BE787251A - Nouvelles benzodiazepines et leur preparation - Google Patents

Nouvelles benzodiazepines et leur preparation

Info

Publication number
BE787251A
BE787251A BE787251DA BE787251A BE 787251 A BE787251 A BE 787251A BE 787251D A BE787251D A BE 787251DA BE 787251 A BE787251 A BE 787251A
Authority
BE
Belgium
Prior art keywords
preparation
benzodiazepines
new
new benzodiazepines
Prior art date
Application number
Other languages
English (en)
French (fr)
Inventor
J B Hester Jr
A R Hanze
Pour Lequel Agit J W Hanze
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Publication date
Publication of BE787251A publication Critical patent/BE787251A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/116Heterocyclic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Polymers & Plastics (AREA)
  • Food Science & Technology (AREA)
  • Zoology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Anesthesiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Animal Husbandry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE787251D 1971-08-04 Nouvelles benzodiazepines et leur preparation BE787251A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US16909171A 1971-08-04 1971-08-04

Publications (1)

Publication Number Publication Date
BE787251A true BE787251A (fr) 1973-02-05

Family

ID=22614230

Family Applications (1)

Application Number Title Priority Date Filing Date
BE787251D BE787251A (fr) 1971-08-04 Nouvelles benzodiazepines et leur preparation

Country Status (8)

Country Link
JP (3) JPS5714351B1 (enrdf_load_stackoverflow)
AU (1) AU461139B2 (enrdf_load_stackoverflow)
BE (1) BE787251A (enrdf_load_stackoverflow)
CH (3) CH591488A5 (enrdf_load_stackoverflow)
DE (1) DE2237592C2 (enrdf_load_stackoverflow)
FR (1) FR2150732B1 (enrdf_load_stackoverflow)
GB (4) GB1389437A (enrdf_load_stackoverflow)
ZA (1) ZA724880B (enrdf_load_stackoverflow)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3917627A (en) * 1971-08-04 1975-11-04 Upjohn Co 6-Substituted 4H-imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines and process for their production
FR2183716A1 (en) * 1972-05-05 1973-12-21 Centre Etd Ind Pharma Substd-6-phenyl-4h-imidazo (1,2-a)-1,4-benzo diazepines - - tranquillisers anxiolytics,sedatives and muscle-relaxants
ZA755418B (en) * 1974-09-11 1977-06-29 Hoffmann La Roche Diazepine derivatives
US3910946A (en) * 1974-09-12 1975-10-07 Upjohn Co 4H-Imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines
CA1060892A (en) * 1974-11-06 1979-08-21 Parke, Davis And Company Diazepine compounds and method for their production
AT361486B (de) * 1975-08-07 1981-03-10 Hoffmann La Roche Verfahren zur herstellung von neuen imidazo(1,5 -a) (1,4)diazepinverbindungen, ihren salzen und optisch aktiven formen
US4118386A (en) * 1977-04-04 1978-10-03 Hoffmann-La Roche Inc. Synthesis of imidazo[1,5-a]diazepine-3-carboxylates
AU6909194A (en) * 1993-05-14 1994-12-12 Board Of Regents, The University Of Texas System Preparation of n-cyanodithioimino-carbonates and 3-mercapto-5-amino-1h-1,2,4-triazole
WO1996023790A1 (de) * 1995-02-02 1996-08-08 F. Hoffmann-La Roche Ag Acetylimidazobenzodiazepine
JP6715830B2 (ja) 2014-06-26 2020-07-01 ザ・ジョンズ・ホプキンス・ユニバーシティ 過敏性腸症候群および末梢神経系の他の病気の治療のための末梢限局性gabaポジティブアロステリックモジュレーター
WO2018083051A1 (en) * 2016-11-01 2018-05-11 F. Hoffmann-La Roche Ag 1,3-dihydro-1,4-benzodiazepine-2-thiones for the treatment of cns related diseases
CN113717176B (zh) * 2021-10-09 2022-07-05 上海再启生物技术有限公司 一种制备瑞马唑仑的方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3987052A (en) * 1969-03-17 1976-10-19 The Upjohn Company 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines

Also Published As

Publication number Publication date
AU461139B2 (en) 1975-05-15
GB1389434A (en) 1975-04-03
GB1389436A (en) 1975-04-03
FR2150732A1 (enrdf_load_stackoverflow) 1973-04-13
JPS5547686A (en) 1980-04-04
CH591488A5 (enrdf_load_stackoverflow) 1977-09-30
ZA724880B (en) 1973-06-27
CH584206A5 (enrdf_load_stackoverflow) 1977-01-31
FR2150732B1 (enrdf_load_stackoverflow) 1976-04-16
GB1389435A (en) 1975-04-03
DE2237592A1 (de) 1973-02-15
DE2237592C2 (de) 1985-08-14
AU4467372A (en) 1974-01-24
JPS5734277B2 (enrdf_load_stackoverflow) 1982-07-22
JPS5714351B1 (enrdf_load_stackoverflow) 1982-03-24
GB1389437A (en) 1975-04-03
JPS5726667A (en) 1982-02-12
CH574444A5 (enrdf_load_stackoverflow) 1976-04-15
JPS5732066B2 (enrdf_load_stackoverflow) 1982-07-08

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: THE UPJOHN CY

Effective date: 19860831