CH522407A - Procédé pour la préparation de solutions pour usages parentéral, oral et topique de la doxycycline - Google Patents

Procédé pour la préparation de solutions pour usages parentéral, oral et topique de la doxycycline

Info

Publication number
CH522407A
CH522407A CH933769A CH933769A CH522407A CH 522407 A CH522407 A CH 522407A CH 933769 A CH933769 A CH 933769A CH 933769 A CH933769 A CH 933769A CH 522407 A CH522407 A CH 522407A
Authority
CH
Switzerland
Prior art keywords
doxycycline
parenteral
oral
solutions
preparation
Prior art date
Application number
CH933769A
Other languages
English (en)
Inventor
Ernst Beutel Rolf
Christel Lohlbach Kathe
Wilhelm Raaf Helmut
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=5699525&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CH522407(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of CH522407A publication Critical patent/CH522407A/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/65Tetracyclines

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
CH933769A 1968-06-28 1969-06-18 Procédé pour la préparation de solutions pour usages parentéral, oral et topique de la doxycycline CH522407A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE1767891A DE1767891C3 (de) 1968-06-28 1968-06-28 Verfahren zur Herstellung von wäßrigen arzneilichen Lösungen für die parenterale, perorale und lokale Anwendung mit einem Gehalt an einem Tetracyclinderivat

Publications (1)

Publication Number Publication Date
CH522407A true CH522407A (fr) 1972-06-30

Family

ID=5699525

Family Applications (1)

Application Number Title Priority Date Filing Date
CH933769A CH522407A (fr) 1968-06-28 1969-06-18 Procédé pour la préparation de solutions pour usages parentéral, oral et topique de la doxycycline

Country Status (18)

Country Link
US (1) US3674859A (fr)
AT (1) AT291441B (fr)
BE (1) BE734723A (fr)
BR (1) BR6909929D0 (fr)
CH (1) CH522407A (fr)
DE (1) DE1767891C3 (fr)
DK (1) DK127168B (fr)
ES (1) ES368496A1 (fr)
FI (1) FI44395B (fr)
FR (1) FR2011764B1 (fr)
GB (1) GB1228629A (fr)
IE (1) IE33167B1 (fr)
IL (1) IL32350A (fr)
MX (1) MX3351E (fr)
MY (1) MY7300015A (fr)
NL (1) NL6908919A (fr)
NO (1) NO130624C (fr)
SE (1) SE373036B (fr)

