CL2007001937A1 - Compuestos derivados de bencilsulfanilpiridina, inhibidores del receptor p2y12; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar un trastorno de agregacion plaquetaria. - Google Patents

Compuestos derivados de bencilsulfanilpiridina, inhibidores del receptor p2y12; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar un trastorno de agregacion plaquetaria.

Info

Publication number
CL2007001937A1
CL2007001937A1 CL200701937A CL2007001937A CL2007001937A1 CL 2007001937 A1 CL2007001937 A1 CL 2007001937A1 CL 200701937 A CL200701937 A CL 200701937A CL 2007001937 A CL2007001937 A CL 2007001937A CL 2007001937 A1 CL2007001937 A1 CL 2007001937A1
Authority
CL
Chile
Prior art keywords
compounds
plaquetary
bencilsulfanilpiridina
agregation
disorder
Prior art date
Application number
CL200701937A
Other languages
English (en)
Inventor
Antonsson Bach Peter Br Thomas
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38894825&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2007001937(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of CL2007001937A1 publication Critical patent/CL2007001937A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/455Nicotinic acids, e.g. niacin; Derivatives thereof, e.g. esters, amides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/04Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/08Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
CL200701937A 2006-07-04 2007-07-03 Compuestos derivados de bencilsulfanilpiridina, inhibidores del receptor p2y12; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar un trastorno de agregacion plaquetaria. CL2007001937A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE0601463 2006-07-04
SE0602091 2006-10-04
SE0700059 2007-01-12

Publications (1)

Publication Number Publication Date
CL2007001937A1 true CL2007001937A1 (es) 2008-07-25

Family

ID=38894825

Family Applications (1)

Application Number Title Priority Date Filing Date
CL200701937A CL2007001937A1 (es) 2006-07-04 2007-07-03 Compuestos derivados de bencilsulfanilpiridina, inhibidores del receptor p2y12; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar un trastorno de agregacion plaquetaria.

Country Status (16)

Country Link
US (2) US20080039437A1 (es)
EP (1) EP2044050A1 (es)
JP (1) JP2009542644A (es)
KR (1) KR20090034935A (es)
AR (1) AR061805A1 (es)
AU (1) AU2007270086A1 (es)
BR (1) BRPI0713967A2 (es)
CA (1) CA2655633A1 (es)
CL (1) CL2007001937A1 (es)
EC (1) ECSP099040A (es)
IL (1) IL195982A0 (es)
MX (1) MX2008016548A (es)
NO (1) NO20085215L (es)
TW (1) TW200811133A (es)
UY (1) UY30457A1 (es)
WO (1) WO2008004946A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2008016551A (es) * 2006-07-04 2009-02-06 Astrazeneca Ab Analogos de piridina nuevos.
TW200902513A (en) * 2007-07-13 2009-01-16 Astrazeneca Ab New pyridine analogues
WO2010005384A1 (en) * 2008-07-07 2010-01-14 Astrazeneca Ab Ketone pyridine analogues and their use in the treatment of cardiovascular disorders
WO2013033178A1 (en) 2011-08-30 2013-03-07 University Of Utah Research Foundation Methods and compositions for treating nephrogenic diabetes insipidus

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6156758A (en) * 1999-09-08 2000-12-05 Isis Pharmaceuticals, Inc. Antibacterial quinazoline compounds
DE60114994T2 (de) * 2000-02-04 2006-08-03 Portola Pharmaceuticals, Inc., South San Francisco Blutplättchen-adp-rezeptor-inhibitoren
US6906063B2 (en) * 2000-02-04 2005-06-14 Portola Pharmaceuticals, Inc. Platelet ADP receptor inhibitors
US7132408B2 (en) * 2000-08-21 2006-11-07 Inspire Pharmaceuticals, Inc. Composition and method for inhibiting platelet aggregation
US7018985B1 (en) * 2000-08-21 2006-03-28 Inspire Pharmaceuticals, Inc. Composition and method for inhibiting platelet aggregation
US7452870B2 (en) * 2000-08-21 2008-11-18 Inspire Pharmaceuticals, Inc. Drug-eluting stents coated with P2Y12 receptor antagonist compound
FR2820057A1 (fr) * 2001-01-30 2002-08-02 Ct De Transfert De Technologie Membrane pour chambre d'encapsulation de cellules produisant au moins une substance biologiquement active et organe bio-artificiel comprenant une telle membrane
CN1867560A (zh) * 2003-08-13 2006-11-22 武田药品工株式会社 4-嘧啶酮衍生物及其作为肽基肽酶抑制剂的用途
CN1863789B (zh) * 2003-10-03 2010-06-09 博尔托拉制药公司 取代的异喹啉酮
US7335648B2 (en) * 2003-10-21 2008-02-26 Inspire Pharmaceuticals, Inc. Non-nucleotide composition and method for inhibiting platelet aggregation
US7749981B2 (en) * 2003-10-21 2010-07-06 Inspire Pharmaceuticals, Inc. Drug-eluting stents coated with non-nucleotide P2Y12 receptor antagonist compound
US7504497B2 (en) * 2003-10-21 2009-03-17 Inspire Pharmaceuticals, Inc. Orally bioavailable compounds and methods for inhibiting platelet aggregation
US8071624B2 (en) * 2004-06-24 2011-12-06 Incyte Corporation N-substituted piperidines and their use as pharmaceuticals
AU2006204159A1 (en) * 2005-01-06 2006-07-13 Astrazeneca Ab Novel pyridine compounds
BRPI0713400A2 (pt) * 2006-07-04 2012-04-17 Astrazeneca Ab composto, composição farmacêutica, uso de um composto, e, método de tratamento de um distúrbio de agregação plaquetária
MX2008016551A (es) * 2006-07-04 2009-02-06 Astrazeneca Ab Analogos de piridina nuevos.
BRPI0713957A2 (pt) * 2006-07-04 2013-04-02 Astrazeneca Ab composto, composiÇço farmacÊutica, uso de um composto, e, mÉtodo de tratamento de um distérbio de agregaÇço plaquetÁria

Also Published As

Publication number Publication date
CA2655633A1 (en) 2008-01-10
TW200811133A (en) 2008-03-01
EP2044050A1 (en) 2009-04-08
US20080039437A1 (en) 2008-02-14
ECSP099040A (es) 2009-02-27
JP2009542644A (ja) 2009-12-03
NO20085215L (no) 2009-01-13
US20100069350A1 (en) 2010-03-18
KR20090034935A (ko) 2009-04-08
AR061805A1 (es) 2008-09-24
MX2008016548A (es) 2009-02-12
BRPI0713967A2 (pt) 2012-11-27
IL195982A0 (en) 2009-09-01
WO2008004946A1 (en) 2008-01-10
UY30457A1 (es) 2008-02-29
AU2007270086A1 (en) 2008-01-10

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