CH584206A5 - - Google Patents

Info

Publication number
CH584206A5
CH584206A5 CH1435775A CH1435775A CH584206A5 CH 584206 A5 CH584206 A5 CH 584206A5 CH 1435775 A CH1435775 A CH 1435775A CH 1435775 A CH1435775 A CH 1435775A CH 584206 A5 CH584206 A5 CH 584206A5
Authority
CH
Switzerland
Application number
CH1435775A
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of CH584206A5 publication Critical patent/CH584206A5/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/116Heterocyclic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Polymers & Plastics (AREA)
  • Food Science & Technology (AREA)
  • Zoology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Anesthesiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Animal Husbandry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH1435775A 1971-08-04 1972-07-28 CH584206A5 (enrdf_load_stackoverflow)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US16909171A 1971-08-04 1971-08-04

Publications (1)

Publication Number Publication Date
CH584206A5 true CH584206A5 (enrdf_load_stackoverflow) 1977-01-31

Family

ID=22614230

Family Applications (3)

Application Number Title Priority Date Filing Date
CH1435675A CH591488A5 (enrdf_load_stackoverflow) 1971-08-04 1972-07-28
CH1435775A CH584206A5 (enrdf_load_stackoverflow) 1971-08-04 1972-07-28
CH1130272A CH574444A5 (enrdf_load_stackoverflow) 1971-08-04 1972-07-28

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CH1435675A CH591488A5 (enrdf_load_stackoverflow) 1971-08-04 1972-07-28

Family Applications After (1)

Application Number Title Priority Date Filing Date
CH1130272A CH574444A5 (enrdf_load_stackoverflow) 1971-08-04 1972-07-28

Country Status (8)

Country Link
JP (3) JPS5714351B1 (enrdf_load_stackoverflow)
AU (1) AU461139B2 (enrdf_load_stackoverflow)
BE (1) BE787251A (enrdf_load_stackoverflow)
CH (3) CH591488A5 (enrdf_load_stackoverflow)
DE (1) DE2237592C2 (enrdf_load_stackoverflow)
FR (1) FR2150732B1 (enrdf_load_stackoverflow)
GB (4) GB1389437A (enrdf_load_stackoverflow)
ZA (1) ZA724880B (enrdf_load_stackoverflow)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3917627A (en) * 1971-08-04 1975-11-04 Upjohn Co 6-Substituted 4H-imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines and process for their production
FR2183716A1 (en) * 1972-05-05 1973-12-21 Centre Etd Ind Pharma Substd-6-phenyl-4h-imidazo (1,2-a)-1,4-benzo diazepines - - tranquillisers anxiolytics,sedatives and muscle-relaxants
ZA755418B (en) * 1974-09-11 1977-06-29 Hoffmann La Roche Diazepine derivatives
US3910946A (en) * 1974-09-12 1975-10-07 Upjohn Co 4H-Imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines
CA1060892A (en) * 1974-11-06 1979-08-21 Parke, Davis And Company Diazepine compounds and method for their production
AT361486B (de) * 1975-08-07 1981-03-10 Hoffmann La Roche Verfahren zur herstellung von neuen imidazo(1,5 -a) (1,4)diazepinverbindungen, ihren salzen und optisch aktiven formen
US4118386A (en) * 1977-04-04 1978-10-03 Hoffmann-La Roche Inc. Synthesis of imidazo[1,5-a]diazepine-3-carboxylates
AU6909194A (en) * 1993-05-14 1994-12-12 Board Of Regents, The University Of Texas System Preparation of n-cyanodithioimino-carbonates and 3-mercapto-5-amino-1h-1,2,4-triazole
WO1996023790A1 (de) * 1995-02-02 1996-08-08 F. Hoffmann-La Roche Ag Acetylimidazobenzodiazepine
JP6715830B2 (ja) 2014-06-26 2020-07-01 ザ・ジョンズ・ホプキンス・ユニバーシティ 過敏性腸症候群および末梢神経系の他の病気の治療のための末梢限局性gabaポジティブアロステリックモジュレーター
WO2018083051A1 (en) * 2016-11-01 2018-05-11 F. Hoffmann-La Roche Ag 1,3-dihydro-1,4-benzodiazepine-2-thiones for the treatment of cns related diseases
CN113717176B (zh) * 2021-10-09 2022-07-05 上海再启生物技术有限公司 一种制备瑞马唑仑的方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3987052A (en) * 1969-03-17 1976-10-19 The Upjohn Company 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines

Also Published As

Publication number Publication date
AU461139B2 (en) 1975-05-15
GB1389434A (en) 1975-04-03
GB1389436A (en) 1975-04-03
FR2150732A1 (enrdf_load_stackoverflow) 1973-04-13
JPS5547686A (en) 1980-04-04
CH591488A5 (enrdf_load_stackoverflow) 1977-09-30
BE787251A (fr) 1973-02-05
ZA724880B (en) 1973-06-27
FR2150732B1 (enrdf_load_stackoverflow) 1976-04-16
GB1389435A (en) 1975-04-03
DE2237592A1 (de) 1973-02-15
DE2237592C2 (de) 1985-08-14
AU4467372A (en) 1974-01-24
JPS5734277B2 (enrdf_load_stackoverflow) 1982-07-22
JPS5714351B1 (enrdf_load_stackoverflow) 1982-03-24
GB1389437A (en) 1975-04-03
JPS5726667A (en) 1982-02-12
CH574444A5 (enrdf_load_stackoverflow) 1976-04-15
JPS5732066B2 (enrdf_load_stackoverflow) 1982-07-08

Similar Documents

Publication Publication Date Title
FR2150732B1 (enrdf_load_stackoverflow)
AU2691671A (enrdf_load_stackoverflow)
AU2684071A (enrdf_load_stackoverflow)
AU2726271A (enrdf_load_stackoverflow)
AU2742671A (enrdf_load_stackoverflow)
AU2894671A (enrdf_load_stackoverflow)
AU2941471A (enrdf_load_stackoverflow)
AU2952271A (enrdf_load_stackoverflow)
AU3005371A (enrdf_load_stackoverflow)
AU2875571A (enrdf_load_stackoverflow)
AU2907471A (enrdf_load_stackoverflow)
AU2684171A (enrdf_load_stackoverflow)
AU2706571A (enrdf_load_stackoverflow)
AU2724971A (enrdf_load_stackoverflow)
AU2740271A (enrdf_load_stackoverflow)
AU2755871A (enrdf_load_stackoverflow)
AU2836771A (enrdf_load_stackoverflow)
AU2837671A (enrdf_load_stackoverflow)
AU2854371A (enrdf_load_stackoverflow)
AU3025871A (enrdf_load_stackoverflow)
AU3038671A (enrdf_load_stackoverflow)
AU2963771A (enrdf_load_stackoverflow)
AU2880771A (enrdf_load_stackoverflow)
AU2885171A (enrdf_load_stackoverflow)
AU2940971A (enrdf_load_stackoverflow)

Legal Events

Date Code Title Description
PL Patent ceased
PL Patent ceased