CL2008000790A1 - Compuestos derivados de purina sustituida; metodo de sintesis; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como aterosclerosis, artritis, psoriasis y cancer. - Google Patents
Compuestos derivados de purina sustituida; metodo de sintesis; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como aterosclerosis, artritis, psoriasis y cancer.Info
- Publication number
- CL2008000790A1 CL2008000790A1 CL200800790A CL2008000790A CL2008000790A1 CL 2008000790 A1 CL2008000790 A1 CL 2008000790A1 CL 200800790 A CL200800790 A CL 200800790A CL 2008000790 A CL2008000790 A CL 2008000790A CL 2008000790 A1 CL2008000790 A1 CL 2008000790A1
- Authority
- CL
- Chile
- Prior art keywords
- aterosclerosis
- purina
- psoriasis
- arthritis
- cancer
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US91930007P | 2007-03-21 | 2007-03-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2008000790A1 true CL2008000790A1 (es) | 2008-05-30 |
Family
ID=39535224
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL200800790A CL2008000790A1 (es) | 2007-03-21 | 2008-03-19 | Compuestos derivados de purina sustituida; metodo de sintesis; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como aterosclerosis, artritis, psoriasis y cancer. |
Country Status (13)
Country | Link |
---|---|
US (1) | US20080233127A1 (es) |
EP (1) | EP2125815A2 (es) |
JP (1) | JP2010522209A (es) |
CN (1) | CN101730697A (es) |
AR (1) | AR065813A1 (es) |
AU (1) | AU2008228758A1 (es) |
BR (1) | BRPI0809140A2 (es) |
CA (1) | CA2681326A1 (es) |
CL (1) | CL2008000790A1 (es) |
MX (1) | MX2009010067A (es) |
PE (1) | PE20090060A1 (es) |
TW (1) | TW200902531A (es) |
WO (1) | WO2008116129A2 (es) |
Families Citing this family (51)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE448532T1 (de) * | 1996-09-04 | 2009-11-15 | Intertrust Tech Corp | Zuverlässige infrastrukturhilfssysteme, verfahren und techniken für sicheren elektronischen handel, elektronische transaktionen, handelsablaufsteuerung und automatisierung, verteilte verarbeitung und rechteverwaltung |
AU2008282728B2 (en) | 2007-08-02 | 2012-04-19 | Amgen Inc. | Pl3 kinase modulators and methods of use |
CN101889015B (zh) | 2007-10-05 | 2014-06-04 | 维拉斯通股份有限公司 | 嘧啶取代的嘌呤衍生物 |
CA2703138A1 (en) * | 2007-10-26 | 2009-04-30 | F. Hoffmann-La Roche Ag | Purine derivatives useful as pi3 kinase inhibitors |
WO2009085230A1 (en) | 2007-12-19 | 2009-07-09 | Amgen Inc. | Inhibitors of pi3 kinase |
WO2009146406A1 (en) * | 2008-05-30 | 2009-12-03 | Genentech, Inc. | Purine pi3k inhibitor compounds and methods of use |
ES2432821T3 (es) * | 2008-07-31 | 2013-12-05 | Genentech, Inc. | Compuestos de pirimidina, composiciones y métodos de utilización |
TWI378933B (en) | 2008-10-14 | 2012-12-11 | Daiichi Sankyo Co Ltd | Morpholinopurine derivatives |
WO2010103094A1 (en) | 2009-03-13 | 2010-09-16 | Cellzome Limited | PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS |
MX2011010105A (es) | 2009-03-27 | 2012-01-12 | Pathway Therapeutics Inc | Sulfonamidas de pirimidinilo y 1,3,5-triazinilo benzimidazol y su uso en terapia de cancer. |
CA2950529C (en) | 2009-04-03 | 2019-04-30 | Verastem, Inc. | Pyrimidine substituted purine compounds as kinase (s) inhibitors |
US20120071475A1 (en) | 2009-04-27 | 2012-03-22 | Shionogi & Co., Ltd. | Urea derivatives having pi3k-inhibiting activity |
