CA2960090A1 - Compound - Google Patents
Compound Download PDFInfo
- Publication number
- CA2960090A1 CA2960090A1 CA2960090A CA2960090A CA2960090A1 CA 2960090 A1 CA2960090 A1 CA 2960090A1 CA 2960090 A CA2960090 A CA 2960090A CA 2960090 A CA2960090 A CA 2960090A CA 2960090 A1 CA2960090 A1 CA 2960090A1
- Authority
- CA
- Canada
- Prior art keywords
- ethylacetamide
- methyloxy
- methyl
- triazolo
- sulphonic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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| WO2016090219A1 (en) | 2014-12-05 | 2016-06-09 | H. Lee Moffitt Cancer Center And Research Institute, Inc. | Bromodomain inhibitor as adjuvant in cancer immunotherapy |
| EP3270917A4 (en) | 2015-03-18 | 2018-08-08 | Arvinas, Inc. | Compounds and methods for the enhanced degradation of targeted proteins |
| EP3337476A4 (en) | 2015-08-19 | 2019-09-04 | Arvinas, Inc. | Compounds and methods for the targeted degradation of bromodomain-containing proteins |
| US20190284192A1 (en) | 2016-11-10 | 2019-09-19 | Luoxin Pharmaceutical (Shanghai) Co., Ltd. | Nitrogenous macrocyclic compound, preparation method therefor, pharmaceutical composition and application thereof |
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| EP3743066A4 (en) | 2018-01-26 | 2021-09-08 | Yale University | IMIDE-BASED PROTEOLYSIS MODULATORS AND RELATED METHODS OF USE |
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| PH12022551486A1 (en) | 2019-12-19 | 2023-11-13 | Arvinas Operations Inc | Compounds and methods for the targeted degradation of androgen receptor |
| CN111533745A (zh) * | 2020-05-20 | 2020-08-14 | 成都药明康德新药开发有限公司 | 叔丁基-3-(氨基甲基)二氢-5h-三唑并二氮杂卓-8(9h)-甲酸基酯制法 |
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- 2015-09-30 BR BR112017006342A patent/BR112017006342A2/pt not_active Application Discontinuation
-
2018
- 2018-04-18 US US15/955,857 patent/US10450319B2/en not_active Expired - Fee Related
-
2019
- 2019-09-05 US US16/561,208 patent/US20190389870A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN106715439A (zh) | 2017-05-24 |
| WO2016050821A1 (en) | 2016-04-07 |
| US20170298071A1 (en) | 2017-10-19 |
| US9975901B2 (en) | 2018-05-22 |
| RU2697393C2 (ru) | 2019-08-14 |
| AU2015326910A1 (en) | 2017-03-30 |
| JP2017530155A (ja) | 2017-10-12 |
| RU2017107760A (ru) | 2018-11-02 |
| RU2017107760A3 (enExample) | 2019-03-01 |
| AU2015326910B2 (en) | 2018-03-01 |
| BR112017006342A2 (pt) | 2017-12-19 |
| US20180305365A1 (en) | 2018-10-25 |
| US20190389870A1 (en) | 2019-12-26 |
| EP3201199A1 (en) | 2017-08-09 |
| US10450319B2 (en) | 2019-10-22 |
| KR20170055549A (ko) | 2017-05-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |
Effective date: 20211221 |
|
| FZDE | Discontinued |
Effective date: 20211221 |