CH626074A5 - - Google Patents

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Publication number
CH626074A5
CH626074A5 CH752880A CH752880A CH626074A5 CH 626074 A5 CH626074 A5 CH 626074A5 CH 752880 A CH752880 A CH 752880A CH 752880 A CH752880 A CH 752880A CH 626074 A5 CH626074 A5 CH 626074A5
Authority
CH
Switzerland
Prior art keywords
derivatives
reaction
general formula
acid ester
group
Prior art date
Application number
CH752880A
Other languages
German (de)
English (en)
Inventor
Gabor Dr Bernath
Lajos Dr Gera
Gyoergy Goendoes
Judit Dr Hermann-Voeroes
Matyas Dr Szentivanyi
Zoltan Ecsery
Erzsebet Janvari-Kanyo
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of CH626074A5 publication Critical patent/CH626074A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/91Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/90Oxygen atoms with acyclic radicals attached in position 2 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH752880A 1975-10-03 1980-10-08 CH626074A5 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU75CI00001614A HU172460B (hu) 1975-10-03 1975-10-03 Sposob poluchenija novykh proizvodnykh 5,6-digidro-3h-pirimidin-4-ona

Publications (1)

Publication Number Publication Date
CH626074A5 true CH626074A5 (fr) 1981-10-30

Family

ID=10994582

Family Applications (2)

Application Number Title Priority Date Filing Date
CH1248376A CH626072A5 (fr) 1975-10-03 1976-10-01
CH752880A CH626074A5 (fr) 1975-10-03 1980-10-08

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CH1248376A CH626072A5 (fr) 1975-10-03 1976-10-01

Country Status (14)

Country Link
US (1) US4113868A (fr)
JP (1) JPS5257185A (fr)
AU (1) AU507798B2 (fr)
CH (2) CH626072A5 (fr)
CS (1) CS193563B2 (fr)
DD (1) DD127444A1 (fr)
DE (1) DE2643384A1 (fr)
FI (1) FI66603C (fr)
FR (1) FR2326193A1 (fr)
GB (1) GB1559985A (fr)
HU (1) HU172460B (fr)
IL (1) IL50577A (fr)
PL (2) PL110639B1 (fr)
SU (1) SU627752A3 (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU179687B (en) * 1978-11-01 1982-11-29 Chinoin Gyogyszer Es Vegyeszet Process for producing 5,6,7,8-- etrahydro-4-bracket-3h-bracket closed-quinasolinones
US4814335A (en) * 1982-12-30 1989-03-21 Biomeasure, Incorporated Antiviral compounds
JPS59210071A (ja) * 1982-12-30 1984-11-28 バイオメジヤ−・インコ−ポレ−テツド 抗ウイルス作用を有する化合物
US5629264A (en) * 1995-03-23 1997-05-13 Rohm And Haas Company 2-aryl-5,6-dihydropyrimidinones and herbicidal use thereof
AU2004200A (en) * 1999-01-14 2000-08-01 Meiji Seika Kaisha Ltd. Poly(adp-ribose) polymerase inhibitors consisting of pyrimidine derivatives
DE10123163A1 (de) * 2001-05-09 2003-01-16 Gruenenthal Gmbh Substituierte Cyclohexan-1,4-diaminderivate
AUPS019702A0 (en) * 2002-01-29 2002-02-21 Fujisawa Pharmaceutical Co., Ltd. Condensed heterocyclic compounds

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3047462A (en) * 1959-03-06 1962-07-31 Lab Jacques Logeais Soc D Expl Quinazolone anti-inflammatory composition
GB1233943A (fr) * 1968-10-31 1971-06-03
US3696102A (en) * 1970-03-09 1972-10-03 Pfizer & Co C Process for the synthesis of substituted quinazolin-4-ones
US3996227A (en) * 1971-07-08 1976-12-07 Sandoz, Inc. 7-Methyl-1-isopropyl-4-phenyl-5,6,7,8-tetrahydro-2(1H)-quinazolinone
US3945960A (en) * 1973-07-26 1976-03-23 Sandoz, Inc. Antiinflammatory and analgesic cycloalkano-pyrimidin-2(1H)-ones
US3994894A (en) * 1975-01-08 1976-11-30 Sandoz, Inc. Cyclopentano[1,2-c]pyrimidin-2(1H)-ones

Also Published As

Publication number Publication date
FI762806A (fr) 1977-04-04
PL111251B1 (en) 1980-08-30
GB1559985A (en) 1980-01-30
SU627752A3 (ru) 1978-10-05
FR2326193B1 (fr) 1979-09-28
US4113868A (en) 1978-09-12
FR2326193A1 (fr) 1977-04-29
PL110639B1 (en) 1980-07-31
AU507798B2 (en) 1980-02-28
JPS5257185A (en) 1977-05-11
HU172460B (hu) 1978-09-28
IL50577A (en) 1979-12-30
AU1820376A (en) 1978-04-06
DD127444A1 (fr) 1977-09-21
FI66603B (fi) 1984-07-31
DE2643384A1 (de) 1977-06-02
CS193563B2 (en) 1979-10-31
IL50577A0 (en) 1976-11-30
FI66603C (fi) 1984-11-12
CH626072A5 (fr) 1981-10-30

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Legal Events

Date Code Title Description
PL Patent ceased