CA2990445C - Thermo-kinetic mixing for pharmaceutical applications - Google Patents
Thermo-kinetic mixing for pharmaceutical applications Download PDFInfo
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- CA2990445C CA2990445C CA2990445A CA2990445A CA2990445C CA 2990445 C CA2990445 C CA 2990445C CA 2990445 A CA2990445 A CA 2990445A CA 2990445 A CA2990445 A CA 2990445A CA 2990445 C CA2990445 C CA 2990445C
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Classifications
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- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
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- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
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Landscapes
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- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (1)
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| CA2990445C (en) * | 2007-08-21 | 2020-05-05 | Board Of Regents, The University Of Texas System | Thermo-kinetic mixing for pharmaceutical applications |
| US9545361B1 (en) * | 2011-07-25 | 2017-01-17 | Dispersol Technologies, Llc | Multiple speed process for preserving heat sensitive portions of a thermokinetically melt blended batch |
| WO2010005726A2 (en) | 2008-06-16 | 2010-01-14 | Bind Biosciences Inc. | Therapeutic polymeric nanoparticles with mtor inhibitors and methods of making and using same |
| JP2012501965A (ja) * | 2008-06-16 | 2012-01-26 | バインド バイオサイエンシズ インコーポレイテッド | 薬剤を装填したポリマーナノ粒子及びその製造方法と使用方法 |
| EP2309991B1 (en) | 2008-06-16 | 2019-03-06 | Pfizer Inc | Therapeutic polymeric nanoparticles comprising vinca alkaloids and methods of making and using same |
| CA2741862C (en) * | 2008-10-31 | 2017-10-17 | Mahmoud A. Elsohly | Compositions containing delta-9-thc-amino acid esters and process of preparation |
| US8563041B2 (en) | 2008-12-12 | 2013-10-22 | Bind Therapeutics, Inc. | Therapeutic particles suitable for parenteral administration and methods of making and using same |
| EP2379064B1 (en) * | 2008-12-15 | 2020-02-26 | Pfizer Inc. | Long circulating nanoparticles for sustained release of therapeutic agents |
| NZ594207A (en) | 2009-02-06 | 2013-03-28 | Egalet Ltd | Immediate release composition resistant to abuse by intake of alcohol |
| NZ597283A (en) | 2009-06-24 | 2013-07-26 | Egalet Ltd | Controlled release formulations |
| WO2011072218A2 (en) | 2009-12-11 | 2011-06-16 | Bind Biosciences | Stable formulations for lyophilizing therapeutic particles |
| ES2780156T3 (es) | 2009-12-15 | 2020-08-24 | Pfizer | Composiciones terapéuticas de nanopartículas poliméricas con alta temperatura de transición vítrea o copolímeros de alto peso molecular |
| US20140039031A1 (en) * | 2011-02-23 | 2014-02-06 | Dispersol Technologies. LLC | Pharmaceutical formulations of acetyl-11-keto-b-boswellic acid, diindolylmethane, and curcumin for pharmaceutical applications |
| CN102204868B (zh) * | 2011-05-18 | 2014-01-22 | 北京化工大学 | 采用多元辅料制备吲哚美辛速释制剂的热熔挤出工艺 |
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| US9877923B2 (en) | 2012-09-17 | 2018-01-30 | Pfizer Inc. | Process for preparing therapeutic nanoparticles |
| CA2935307C (en) | 2013-12-31 | 2023-05-09 | Ascendia Pharmaceuticals, Llc | Pharmaceutical compositions for poorly water-soluble compounds |
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| CN107205935A (zh) * | 2015-01-20 | 2017-09-26 | 默克专利股份有限公司 | 用聚乙烯醇作载体聚合物的化合物固体分散体 |
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| EP4552641A3 (en) * | 2016-05-09 | 2025-07-30 | AustinPx, LLC | Improved drug formulations |
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2008
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- 2008-08-21 WO PCT/US2008/073913 patent/WO2009026461A2/en not_active Ceased
- 2008-08-21 JP JP2010522038A patent/JP6073043B2/ja active Active
- 2008-08-21 CN CN2008801123533A patent/CN101835492B/zh active Active
- 2008-08-21 CA CA2697099A patent/CA2697099C/en active Active
- 2008-08-21 CA CA3076115A patent/CA3076115C/en active Active
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- 2008-08-21 EP EP08798412A patent/EP2187968A4/en not_active Ceased
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2013
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2014
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2018
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Also Published As
| Publication number | Publication date |
|---|---|
| CN101835492B (zh) | 2012-11-21 |
| WO2009026461A2 (en) | 2009-02-26 |
| JP2014221816A (ja) | 2014-11-27 |
| CA2697099A1 (en) | 2009-02-26 |
| US10022385B2 (en) | 2018-07-17 |
| US10668085B2 (en) | 2020-06-02 |
| US20090053315A1 (en) | 2009-02-26 |
| JP2016121195A (ja) | 2016-07-07 |
| US20230172949A1 (en) | 2023-06-08 |
| JP6073043B2 (ja) | 2017-02-01 |
| US20180360850A1 (en) | 2018-12-20 |
| CA3076115C (en) | 2022-06-28 |
| US12023343B2 (en) | 2024-07-02 |
| WO2009026461A3 (en) | 2009-04-30 |
| CN101835492A (zh) | 2010-09-15 |
| EP2187968A2 (en) | 2010-05-26 |
| US20130303630A1 (en) | 2013-11-14 |
| JP2019052173A (ja) | 2019-04-04 |
| JP2010536877A (ja) | 2010-12-02 |
| CA3076115A1 (en) | 2009-02-26 |
| US9339440B2 (en) | 2016-05-17 |
| US11439650B2 (en) | 2022-09-13 |
| EP2187968A4 (en) | 2013-02-20 |
| CA2697099C (en) | 2018-02-20 |
| US20160250230A1 (en) | 2016-09-01 |
| US20200261473A1 (en) | 2020-08-20 |
| US8486423B2 (en) | 2013-07-16 |
| CA2990445A1 (en) | 2009-02-26 |
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