Families Citing this family (72)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1350196A (en) * 1972-10-26 1974-04-18 Pfizer Doxycyline parenteral composition
US3957980A (en) * 1972-10-26 1976-05-18 Pfizer Inc. Doxycycline parenteral compositions
US3928592A (en) * 1974-02-22 1975-12-23 Lilly Co Eli Antibiotic pharmaceutical compositions
GB1538903A (en) * 1975-04-11 1979-01-24 Nelson Res & Dev Carrier for a topically applied physiologically active agent or cosmetic agent
US4018889A (en) * 1976-01-02 1977-04-19 Pfizer Inc. Oxytetracycline compositions
GB1592053A (en) * 1976-12-16 1981-07-01 Norbrook Lab Ltd Oxytetracycline compositions
US4213963A (en) * 1978-12-14 1980-07-22 Janssen Pharmaceutica N.V. Fluspirilene-containing compositions
IE74244B1 (en) * 1985-10-01 1997-07-16 Bimeda Res Dev Ltd A process for preparing an antibiotic composition
US6756365B2 (en) * 1991-11-06 2004-06-29 Trustees Of Tufts College Reducing tetracycline resistance in living cells
US6849615B2 (en) 1999-09-14 2005-02-01 Paratek Pharmaceuticals, Inc. 13-substituted methacycline compounds
US8106225B2 (en) * 1999-09-14 2012-01-31 Trustees Of Tufts College Methods of preparing substituted tetracyclines with transition metal-based chemistries
ES2260051T3 (es) 1999-09-14 2006-11-01 Trustees Of Tufts College Metodo para preparar tetraciclinas substituidas con quimicas basadas en metales de transicion.
US6500812B2 (en) 1999-09-14 2002-12-31 Paratek Pharmaceuticals, Inc. 13-substituted methacycline compounds
AU3105801A (en) 2000-01-24 2001-07-31 Trustees Of Tufts College Tetracycline compounds for treatment of cryptosporidium parvum related disorders
HUP0300082A2 (en) * 2000-03-31 2003-05-28 Paratek Pharmaceuticals 7- and 9-carbamate, urea, thiourea, thiocarbamate, and heteroaryl-amino substituted tetracycline derivatives, process for their preparation and use and pharmaceutical compositions containing them
AU2001259701A1 (en) 2000-05-15 2001-11-26 Paratek Pharmaceuticals, Inc 7-substituted fused ring tetracycline compounds
WO2001098236A2 (fr) * 2000-06-16 2001-12-27 Trustees Of Tufts College Composes de tetracycline 7-phenyl-substituee
US20020132798A1 (en) * 2000-06-16 2002-09-19 Nelson Mark L. 7-phenyl-substituted tetracycline compounds
US20040224927A1 (en) * 2000-06-16 2004-11-11 Trustees Of Tufts College 7-N-substituted phenyl tetracycline compounds
ATE544745T1 (de) 2000-07-07 2012-02-15 Tufts College 9-substituierte minocyclinverbindungen
US7094806B2 (en) * 2000-07-07 2006-08-22 Trustees Of Tufts College 7, 8 and 9-substituted tetracycline compounds
CA2415086A1 (fr) 2000-07-07 2002-01-17 Trustees Of Tufts College Composes de tetracycline substitues en 7, 8 et 9
AU2001271642B2 (en) 2000-07-07 2006-01-05 Paratek Pharmaceuticals, Inc. 7-substituted tetracycline compounds
MXPA03000036A (es) 2000-07-07 2003-07-14 Tufts College Compuestos de metaciclina sustituidos en posicion 13.
US20050143353A1 (en) * 2000-07-07 2005-06-30 Paratek Pharmaceuticals, Inc. 13-Substituted methacycline compounds
MXPA03008165A (es) 2001-03-13 2003-12-12 Paratek Pharm Innc Compuestos tetraciclina sustituidos en la posicion 7,9.
JP2005504722A (ja) 2001-03-14 2005-02-17 パラテック ファーマシューティカルズ インコーポレイテッド 相乗的抗真菌薬剤としての置換テトラサイクリン化合物
CA2457234A1 (fr) * 2001-03-14 2002-09-19 Mark L. Nelson Composes de tetracycline substitues, en tant qu'agents antifongiques
DE60235083D1 (de) 2001-04-24 2010-03-04 Paratek Pharm Innc Substituierte tetracyclin-verbindungen zur behandlung von malaria
US8088820B2 (en) * 2001-04-24 2012-01-03 Paratek Pharmaceuticals, Inc. Substituted tetracycline compounds for the treatment of malaria
AU2003235759A1 (en) * 2002-01-08 2003-07-24 Paratek Pharmaceuticals, Inc. 4-dedimethylamino tetracycline compounds
CA2473931C (fr) * 2002-01-23 2010-10-26 Dentsply International, Inc. Solution d'irrigation et procedes d'utilisation
EA201000491A1 (ru) 2002-03-08 2010-08-30 Паратек Фармасьютикалс, Инк. Аминометилзамещенные тетрациклиновые соединения
WO2003079984A2 (fr) 2002-03-21 2003-10-02 Paratek Pharmaceuticals, Inc. Composes de tetracycline substituee
KR101148415B1 (ko) 2002-07-12 2012-05-21 파라테크 파마슈티컬스, 인크. 3, 10, 및 12a 치환된 테트라시클린 화합물
AU2003287218C1 (en) 2002-10-24 2010-07-15 Paratek Pharmaceuticals, Inc. Substituted tetracycline compounds for the treatment of malaria
EP2298323A3 (fr) 2003-07-09 2011-05-11 Paratek Pharmaceuticals, Inc. Composés de tétracycline substitués
US20060287283A1 (en) * 2003-07-09 2006-12-21 Paratek Pharmaceuticals, Inc. Prodrugs of 9-aminomethyl tetracycline compounds
EP2292590A3 (fr) 2003-07-09 2012-05-02 Paratek Pharmaceuticals, Inc. Promédicaments de composés de tétracycline 9-aminométhylé
