CH624933A5 - - Google Patents

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Publication number
CH624933A5
CH624933A5 CH959477A CH959477A CH624933A5 CH 624933 A5 CH624933 A5 CH 624933A5 CH 959477 A CH959477 A CH 959477A CH 959477 A CH959477 A CH 959477A CH 624933 A5 CH624933 A5 CH 624933A5
Authority
CH
Switzerland
Prior art keywords
formula
carbon atoms
radical
pyrrolidine
proline
Prior art date
Application number
CH959477A
Other languages
English (en)
French (fr)
Inventor
Jean-Pierre Kaplan
Henry Najer
Daniel Charles Leon Obitz
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR7623910A external-priority patent/FR2360572A1/fr
Priority claimed from FR7635476A external-priority patent/FR2372157A1/fr
Priority claimed from FR7719391A external-priority patent/FR2395261A2/fr
Application filed by Synthelabo filed Critical Synthelabo
Publication of CH624933A5 publication Critical patent/CH624933A5/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24Oxygen or sulfur atoms
    • C07D207/262-Pyrrolidones
    • C07D207/2732-Pyrrolidones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
    • C07D207/277Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D207/282-Pyrrolidone-5- carboxylic acids; Functional derivatives thereof, e.g. esters, nitriles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH959477A 1976-08-05 1977-08-04 CH624933A5 (xx)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR7623910A FR2360572A1 (fr) 1976-08-05 1976-08-05 Pyrrolidines substituees et leur preparation
FR7635476A FR2372157A1 (fr) 1976-11-25 1976-11-25 Procede de synthese stereospecifique de n-alkyl- pyrrolidines optiquement actives
FR7719391A FR2395261A2 (fr) 1977-06-24 1977-06-24 Pyrrolidines substituees et leur preparation

Publications (1)

Publication Number Publication Date
CH624933A5 true CH624933A5 (xx) 1981-08-31

Family

ID=27250658

Family Applications (2)

Application Number Title Priority Date Filing Date
CH959477A CH624933A5 (xx) 1976-08-05 1977-08-04
CH4181A CH626341A5 (en) 1976-08-05 1981-01-06 Process for the stereospecific synthesis of N-substituted pyrrolidines and their use

Family Applications After (1)

Application Number Title Priority Date Filing Date
CH4181A CH626341A5 (en) 1976-08-05 1981-01-06 Process for the stereospecific synthesis of N-substituted pyrrolidines and their use

Country Status (20)

Country Link
JP (1) JPS5325563A (xx)
AT (1) AT364818B (xx)
AU (1) AU510454B2 (xx)
CA (1) CA1083586A (xx)
CH (2) CH624933A5 (xx)
DE (1) DE2735036C2 (xx)
DK (1) DK350377A (xx)
ES (1) ES461342A1 (xx)
FI (1) FI772363A (xx)
GB (1) GB1555890A (xx)
GR (1) GR63594B (xx)
IE (1) IE45544B1 (xx)
IL (1) IL52645A (xx)
IT (1) IT1085696B (xx)
LU (1) LU77917A1 (xx)
NL (1) NL7708571A (xx)
NO (2) NO772745L (xx)
NZ (1) NZ184832A (xx)
PT (1) PT66894B (xx)
SE (2) SE7708902L (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1095415B (it) * 1978-02-16 1985-08-10 Ravizza Spa Processo per la produzione di una benzamide otticamente attiva,benzamide otticamente attiva cosi'ottenuta e composizioni
IT1141095B (it) * 1980-11-27 1986-10-01 Ravizza Spa Processo di risoluzione della sulpiride racema
SE8602339D0 (sv) * 1986-05-22 1986-05-22 Astra Laekemedel Ab An efficient stereoconservative synthesis of 1-substituted (s)- and (r)-2-aminomethylpyrrolidines
DE4425070A1 (de) * 1994-07-15 1996-01-18 Degussa Verfahren zur Herstellung optisch aktiver l-substituierter 2-(Aminomethyl)pyrrolidine
US7531673B2 (en) * 2004-02-18 2009-05-12 Dr. Reddy's Laboratories Limited Preparation of amino acid amides
CN104086475B (zh) * 2014-07-15 2016-10-05 苏州天马精细化学品股份有限公司 一种n-苄氧羰基-l-脯氨酰胺的制备方法
CN106045869A (zh) * 2016-06-30 2016-10-26 宜兴市前成生物有限公司 一种制备dl‑谷氨酸的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1528014A (fr) * 1967-04-24 1968-06-07 Ile De France Procédé de préparation des isomères optiques de la éthyl-1, aminométhyl-2-pyrrolidine
CH507938A (fr) * 1968-08-01 1971-05-31 Ile De France Procédé de préparation de benzamides hétérocycliques

Also Published As

Publication number Publication date
ATA577377A (de) 1981-04-15
NO772745L (no) 1978-02-07
GR63594B (en) 1979-11-26
ES461342A1 (es) 1978-06-01
FI772363A (xx) 1978-02-06
DE2735036A1 (de) 1978-02-16
PT66894B (fr) 1979-01-26
CA1083586A (en) 1980-08-12
DE2735036C2 (de) 1983-10-13
SE7708902L (sv) 1978-02-06
IE45544B1 (en) 1982-09-22
AU2764177A (en) 1979-02-08
LU77917A1 (xx) 1977-11-14
PT66894A (fr) 1977-09-01
IL52645A0 (en) 1977-10-31
NL7708571A (nl) 1978-02-07
GB1555890A (en) 1979-11-14
JPS5325563A (en) 1978-03-09
IT1085696B (it) 1985-05-28
SE8009074L (sv) 1980-12-22
DK350377A (da) 1978-02-06
IL52645A (en) 1980-02-29
NO812871L (no) 1978-02-07
NZ184832A (en) 1979-11-01
AT364818B (de) 1981-11-25
IE45544L (en) 1978-02-05
CH626341A5 (en) 1981-11-13
AU510454B2 (en) 1980-06-26

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Date Code Title Description
PL Patent ceased