CA3047002A1 - Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase - Google Patents
Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase Download PDFInfo
- Publication number
- CA3047002A1 CA3047002A1 CA3047002A CA3047002A CA3047002A1 CA 3047002 A1 CA3047002 A1 CA 3047002A1 CA 3047002 A CA3047002 A CA 3047002A CA 3047002 A CA3047002 A CA 3047002A CA 3047002 A1 CA3047002 A1 CA 3047002A1
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- Prior art keywords
- alkyl
- compound
- independently selected
- membered
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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| JP2020506895A (ja) | 2017-01-17 | 2020-03-05 | ボード オブ レジェンツ, ザ ユニバーシティ オブ テキサス システムBoard Of Regents, The University Of Texas System | インドールアミン2,3−ジオキシゲナーゼおよび/またはトリプトファンジオキシゲナーゼの阻害剤として有用な化合物 |
| US11046649B2 (en) | 2018-07-17 | 2021-06-29 | Board Of Regents, The University Of Texas System | Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase |
| EP3858813A4 (en) * | 2018-09-27 | 2022-06-22 | Shenzhen Chipscreen Biosciences Co., Ltd. | QUINOLONE DERIVATIVE WITH INDOLEAMINE-2,3-DIOXYGENASE INHIBITED ACTIVITY |
| US12091405B2 (en) | 2018-11-01 | 2024-09-17 | Merck Sharp & Dohme Llc | Substituted pyrazole compounds as indoleamine 2,3-dioxygenase inhibitors |
| WO2020112581A1 (en) * | 2018-11-28 | 2020-06-04 | Merck Sharp & Dohme Corp. | Novel substituted piperazine amide compounds as indoleamine 2, 3-dioxygenase (ido) inhibitors |
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| KR20190003687A (ko) | 2016-05-04 | 2019-01-09 | 브리스톨-마이어스 스큅 컴퍼니 | 인돌아민 2,3-디옥시게나제의 억제제 및 그의 사용 방법 |
| JP2019528301A (ja) | 2016-08-26 | 2019-10-10 | ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company | インドールアミン2,3−ジオキシゲナーゼの阻害剤およびその使用方法 |
| JP2020506895A (ja) | 2017-01-17 | 2020-03-05 | ボード オブ レジェンツ, ザ ユニバーシティ オブ テキサス システムBoard Of Regents, The University Of Texas System | インドールアミン2,3−ジオキシゲナーゼおよび/またはトリプトファンジオキシゲナーゼの阻害剤として有用な化合物 |
| WO2018136887A1 (en) | 2017-01-23 | 2018-07-26 | Tesaro, Inc. | Compounds |
| US11046649B2 (en) | 2018-07-17 | 2021-06-29 | Board Of Regents, The University Of Texas System | Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase |
-
2018
- 2018-01-16 JP JP2019538180A patent/JP2020506895A/ja active Pending
- 2018-01-16 CA CA3047002A patent/CA3047002A1/en not_active Abandoned
- 2018-01-16 WO PCT/US2018/013914 patent/WO2018136437A2/en not_active Ceased
- 2018-01-16 CN CN201880006825.0A patent/CN110191709A/zh active Pending
- 2018-01-16 US US16/478,076 patent/US11173145B2/en active Active
- 2018-01-16 EP EP18741114.5A patent/EP3570832A4/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| US20190365718A1 (en) | 2019-12-05 |
| WO2018136437A3 (en) | 2018-08-30 |
| WO2018136437A2 (en) | 2018-07-26 |
| EP3570832A2 (en) | 2019-11-27 |
| CN110191709A (zh) | 2019-08-30 |
| US11173145B2 (en) | 2021-11-16 |
| EP3570832A4 (en) | 2020-06-10 |
| JP2020506895A (ja) | 2020-03-05 |
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Legal Events
| Date | Code | Title | Description |
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| FZDE | Discontinued |
Effective date: 20230718 |