CN103040773A (zh) * 2003-07-25 2013-04-17 沃纳奇尔科特有限责任公司 多西环素金属络合物固体剂型
EP2332904A3 (fr) 2004-01-15 2012-04-11 Paratek Pharmaceuticals, Inc. Derives des composes de tetracycline
TWI261038B (en) * 2004-08-11 2006-09-01 Bo-Cheng Chen Bicycle gear-shifting handgrip
EP1805134B1 (fr) * 2004-10-25 2012-06-20 Paratek Pharmaceuticals, Inc. 4-aminotetracyclines et procedes d'utilisation
CA2585248A1 (fr) 2004-10-25 2006-05-04 Paratek Pharmaceuticals, Inc. Composes de tetracycline substitues
SG158869A1 (en) * 2005-01-21 2010-02-26 Warner Chilcott Co Llc A tetracycline metal complex in a solid dosage form
US8088755B2 (en) * 2005-02-04 2012-01-03 Paratek Pharmaceuticals, Inc. 11a, 12-derivatives of tetracycline compounds
US20070093455A1 (en) * 2005-07-21 2007-04-26 Paul Abato 10-substituted tetracyclines and methods of use thereof
CA2639406A1 (fr) 2006-01-24 2007-08-02 Paratek Pharmaceuticals, Inc. Procede permettant d'accroitre la biodisponibilite orale de tetracyclines
JP4205731B2 (ja) * 2006-04-05 2009-01-07 株式会社日本触媒 ポリビニルピロリドン粉体組成物およびその製造方法
CA2649221A1 (fr) * 2006-04-17 2007-10-25 Evgeny Tsiperman Isolement de derives de la tetracycline
US8198470B2 (en) * 2006-04-24 2012-06-12 Teva Pharmaceutical Industries Ltd. Crystalline form II of tigecycline and processes for preparation thereof
US7871993B2 (en) * 2006-04-24 2011-01-18 Teva Pharmaceutical Industries Ltd. Tigecycline crystalline forms and processes for preparation thereof
CA2652346A1 (fr) * 2006-05-15 2007-11-22 Paratek Pharmaceuticals, Inc. Methodes de regulation de l'expression de genes ou de produits geniques a l'aide de composes de tetracycline substituee
WO2008045507A2 (fr) 2006-10-11 2008-04-17 Paratek Pharmaceuticals, Inc. Composés de tétracycline substitués utilisés pour le traitement d'infections à bacillus anthracis
CA2673466C (fr) * 2006-12-21 2016-06-14 Paratek Pharmaceuticals, Inc. Composes de tetracycline substituee
CA2892739A1 (fr) 2006-12-21 2008-07-03 Paratek Pharmaceuticals, Inc. Utilisation de composes a base de tetracycline substituee dans le traitement d'affections cutanees inflammatoires
JP5121470B2 (ja) * 2007-01-26 2013-01-16 株式会社日本触媒 ポリビニルピロリドン粉体組成物
CA2688725A1 (en) * 2007-04-12 2008-10-23 Paratek Pharmaceuticals, Inc. Methods for treating spinal muscular atrophy using tetracycline compounds
EP2216323A3 (fr) 2007-04-27 2010-12-29 Paratek Pharmaceuticals, Inc. Procédés de synthèse et de purification de composés d'aminoalkyle de tétracycline
BRPI0823405A2 (pt) 2007-07-06 2012-12-25 Paratek Pharm Innc mÉtodos para sintetizar compostos de tetraciclina substituÍda
CN102015602A (zh) 2008-03-05 2011-04-13 帕拉特克药品公司 米诺环素化合物及其使用方法
PT2271348T (pt) 2008-03-28 2018-04-16 Paratek Pharm Innc Formulação de comprimido oral de composto de tetraciclina
EP2276342A4 (fr) * 2008-04-14 2012-02-22 Paratek Pharm Innc Composés à base de tétracyclines substituées
TWI680117B (zh) 2008-05-23 2019-12-21 派洛泰克藥物股份有限公司 四環素化合物之甲苯磺酸鹽及同素異形體
CN102215681A (zh) * 2008-09-19 2011-10-12 帕拉特克药品公司 用于治疗类风湿性关节炎的四环素化合物和相关的治疗方法
US20120121706A1 (en) 2009-04-10 2012-05-17 Tufts Medical Center, Inc. PAR-1 Activation by Metalloproteinase-1 (MMP-1)
HUE033161T2 (en) 2010-05-12 2017-11-28 Rempex Pharmaceuticals Inc Tetracycline compositions
CN101862293B (zh) * 2010-06-22 2012-02-29 华南农业大学 盐酸多西环素的油混悬液及其制备方法和应用
LT2707003T (lt) 2011-05-12 2019-10-10 Paratek Pharmaceuticals, Inc. Kristalinės (4s,4as,5ar,12as)-4-dimetilamino-3,10,12,12a-tetrahidroksi-7-[(metoksi(metil)amino)-metil]-1,11-diokso-1,4,4a,5,5a,6,11,12a-oktahidro-naftacen-2-karboksirūgšties amido druskos ir jų panaudojimo būdai
PT108978B (pt) 2015-11-24 2020-03-09 Hovione Farm S A Sais de tetraciclinas
RU2019113715A (ru) 2016-11-01 2020-12-03 Паратек Фармасьютикалс, Инк. 9-аминометилминоциклиновые соединения и их применение для лечениия внебольничной бактериальной пневмонии(вбп)
KR102662461B1 (ko) 2017-07-21 2024-04-30 알미랄 엘엘씨 비염증성 병변의 치료

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1430859A (fr) * 1960-05-23 1966-05-25

Also Published As

Publication number Publication date
DK127168B (da) 1973-10-01
DE1767891B2 (de) 1980-02-21
US3674859A (en) 1972-07-04
AT291441B (de) 1971-07-12
ES368496A1 (es) 1971-05-01
NO130624C (fr) 1975-01-15
DE1767891A1 (de) 1971-07-08
BR6909929D0 (pt) 1973-02-08
IE33167L (en) 1969-12-28
IL32350A (en) 1972-05-30
MX3351E (es) 1980-10-08
NL6908919A (fr) 1969-12-30
NO130624B (fr) 1974-10-07
BE734723A (fr) 1969-12-18
FR2011764A1 (fr) 1970-03-06
MY7300015A (en) 1973-12-31
FI44395B (fr) 1971-08-02
IE33167B1 (en) 1974-04-03
DE1767891C3 (de) 1980-10-30
FR2011764B1 (fr) 1973-07-13
GB1228629A (fr) 1971-04-15
IL32350A0 (en) 1969-08-27
SE373036B (fr) 1975-01-27

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