CH583231A5 - - Google Patents

Info

Publication number
CH583231A5
CH583231A5 CH1041576A CH1041576A CH583231A5 CH 583231 A5 CH583231 A5 CH 583231A5 CH 1041576 A CH1041576 A CH 1041576A CH 1041576 A CH1041576 A CH 1041576A CH 583231 A5 CH583231 A5 CH 583231A5
Authority
CH
Switzerland
Application number
CH1041576A
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of CH583231A5 publication Critical patent/CH583231A5/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
CH1041576A 1972-06-19 1973-06-14 CH583231A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2229695A DE2229695A1 (de) 1972-06-19 1972-06-19 2-(heteroaryl-methyl)-5,9 beta-dialkyl6,7-benzomorphane, deren saeureadditionssalze sowie verfahren zu deren herstellung

Publications (1)

Publication Number Publication Date
CH583231A5 true CH583231A5 (de) 1976-12-31

Family

ID=5848060

Family Applications (9)

Application Number Title Priority Date Filing Date
CH1041576A CH583231A5 (de) 1972-06-19 1973-06-14
CH1041076A CH583230A5 (de) 1972-06-19 1973-06-14
CH1041176A CH582697A5 (de) 1972-06-19 1973-06-14
CH1040876A CH583228A5 (de) 1972-06-19 1973-06-14
CH1041476A CH589649A5 (de) 1972-06-19 1973-06-14
CH1041376A CH582698A5 (de) 1972-06-19 1973-06-14
CH1041276A CH589648A5 (de) 1972-06-19 1973-06-14
CH1040976A CH583229A5 (de) 1972-06-19 1973-06-14
CH864373A CH583227A5 (de) 1972-06-19 1973-06-14

Family Applications After (8)

Application Number Title Priority Date Filing Date
CH1041076A CH583230A5 (de) 1972-06-19 1973-06-14
CH1041176A CH582697A5 (de) 1972-06-19 1973-06-14
CH1040876A CH583228A5 (de) 1972-06-19 1973-06-14
CH1041476A CH589649A5 (de) 1972-06-19 1973-06-14
CH1041376A CH582698A5 (de) 1972-06-19 1973-06-14
CH1041276A CH589648A5 (de) 1972-06-19 1973-06-14
CH1040976A CH583229A5 (de) 1972-06-19 1973-06-14
CH864373A CH583227A5 (de) 1972-06-19 1973-06-14

Country Status (13)

Country Link
US (1) US3931194A (de)
JP (1) JPS5711908B2 (de)
AT (6) AT325218B (de)
BE (1) BE801079A (de)
CH (9) CH583231A5 (de)
DE (1) DE2229695A1 (de)
DK (1) DK136904C (de)
ES (8) ES416037A1 (de)
FR (1) FR2189056B1 (de)
GB (1) GB1433817A (de)
NL (1) NL7308483A (de)
NO (1) NO137694C (de)
SE (1) SE405121B (de)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2437610A1 (de) * 1974-08-05 1976-02-26 Boehringer Sohn Ingelheim Neue 5,9-beta-disubstituierte 2-tetrahydrofurfuryl-6,7-benzomorphane, deren saeureadditionssalze, ihre verwendung als arzneimittel und verfahren zu deren herstellung
GB1575009A (en) * 1976-06-21 1980-09-17 Acf Chemiefarma Nv 6,7-benzomorphan derivatives
JPS63177704A (ja) * 1987-01-16 1988-07-21 松山株式会社 農作業機連結装置
US8329897B2 (en) 2007-07-26 2012-12-11 Vitae Pharmaceuticals, Inc. Synthesis of inhibitors of 11β-hydroxysteroid dehydrogenase type 1
TW200927115A (en) * 2007-11-16 2009-07-01 Boehringer Ingelheim Int Aryl-and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use
CA2708303A1 (en) 2007-12-11 2009-06-18 Vitae Pharmaceuticals, Inc. Cyclic urea inhibitors of 11.beta.-hydroxysteroid dehydrogenase 1
TW200934490A (en) 2008-01-07 2009-08-16 Vitae Pharmaceuticals Inc Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1
WO2009094169A1 (en) 2008-01-24 2009-07-30 Vitae Pharmaceuticals, Inc. Cyclic carbazate and semicarbazide inhibitors of 11beta-hydroxysteroid dehydrogenase 1
EP2245014B1 (de) * 2008-02-12 2011-11-02 Boehringer Ingelheim International GmbH Harnstoff-derivate von benzomorphanen, entsprechende gerüste, medikamente mit solchen verbindungen und ihre verwendung
EP2254872A2 (de) 2008-02-15 2010-12-01 Vitae Pharmaceuticals, Inc. Cycloalkyllactamderivate als inhibitoren von 11-beta-hydroxysteroiddehydrogenase 1
CA2723039A1 (en) 2008-05-01 2009-11-05 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
WO2009134387A1 (en) 2008-05-01 2009-11-05 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
KR20110002492A (ko) 2008-05-01 2011-01-07 비타이 파마슈티컬즈, 인코포레이티드 11베타-하이드록시스테로이드 탈수소효소 1의 고리형 억제제
TW200950780A (en) 2008-05-13 2009-12-16 Boehringer Ingelheim Int Alicyclic carboxylic acid derivatives of benzomorphans and related scaffolds, medicaments containing such compounds and their use
AU2009274567B2 (en) 2008-07-25 2013-04-04 Boehringer Ingelheim International Gmbh Cyclic inhibitors of 11 beta-hydroxysteroid dehydrogenase 1
CA2729998A1 (en) 2008-07-25 2010-01-28 Boehringer Ingelheim International Gmbh Inhibitors of 11beta-hydroxysteroid dehydrogenase 1
UA109255C2 (ru) 2009-04-30 2015-08-10 Берінгер Інгельхайм Інтернешнл Гмбх Циклические ингибиторы 11бета-гидроксистероиддегидрогеназы 1
US8927539B2 (en) 2009-06-11 2015-01-06 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1 based on the 1,3-oxazinan-2-one structure
TWI531571B (zh) * 2009-11-06 2016-05-01 維它藥物公司 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜芳基羰基衍生物
EP2582698B1 (de) 2010-06-16 2016-09-14 Vitae Pharmaceuticals, Inc. Substituierte 5-,6- und 7-gliedrige heterocyclen, medikamente mit derartigen verbindungen und ihre verwendung
TWI537258B (zh) 2010-11-05 2016-06-11 百靈佳殷格翰國際股份有限公司 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜環芳基羰基衍生物
JP2014524438A (ja) 2011-08-17 2014-09-22 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング インデノピリジン誘導体

