3,2-d]pirimidin-carboxamida, inhibidoers de fosfodiesterasa tipo 4 y tipo 5; composcin farmaceutica que o comprende, combinacion fija, no fija y kit, uso del compuesto en la preparacion de un medicamento para trata enfermedaes de las vias respiratorias |
Country Status (21)
Country | Link |
---|---|
US (2) | US20140112945A1 (es) |
EP (1) | EP2721030B1 (es) |
JP (1) | JP5980318B2 (es) |
KR (1) | KR20140037195A (es) |
CN (1) | CN103582644B (es) |
AR (1) | AR086915A1 (es) |
AU (1) | AU2012269133A1 (es) |
BR (1) | BR112013031791A2 (es) |
CA (1) | CA2837248A1 (es) |
CL (1) | CL2013003556A1 (es) |
CO (1) | CO6852074A2 (es) |
CR (1) | CR20130656A (es) |
DO (1) | DOP2013000298A (es) |
EA (1) | EA023713B1 (es) |
EC (1) | ECSP13013076A (es) |
ES (1) | ES2564882T3 (es) |
MA (1) | MA35269B1 (es) |
MX (1) | MX2013014888A (es) |
PE (1) | PE20140648A1 (es) |
TN (1) | TN2013000439A1 (es) |
WO (1) | WO2012171900A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2980667A1 (en) | 2015-04-09 | 2016-10-13 | Galderma Sa | A pharmaceutical composition and the use thereof |
JP2018510891A (ja) | 2015-04-09 | 2018-04-19 | ガルデルマ・ソシエテ・アノニム | 抗菌性インジゴナチュラリス又はインジゴ産生植物抽出物及びその使用 |
KR20170133497A (ko) | 2015-04-09 | 2017-12-05 | 갈데르마 소시에떼아노님 | 인디고 내추럴리스로부터의 추출물 및 그의 제조 방법 |
Family Cites Families (30)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8828477D0 (en) | 1988-12-06 | 1989-01-05 | Riker Laboratories Inc | Medical aerosol formulations |
EP0407028B2 (en) | 1989-05-31 | 1999-07-07 | FISONS plc | Medicament inhalation device and formulation |
GB8921222D0 (en) | 1989-09-20 | 1989-11-08 | Riker Laboratories Inc | Medicinal aerosol formulations |
IE67185B1 (en) | 1990-02-02 | 1996-03-06 | Fisons Plc | Propellant compositions |
DE4003272A1 (de) | 1990-02-03 | 1991-08-08 | Boehringer Ingelheim Kg | Neue treibgasmischungen und ihre verwendung in arzneimittelzubereitungen |
EP0526481B1 (en) | 1990-03-23 | 1995-04-26 | Minnesota Mining And Manufacturing Company | The use of soluble fluorosurfactants for the preparation of metered-dose aerosol formulations |
EP0553298B1 (en) | 1990-10-18 | 1994-11-17 | Minnesota Mining And Manufacturing Company | Aerosol formulation comprising beclomethasone 17,21 dipropionate |
AU650953B2 (en) | 1991-03-21 | 1994-07-07 | Novartis Ag | Inhaler |
IL104068A (en) | 1991-12-12 | 1998-10-30 | Glaxo Group Ltd | Pharmaceutical preparations in a spray without surfactant containing 1, 1, 1, 2 tetrafluoroethane or 1,1,2,3,3 petafluor N propane as propellant |
GB9213874D0 (en) | 1992-06-30 | 1992-08-12 | Fisons Plc | Process to novel medicament form |
GB9306703D0 (en) | 1993-03-31 | 1993-05-26 | Fisons Plc | Inhalation device |
IL111194A (en) | 1993-10-08 | 1998-02-08 | Fisons Plc | Process for the production of drug patramulations |
AU735934B2 (en) * | 1997-01-15 | 2001-07-19 | Altana Pharma Ag | Phthalazinones |
AU3328499A (en) * | 1998-03-14 | 1999-10-11 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Phthalazinone pde iii/iv inhibitors |
NZ509489A (en) | 1998-08-04 | 2002-10-25 | Jago Res A | Medicinal aerosol formulations comprising cromoglycic acid and/or nedocromil |
US6397838B1 (en) | 1998-12-23 | 2002-06-04 | Battelle Pulmonary Therapeutics, Inc. | Pulmonary aerosol delivery device and method |
JP4530548B2 (ja) | 1999-04-23 | 2010-08-25 | バテル・メモリアル・インスティテュート | 効率がよい物質移動用電気流体力学式エーロゾル噴霧器およびエーロゾルを生成しかつ所望の位置に給送する方法 |
BR0009993A (pt) | 1999-04-23 | 2002-01-08 | Battelle Memorial Institute | Pulverizador de aerossol eletrohidrodinâmico direcionalmente controlado, dispositivo para liberar gotìculas de aerossol eletricamente neutras, aparelho para liberar gotìculas de aerossol terapêuticas, processo para liberar gotìculas de aerossol, e, dispositivo para liberar aerossol |
SK17052002A3 (sk) * | 2000-06-05 | 2003-12-02 | Altana Pharma Ag | Pyridazinónové zlúčeniny, farmaceutický prostriedok s ich obsahom a ich použitie |
