CA3243809A1 - ANTIBIOTIC COMPOUNDS, FORMULATIONS AND METHODS OF USE - Google Patents

ANTIBIOTIC COMPOUNDS, FORMULATIONS AND METHODS OF USE

Info

Publication number
CA3243809A1
CA3243809A1 CA3243809A CA3243809A CA3243809A1 CA 3243809 A1 CA3243809 A1 CA 3243809A1 CA 3243809 A CA3243809 A CA 3243809A CA 3243809 A CA3243809 A CA 3243809A CA 3243809 A1 CA3243809 A1 CA 3243809A1
Authority
CA
Canada
Prior art keywords
optionally substituted
moiety
polymyxin
amino
substituted alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CA3243809A
Other languages
English (en)
French (fr)
Inventor
Nathaniel I. Martin
Jaco SLINGERLAND
Original Assignee
Universiteit Leiden
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Universiteit Leiden filed Critical Universiteit Leiden
Publication of CA3243809A1 publication Critical patent/CA3243809A1/en
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/60Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation occurring through the 4-amino group of 2,4-diamino-butanoic acid
    • C07K7/62Polymyxins; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Public Health (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
CA3243809A 2022-02-11 2023-02-13 ANTIBIOTIC COMPOUNDS, FORMULATIONS AND METHODS OF USE Pending CA3243809A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
NL2030897A NL2030897B1 (en) 2022-02-11 2022-02-11 Antibiotic compounds, formulations and methods of use
NL2030897 2022-02-11
PCT/NL2023/050065 WO2023153932A1 (en) 2022-02-11 2023-02-13 Antibiotic compounds, formulations and methods of use

Publications (1)

Publication Number Publication Date
CA3243809A1 true CA3243809A1 (en) 2023-08-17

Family

ID=85283807

Family Applications (1)

Application Number Title Priority Date Filing Date
CA3243809A Pending CA3243809A1 (en) 2022-02-11 2023-02-13 ANTIBIOTIC COMPOUNDS, FORMULATIONS AND METHODS OF USE

Country Status (7)

Country Link
US (1) US20250171498A1 (https=)
EP (1) EP4476239A1 (https=)
JP (1) JP2025505237A (https=)
CN (1) CN118871454A (https=)
CA (1) CA3243809A1 (https=)
NL (1) NL2030897B1 (https=)
WO (1) WO2023153932A1 (https=)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112014012016A2 (pt) * 2011-11-18 2017-05-16 Cantab Anti-Infectives Ltd compostos
EP3636659A1 (en) * 2018-10-08 2020-04-15 Universitat de Barcelona Polymyxin-based compounds useful as antibacterial agents
WO2021150792A1 (en) * 2020-01-21 2021-07-29 Micurx Pharmaceuticals, Inc. Novel compounds and composition for targeted therapy of kidney-associated cancers
CN118201946A (zh) * 2021-08-12 2024-06-14 奥克兰联合服务有限公司 脂化多粘菌素类似物

Also Published As

Publication number Publication date
JP2025505237A (ja) 2025-02-21
US20250171498A1 (en) 2025-05-29
CN118871454A (zh) 2024-10-29
NL2030897B1 (en) 2023-08-18
WO2023153932A1 (en) 2023-08-17
EP4476239A1 (en) 2024-12-18

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