CH627184A5 - Process for the preparation of antibacterial agents - Google Patents

Process for the preparation of antibacterial agents Download PDF

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Publication number
CH627184A5
CH627184A5 CH1249577A CH1249577A CH627184A5 CH 627184 A5 CH627184 A5 CH 627184A5 CH 1249577 A CH1249577 A CH 1249577A CH 1249577 A CH1249577 A CH 1249577A CH 627184 A5 CH627184 A5 CH 627184A5
Authority
CH
Switzerland
Prior art keywords
compound
formula
group
acid
mixture
Prior art date
Application number
CH1249577A
Other languages
English (en)
French (fr)
Inventor
Takayuki Naito
Jun Okumura
Hajime Kamachi
Seiji Iimura
Hideaki Hoshi
Masahisa Oka
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/784,885 external-priority patent/US4082912A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of CH627184A5 publication Critical patent/CH627184A5/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/24Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/24Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CH1249577A 1977-04-05 1977-10-13 Process for the preparation of antibacterial agents CH627184A5 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/784,885 US4082912A (en) 1976-06-30 1977-04-05 Certain 7-acylamido-3-(2-carboxyalkyl-2,3-dihydro-s-triazolo[4,3-b]pyridazin-3-on-6-ylmethyl)-3-cephem-4-carboxylic acids their salts and easily hydrolyzed esters

Publications (1)

Publication Number Publication Date
CH627184A5 true CH627184A5 (en) 1981-12-31

Family

ID=25133827

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1249577A CH627184A5 (en) 1977-04-05 1977-10-13 Process for the preparation of antibacterial agents

Country Status (17)

Country Link
JP (1) JPS53124290A (fi)
AU (1) AU517919B2 (fi)
BE (1) BE859774A (fi)
CA (1) CA1113455A (fi)
CH (1) CH627184A5 (fi)
DE (1) DE2807847A1 (fi)
DK (1) DK145497C (fi)
FI (1) FI60869C (fi)
FR (1) FR2408614A1 (fi)
GB (1) GB1572201A (fi)
GR (1) GR73550B (fi)
IE (1) IE45613B1 (fi)
LU (1) LU78323A1 (fi)
NL (1) NL7711644A (fi)
SE (1) SE425491B (fi)
YU (1) YU247977A (fi)
ZA (1) ZA775781B (fi)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3000377A1 (de) * 1980-01-07 1981-07-09 Boehringer Mannheim Gmbh, 6800 Mannheim Neue sulfonamide, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
CN114940665B (zh) * 2022-06-10 2024-05-07 河南省科学院高新技术研究中心 一种用作杀菌剂的苯并异噻唑啉酮类化合物及其制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3907786A (en) * 1973-09-04 1975-09-23 Bristol Myers Co 7-{8 {60 -(2-aminomethyl-1,4-cyclohexadienyl)acetamido{9 -3-heterocyclic-thiomethyl-3-cephem-4-carboxylic acids and salts
US3946000A (en) * 1973-10-31 1976-03-23 Bristol-Myers Company 7-[α-(2-Aminomethyl-1-cyclohexenyl)-acetamido]-3-heterocyclic thiomethyl-3-cephem-4-carboxylic acids

Also Published As

Publication number Publication date
NL7711644A (nl) 1978-10-09
FI60869B (fi) 1981-12-31
SE7710823L (sv) 1978-10-06
CA1113455A (en) 1981-12-01
ZA775781B (en) 1978-08-30
FI772860A (fi) 1978-10-06
IE45613B1 (en) 1982-10-06
BE859774A (fr) 1978-04-14
FR2408614B1 (fi) 1980-12-05
GB1572201A (en) 1980-07-23
JPS53124290A (en) 1978-10-30
DK429577A (da) 1978-10-06
FR2408614A1 (fr) 1979-06-08
DK145497C (da) 1983-05-02
AU2932877A (en) 1979-04-12
GR73550B (fi) 1984-03-13
LU78323A1 (fi) 1978-06-12
SE425491B (sv) 1982-10-04
DK145497B (da) 1982-11-29
IE45613L (en) 1978-10-05
DE2807847A1 (de) 1978-10-19
YU247977A (en) 1982-10-31
AU517919B2 (en) 1981-09-03
FI60869C (fi) 1982-04-13

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