PL199420B1 (pl) | 2000-10-09 | 2008-09-30 | 3M Innovative Properties Co | Medyczne preparaty aerozolowe |
NZ527424A (en) * | 2001-02-15 | 2005-02-25 | Altana Pharma Ag | Phthalayinone-piperidino-derivatives as PDE4 inhibitors |
CN1503792A (zh) | 2001-04-25 | 2004-06-09 | ��̹��ҽҩ��˾ | 新的酞嗪酮 |
CA2494650A1 (en) * | 2002-08-10 | 2004-03-04 | Altana Pharma Ag | Pyridazinone-derivatives as pde4 inhibitors |
AU2003260376A1 (en) | 2002-08-10 | 2004-03-11 | Altana Pharma Ag | Piperidine-pyridazones and phthalazones as pde4 inhibitors |
AU2003255376A1 (en) | 2002-08-10 | 2004-03-11 | Altana Pharma Ag | Piperidine-derivatives as pde4 inhibitors |
AU2004204355B2 (en) * | 2003-01-14 | 2009-12-17 | Nycomed Gmbh | PDE4 inhibitors for the treatment of neoplasms of lymphoid cells |
WO2005075456A1 (en) | 2004-02-04 | 2005-08-18 | Altana Pharma Ag | 2-(piperidin-4-yl) -4, 5-dihydro-2h-pyridazin-3-one derivatives as pde4 inhibitors |
EP1720854A1 (en) * | 2004-02-04 | 2006-11-15 | Altana Pharma AG | Phthalzinone derivatives as pde4 inhibitors |
AR070454A1 (es) * | 2008-02-27 | 2010-04-07 | Nycomed Gmbh | Pirrolopirimidincarboxamidas y composiciones farmaceuticas que las comprenden |
AR077898A1 (es) * | 2009-08-26 | 2011-09-28 | Nycomed Gmbh | Metilpirrolopirimidincarboxamidas |
-
2012
- 2012-06-12 KR KR1020147000392A patent/KR20140037195A/ko not_active Application Discontinuation
- 2012-06-12 CA CA2837248A patent/CA2837248A1/en not_active Abandoned
- 2012-06-12 WO PCT/EP2012/061084 patent/WO2012171900A1/en active Application Filing
- 2012-06-12 EP EP12728453.7A patent/EP2721030B1/en active Active
- 2012-06-12 PE PE2013002801A patent/PE20140648A1/es not_active Application Discontinuation
- 2012-06-12 US US14/125,187 patent/US20140112945A1/en not_active Abandoned
- 2012-06-12 AU AU2012269133A patent/AU2012269133A1/en not_active Abandoned
- 2012-06-12 EA EA201400001A patent/EA023713B1/ru not_active IP Right Cessation
- 2012-06-12 BR BR112013031791A patent/BR112013031791A2/pt not_active IP Right Cessation
- 2012-06-12 JP JP2014515155A patent/JP5980318B2/ja not_active Expired - Fee Related
- 2012-06-12 MX MX2013014888A patent/MX2013014888A/es not_active Application Discontinuation
- 2012-06-12 ES ES12728453.7T patent/ES2564882T3/es active Active
- 2012-06-12 AR ARP120102088A patent/AR086915A1/es unknown
- 2012-06-12 CN CN201280028413.XA patent/CN103582644B/zh not_active Expired - Fee Related
-
2013
- 2013-10-29 TN TNP2013000439A patent/TN2013000439A1/fr unknown
- 2013-12-11 CL CL2013003556A patent/CL2013003556A1/es unknown
- 2013-12-11 EC ECSP13013076 patent/ECSP13013076A/es unknown
- 2013-12-11 DO DO2013000298A patent/DOP2013000298A/es unknown
- 2013-12-13 CR CR20130656A patent/CR20130656A/es unknown
-
2014
- 2014-01-10 CO CO14004200A patent/CO6852074A2/es not_active Application Discontinuation
- 2014-01-16 MA MA36689A patent/MA35269B1/fr unknown
-
2015
- 2015-12-03 US US14/958,141 patent/US20160108049A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CA2837248A1 (en) | 2012-12-20 |
JP5980318B2 (ja) | 2016-08-31 |
MX2013014888A (es) | 2014-02-27 |
MA35269B1 (fr) | 2014-07-03 |
AU2012269133A1 (en) | 2014-01-30 |
BR112013031791A2 (pt) | 2017-01-31 |
TN2013000439A1 (en) | 2015-03-30 |
US20160108049A1 (en) | 2016-04-21 |
CR20130656A (es) | 2014-02-18 |
EA023713B1 (ru) | 2016-07-29 |
DOP2013000298A (es) | 2014-03-31 |
CO6852074A2 (es) | 2014-01-30 |
AR086915A1 (es) | 2014-01-29 |
ES2564882T3 (es) | 2016-03-29 |
CN103582644B (zh) | 2016-07-20 |
ECSP13013076A (es) | 2014-01-31 |
EP2721030A1 (en) | 2014-04-23 |
EP2721030B1 (en) | 2015-12-16 |
US20140112945A1 (en) | 2014-04-24 |
EA201400001A1 (ru) | 2014-05-30 |
JP2014517021A (ja) | 2014-07-17 |
WO2012171900A1 (en) | 2012-12-20 |
PE20140648A1 (es) | 2014-05-30 |
KR20140037195A (ko) | 2014-03-26 |
CN103582644A (zh) | 2014-02-12 |
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