BRPI1009022A2 (pt) * | 2009-05-27 | 2016-03-08 | Hoffmann La Roche | "composto, composição farmacêutica, processo para produzir uma composição farmacêutica, uso de um composto, método para tratamento de uma doença ou transtorno e kit" |
US20100331305A1 (en) * | 2009-06-24 | 2010-12-30 | Genentech, Inc. | Oxo-heterocycle fused pyrimidine compounds, compositions and methods of use |
CA2766100C (en) | 2009-06-29 | 2018-05-22 | Incyte Corporation | Pyrimidinones as pi3k inhibitors |
AR080945A1 (es) | 2009-07-07 | 2012-05-23 | Pathway Therapeutics Inc | Pirimidinil y 1,3,5-triazinil benzimidazoles y su uso en la terapia contra el cancer |
CA2780018C (en) * | 2009-11-12 | 2015-10-20 | F. Hoffmann-La Roche Ag | N-7 substituted purine and pyrazolopyrimidine compounds, compositions and methods of use |
US8288381B2 (en) * | 2009-11-12 | 2012-10-16 | Genentech, Inc. | N-9 substituted purine compounds, compositions and methods of use |
WO2011075643A1 (en) | 2009-12-18 | 2011-06-23 | Incyte Corporation | Substituted heteroaryl fused derivatives as pi3k inhibitors |
EP2542536B1 (en) | 2010-03-04 | 2015-01-21 | Cellzome Limited | Morpholino substituted urea derivatives as mtor inhibitors |
EP2558463A1 (en) | 2010-04-14 | 2013-02-20 | Incyte Corporation | Fused derivatives as i3 inhibitors |
US9062055B2 (en) | 2010-06-21 | 2015-06-23 | Incyte Corporation | Fused pyrrole derivatives as PI3K inhibitors |
WO2012007493A1 (en) * | 2010-07-14 | 2012-01-19 | F. Hoffmann-La Roche Ag | Purine compounds selective for ρi3κ p110 delta, and methods of use |
JP5954838B2 (ja) * | 2010-09-14 | 2016-07-20 | エクセリクシス, インク. | Pi3k−デルタの阻害剤ならびにそれらの使用法および製造法 |
SI2651951T1 (sl) | 2010-12-16 | 2015-01-30 | F. Hoffmann-La Roche Ag | Tricikliäśne p13k inhibitorske spojine in postopki uporabe |
TW201249844A (en) | 2010-12-20 | 2012-12-16 | Incyte Corp | N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors |
WO2012125629A1 (en) | 2011-03-14 | 2012-09-20 | Incyte Corporation | Substituted diamino-pyrimidine and diamino-pyridine derivatives as pi3k inhibitors |
WO2012135009A1 (en) | 2011-03-25 | 2012-10-04 | Incyte Corporation | Pyrimidine-4,6-diamine derivatives as pi3k inhibitors |
BR112013024907A2 (pt) | 2011-03-28 | 2016-12-20 | Mei Pharma Inc | composto, composição farmacêutica, método para o tratamento, prevenção ou atenuação de um ou mais sintomas de um distúrbio, doença ou condição mediada por pi3k em um sujeito, método para modular a atividade enzimática de pi3k |
JP2014510122A (ja) | 2011-04-04 | 2014-04-24 | セルゾーム リミテッド | mTOR阻害剤としてのジヒドロピロロピリミジン誘導体 |
IL299533A (en) | 2011-09-02 | 2023-02-01 | Incyte Holdings Corp | Heterocycloamines as P13K inhibitors |
CN103917530B (zh) | 2011-09-21 | 2016-08-24 | 塞尔佐姆有限公司 | 作为mtor抑制剂的吗啉代取代的脲或氨基甲酸衍生物 |
CN103946222B (zh) | 2011-10-07 | 2016-12-28 | 塞尔佐姆有限公司 | 作为mtor抑制剂的吗啉代取代的双环嘧啶脲或氨基甲酸衍生物 |
WO2013095761A1 (en) * | 2011-12-20 | 2013-06-27 | Glaxosmithkline Llc | Imidazopyridine derivatives as pi3 kinase inhibitors |
AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
EP2852661A1 (en) | 2012-05-23 | 2015-04-01 | F. Hoffmann-La Roche AG | Compositions and methods of obtaining and using endoderm and hepatocyte cells |
CN103588792B (zh) * | 2013-03-04 | 2016-03-23 | 中国科学院上海药物研究所 | 吡啶并嘧啶或嘧啶并嘧啶类化合物、其制备方法、药物组合物及其用途 |
US10077277B2 (en) | 2014-06-11 | 2018-09-18 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors |
HUE060953T2 (hu) | 2015-02-27 | 2023-04-28 | Incyte Holdings Corp | Eljárások PI3K inhibitor elõállítására |
