CH495366A - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepin-Derivaten

Info

Publication number
CH495366A
CH495366A CH1129667A CH1129667A CH495366A CH 495366 A CH495366 A CH 495366A CH 1129667 A CH1129667 A CH 1129667A CH 1129667 A CH1129667 A CH 1129667A CH 495366 A CH495366 A CH 495366A
Authority
CH
Switzerland
Prior art keywords
oxime
chloro
amino
alkyl
dependent
Prior art date
Application number
CH1129667A
Other languages
German (de)
English (en)
Inventor
Joseph Dr Hellerbach
Armin Dr Walser
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Priority to CH1059170A priority Critical patent/CH500997A/de
Priority to CH1129667A priority patent/CH495366A/de
Priority to CH1059270A priority patent/CH503750A/de
Priority to CH1059070A priority patent/CH506541A/de
Priority to AT609168A priority patent/AT279621B/de
Priority to IL30374A priority patent/IL30374A0/xx
Priority to DE19681770945 priority patent/DE1770945A1/de
Priority to ES357030A priority patent/ES357030A1/es
Priority to BE719208D priority patent/BE719208A/xx
Priority to NL6811366A priority patent/NL6811366A/xx
Priority to IE976/68A priority patent/IE32263B1/xx
Priority to GB3817068A priority patent/GB1198349A/en
Priority to FR1588550D priority patent/FR1588550A/fr
Priority to FR162501A priority patent/FR7753M/fr
Publication of CH495366A publication Critical patent/CH495366A/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CH1129667A 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten CH495366A (de)

Priority Applications (14)

Application Number Priority Date Filing Date Title
CH1059170A CH500997A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1129667A CH495366A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1059270A CH503750A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1059070A CH506541A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten
AT609168A AT279621B (de) 1967-08-09 1968-06-25 Verfahren zur Herstellung von neuen Nitonen und den Säureadditionssalzen basischer Verbindungen
IL30374A IL30374A0 (en) 1967-08-09 1968-07-16 Benzodiazepine derivatives and process for the manufacture thereof
DE19681770945 DE1770945A1 (de) 1967-08-09 1968-07-22 Verfahren zur Herstellung von Benzodiazepin-Derivaten
ES357030A ES357030A1 (es) 1967-08-09 1968-08-08 Procedimiento para la preparacion de derivados de benzodia-cepina.
BE719208D BE719208A (fr) 1967-08-09 1968-08-08
NL6811366A NL6811366A (fr) 1967-08-09 1968-08-09
IE976/68A IE32263B1 (en) 1967-08-09 1968-08-09 Benzodiazepine derivatives and process for the manufacture thereof
GB3817068A GB1198349A (en) 1967-08-09 1968-08-09 Benzdiaz[1,4]Epine Derivatives
FR1588550D FR1588550A (fr) 1967-08-09 1968-08-09
FR162501A FR7753M (fr) 1967-08-09 1968-08-09

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH1129667A CH495366A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1059070A CH506541A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1059270A CH503750A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Publications (1)

Publication Number Publication Date
CH495366A true CH495366A (de) 1970-08-31

Family

ID=27176471

Family Applications (3)

Application Number Title Priority Date Filing Date
CH1059270A CH503750A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1059070A CH506541A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1129667A CH495366A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Family Applications Before (2)

Application Number Title Priority Date Filing Date
CH1059270A CH503750A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1059070A CH506541A (de) 1967-08-09 1967-08-09 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Country Status (6)

Country Link
BE (1) BE719208A (fr)
CH (3) CH503750A (fr)
DE (1) DE1770945A1 (fr)
FR (2) FR1588550A (fr)
GB (1) GB1198349A (fr)
NL (1) NL6811366A (fr)

Also Published As

Publication number Publication date
DE1770945A1 (de) 1972-01-13
GB1198349A (en) 1970-07-08
NL6811366A (fr) 1969-02-11
CH503750A (de) 1971-02-28
FR7753M (fr) 1970-03-16
BE719208A (fr) 1969-02-10
CH506541A (de) 1971-04-30
FR1588550A (fr) 1970-04-17

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Legal Events

Date Code Title Description
PL Patent ceased