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE582575A (de) * 1958-09-22
FR1281227A (fr) * 1958-09-22 1962-01-12 Smith Kline French Lab Perfectionnements apportés aux procédés pour la préparation de dérivés d'aralcoylbenzomorphane
CS166802B2 (de) * 1971-02-08 1976-03-29 Boehringer Sohn Ingelheim
SE392895B (sv) * 1971-08-24 1977-04-25 Sumitomo Chemical Co Forfarande for framstellning av bensomorfanderivat och deras salter

Also Published As

Publication number Publication date
US3931194A (en) 1976-01-06
AT328627B (de) 1976-03-25
ATA489874A (de) 1975-07-15
AT325218B (de) 1975-10-10
ATA489774A (de) 1975-06-15
ES431515A1 (es) 1976-11-01
SE405121B (sv) 1978-11-20
NO137694B (no) 1977-12-27
ES416037A1 (es) 1976-02-16
ATA490074A (de) 1975-06-15
ATA489474A (de) 1975-06-15
DK136904C (da) 1978-06-26
GB1433817A (en) 1976-04-28
ES431516A1 (es) 1976-11-16
CH583229A5 (de) 1976-12-31
AT329199B (de) 1976-04-26
BE801079A (fr) 1973-12-18
ES431514A1 (es) 1976-11-01
CH589649A5 (de) 1977-07-15
JPS4961170A (de) 1974-06-13
FR2189056B1 (de) 1976-10-22
DE2229695A1 (de) 1974-01-31
NL7308483A (de) 1973-12-21
NO137694C (no) 1978-04-05
CH583228A5 (de) 1976-12-31
DK136904B (da) 1977-12-12
CH582698A5 (de) 1976-12-15
AU5704673A (en) 1974-12-19
JPS5711908B2 (de) 1982-03-08
ES431511A1 (es) 1976-11-01
ES431512A1 (es) 1976-11-01
AT328629B (de) 1976-03-25
AT329200B (de) 1976-04-26
FR2189056A1 (de) 1974-01-25
CH583230A5 (de) 1976-12-31
CH582697A5 (de) 1976-12-15
ATA489974A (de) 1975-07-15
CH583227A5 (de) 1976-12-31
AT328628B (de) 1976-03-25
CH589648A5 (de) 1977-07-15
ES431513A1 (es) 1976-11-01
ES431510A1 (es) 1976-11-01

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Legal Events

Date Code Title Description
PL Patent ceased