BR112017020818A2 (pt) | 2015-03-30 | 2018-07-03 | Daiichi Sankyo Company, Limited | composto, uso de um composto, método, e, medicamento |
EA033106B1 (ru) * | 2015-04-21 | 2019-08-30 | Гуйчжоу Бэйлинг Груп Фармасьютикал Ко., Лтд. | Производное пуринил-n-гидроксипиримидинформамида, способы его получения и его применения |
WO2016183060A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
WO2016183063A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Crystalline forms of a pi3k inhibitor |
JP7068186B2 (ja) | 2016-12-02 | 2022-05-16 | 第一三共株式会社 | 新規エンド-β-N-アセチルグルコサミニダーゼ |
KR20200009088A (ko) | 2017-05-23 | 2020-01-29 | 메이 파마, 아이엔씨. | 병용 요법 |
WO2019018562A1 (en) | 2017-07-19 | 2019-01-24 | Ideaya Biosciences, Inc. | AMIDO COMPOUND AS MODULATORS OF AHR |
JP2020531414A (ja) | 2017-08-14 | 2020-11-05 | エムイーアイ ファーマ,インク. | 併用療法 |
CN112707907B (zh) * | 2019-10-24 | 2023-05-23 | 张飞 | 嘌呤衍生物及其中间体与制备抗癌症药物的应用 |
CN111875606B (zh) * | 2020-07-20 | 2023-04-07 | 武汉工程大学 | 一种基于虚拟对接获得的嘌呤类化合物及其制备方法和应用 |
CN113116895B (zh) * | 2020-12-31 | 2023-08-18 | 天津医科大学肿瘤医院 | 用于治疗神经母细胞瘤的喹啉衍生物 |
CN117503743B (zh) * | 2023-12-08 | 2024-04-16 | 南京鼓楼医院 | 一种nlrp3炎症小体抑制剂及其在制备预防或治疗细胞焦亡的药物中的应用 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS60260579A (ja) * | 1984-01-13 | 1985-12-23 | Yoshitomi Pharmaceut Ind Ltd | プリン誘導体 |
JPS6210085A (ja) * | 1985-07-05 | 1987-01-19 | Yoshitomi Pharmaceut Ind Ltd | トリフルオロメチルプリン誘導体 |
DE60144322D1 (de) * | 2000-04-27 | 2011-05-12 | Astellas Pharma Inc | Kondensierte heteroarylderivate |
EP1626725A4 (en) * | 2003-05-29 | 2006-06-14 | Synta Pharmaceuticals Corp | Heterocyclic compounds for the prevention and treatment of disorders associated with excessive bone formation |
FR2880626B1 (fr) * | 2005-01-13 | 2008-04-18 | Aventis Pharma Sa | Derives de la purine, compositions les contenant et utilisation |
GB2431156A (en) * | 2005-10-11 | 2007-04-18 | Piramed Ltd | 1-cyclyl-3-substituted- -benzenes and -azines as inhibitors of phosphatidylinositol 3-kinase |
-
2008
- 2008-03-07 US US12/044,500 patent/US20080233127A1/en not_active Abandoned
- 2008-03-19 PE PE2008000503A patent/PE20090060A1/es not_active Application Discontinuation
- 2008-03-19 CL CL200800790A patent/CL2008000790A1/es unknown
- 2008-03-19 AR ARP080101182A patent/AR065813A1/es unknown
- 2008-03-21 AU AU2008228758A patent/AU2008228758A1/en not_active Abandoned
- 2008-03-21 MX MX2009010067A patent/MX2009010067A/es unknown
- 2008-03-21 WO PCT/US2008/057771 patent/WO2008116129A2/en active Application Filing
- 2008-03-21 CA CA002681326A patent/CA2681326A1/en not_active Abandoned
- 2008-03-21 EP EP08744161A patent/EP2125815A2/en not_active Withdrawn
- 2008-03-21 TW TW097110236A patent/TW200902531A/zh unknown
- 2008-03-21 JP JP2009554756A patent/JP2010522209A/ja not_active Withdrawn
- 2008-03-21 CN CN200880009067A patent/CN101730697A/zh active Pending
- 2008-03-21 BR BRPI0809140-4A patent/BRPI0809140A2/pt not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CA2681326A1 (en) | 2008-09-25 |
WO2008116129A3 (en) | 2009-02-12 |
MX2009010067A (es) | 2009-10-12 |
US20080233127A1 (en) | 2008-09-25 |
BRPI0809140A2 (pt) | 2014-08-26 |
PE20090060A1 (es) | 2009-01-18 |
TW200902531A (en) | 2009-01-16 |
AR065813A1 (es) | 2009-07-01 |
JP2010522209A (ja) | 2010-07-01 |
CN101730697A (zh) | 2010-06-09 |
AU2008228758A1 (en) | 2008-09-25 |
EP2125815A2 (en) | 2009-12-02 |
WO2008116129A2 (en) | 2008-09-25 |
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