CA3047002A1 - Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase - Google Patents
Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase Download PDFInfo
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- CA3047002A1 CA3047002A1 CA3047002A CA3047002A CA3047002A1 CA 3047002 A1 CA3047002 A1 CA 3047002A1 CA 3047002 A CA3047002 A CA 3047002A CA 3047002 A CA3047002 A CA 3047002A CA 3047002 A1 CA3047002 A1 CA 3047002A1
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- alkyl
- compound
- independently selected
- membered
- cycloalkyl
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- A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
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| WO2018136437A2 (en) | 2017-01-17 | 2018-07-26 | Tesaro, Inc. | Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase |
| WO2020018670A1 (en) * | 2018-07-17 | 2020-01-23 | Board Of Regents, The University Of Texas System | Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase |
| US20210379052A1 (en) * | 2018-09-27 | 2021-12-09 | Shenzhen Chipscreen Biosciences Co., Ltd. | Quinoline derivative having indoleamine-2,3-dioxygenase inhibitory activity |
| US12091405B2 (en) | 2018-11-01 | 2024-09-17 | Merck Sharp & Dohme Llc | Substituted pyrazole compounds as indoleamine 2,3-dioxygenase inhibitors |
| EP3886845B1 (en) * | 2018-11-28 | 2024-09-04 | Merck Sharp & Dohme LLC | Novel substituted piperazine amide compounds as indoleamine 2, 3-dioxygenase (ido) inhibitors |
| KR20220034739A (ko) * | 2019-05-31 | 2022-03-18 | 이케나 온콜로지, 인코포레이티드 | Tead 억제제 및 이의 용도 |
| CN112107685A (zh) * | 2020-07-17 | 2020-12-22 | 深圳市第二人民医院 | 一种基于ido1酶抑制剂设计的治疗骨关节炎的方法 |
| CN115215780B (zh) * | 2022-04-22 | 2023-08-08 | 上海格苓凯生物科技有限公司 | 一种利用n,n-二琥珀酰亚胺基碳酸酯制备异双功能交联剂smcc的方法 |
| EP4535004A4 (en) * | 2022-05-27 | 2025-09-17 | Fujifilm Corp | METHOD FOR AID IN THE DIAGNOSIS OF A BLOOD TUMOR, METHOD FOR OBTAINING DATA FOR THE DIAGNOSIS OF A BLOOD TUMOR AND KIT FOR SAID METHODS |
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2018
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- 2018-01-16 US US16/478,076 patent/US11173145B2/en active Active
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- 2018-01-16 JP JP2019538180A patent/JP2020506895A/ja active Pending
- 2018-01-16 EP EP18741114.5A patent/EP3570832A4/en not_active Withdrawn
- 2018-01-16 CA CA3047002A patent/CA3047002A1/en not_active Abandoned
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| WO2018136437A3 (en) | 2018-08-30 |
| JP2020506895A (ja) | 2020-03-05 |
| CN110191709A (zh) | 2019-08-30 |
| EP3570832A2 (en) | 2019-11-27 |
| US20190365718A1 (en) | 2019-12-05 |
| EP3570832A4 (en) | 2020-06-10 |
| US11173145B2 (en) | 2021-11-16 |
| WO2018136437A2 (en) | 2018-07-26 |
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