CA2932529C - Therapeutic and/or preventive agent comprising 1-indansulfamide derivative for pain - Google Patents

Therapeutic and/or preventive agent comprising 1-indansulfamide derivative for pain Download PDF

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Publication number
CA2932529C
CA2932529C CA2932529A CA2932529A CA2932529C CA 2932529 C CA2932529 C CA 2932529C CA 2932529 A CA2932529 A CA 2932529A CA 2932529 A CA2932529 A CA 2932529A CA 2932529 C CA2932529 C CA 2932529C
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CA
Canada
Prior art keywords
pain
mmol
compound
inden
dihydro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
CA2932529A
Other languages
English (en)
French (fr)
Other versions
CA2932529A1 (en
Inventor
Hiroyuki Higashiyama
Yuji Kazuta
Keisuke Hashimoto
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eisai R&D Management Co Ltd
Original Assignee
Eisai R&D Management Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai R&D Management Co Ltd filed Critical Eisai R&D Management Co Ltd
Publication of CA2932529A1 publication Critical patent/CA2932529A1/en
Application granted granted Critical
Publication of CA2932529C publication Critical patent/CA2932529C/en
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/18Sulfonamides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0021Intradermal administration, e.g. through microneedle arrays or needleless injectors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Rheumatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
CA2932529A 2013-12-19 2014-12-17 Therapeutic and/or preventive agent comprising 1-indansulfamide derivative for pain Active CA2932529C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2013-262743 2013-12-19
JP2013262743 2013-12-19
PCT/JP2014/083374 WO2015093515A1 (ja) 2013-12-19 2014-12-17 1-インダンスルファミド誘導体を含む疼痛の治療および/または予防剤

Publications (2)

Publication Number Publication Date
CA2932529A1 CA2932529A1 (en) 2015-06-25
CA2932529C true CA2932529C (en) 2022-03-22

Family

ID=53402860

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2932529A Active CA2932529C (en) 2013-12-19 2014-12-17 Therapeutic and/or preventive agent comprising 1-indansulfamide derivative for pain

Country Status (14)

Country Link
US (1) US9610262B2 (https=)
EP (1) EP3085369B1 (https=)
JP (1) JP6518595B2 (https=)
KR (1) KR102250214B1 (https=)
CN (1) CN105792821B (https=)
AU (1) AU2014367781B2 (https=)
BR (1) BR112016012833B1 (https=)
CA (1) CA2932529C (https=)
ES (1) ES2673876T3 (https=)
IL (1) IL246036B (https=)
MX (1) MX370898B (https=)
RU (1) RU2678571C1 (https=)
SG (1) SG11201604484UA (https=)
WO (1) WO2015093515A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20200132858A (ko) * 2018-03-20 2020-11-25 에자이 알앤드디 매니지먼트 가부시키가이샤 간질 치료제
TW202345782A (zh) * 2022-04-27 2023-12-01 日商衛材R&D企管股份有限公司 帕金森氏症治療用醫藥組成物
KR102815521B1 (ko) 2022-11-11 2025-06-04 덕산에테르씨티 주식회사 내화성능 및 강도가 보강된 압력용기
KR102803991B1 (ko) 2022-11-11 2025-05-13 덕산에테르씨티 주식회사 내화성능 및 강도가 보강된 압력용기
KR102815520B1 (ko) 2022-11-11 2025-06-04 덕산에테르씨티 주식회사 내화성능 및 강도가 보강된 압력용기
KR102917062B1 (ko) 2023-11-01 2026-02-05 덕산에테르씨티 주식회사 압력 용기의 숄더부 보호용 커버
KR102917063B1 (ko) 2023-11-01 2026-02-23 덕산에테르씨티 주식회사 압력 용기의 숄더부 보호용 커버
KR102917061B1 (ko) 2023-11-01 2026-02-05 덕산에테르씨티 주식회사 압력 용기의 숄더부 보호용 커버

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8716231B2 (en) 2005-12-19 2014-05-06 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain
US20070191452A1 (en) 2006-02-15 2007-08-16 Smith-Swintosky Virginia L Use of benzo-heteroaryl sulfamide derivatives for the treatment of pain
CL2007002994A1 (es) 2006-10-19 2008-02-08 Wyeth Corp Compuestos derivados heterociclicos que contienen sulfamoilo, inhibidores de hsp90; composicion farmaceutica; y uso para el tratamiento del cancer, tal como cancer de mama, de colon y prostata, entre otros.
TWI433674B (zh) 2006-12-28 2014-04-11 Infinity Discovery Inc 環杷明(cyclopamine)類似物類
EP2417101B1 (en) * 2009-04-09 2013-10-23 Merck Sharp & Dohme B.V. Indane derivatives
TW201217312A (en) 2010-09-22 2012-05-01 Gruenenthal Gmbh Substituted benzamide compounds
RU2508295C2 (ru) * 2012-03-22 2014-02-27 Общество с ограниченной ответственностью "Биофармокс" Синтетические пептиды с ненаркотическим типом анальгетического действия
MY169073A (en) * 2012-06-21 2019-02-13 Eisai R&D Man Co Ltd Indanesulfamide derivative

Also Published As

Publication number Publication date
IL246036B (en) 2018-11-29
AU2014367781B2 (en) 2019-07-04
JPWO2015093515A1 (ja) 2017-03-23
EP3085369B1 (en) 2018-04-04
KR102250214B1 (ko) 2021-05-07
EP3085369A1 (en) 2016-10-26
US9610262B2 (en) 2017-04-04
WO2015093515A1 (ja) 2015-06-25
SG11201604484UA (en) 2016-07-28
ES2673876T3 (es) 2018-06-26
EP3085369A4 (en) 2017-05-10
RU2016122189A (ru) 2018-01-24
RU2678571C1 (ru) 2019-01-30
CN105792821A (zh) 2016-07-20
CA2932529A1 (en) 2015-06-25
US20160303058A1 (en) 2016-10-20
JP6518595B2 (ja) 2019-05-22
IL246036A0 (en) 2016-07-31
BR112016012833B1 (pt) 2022-11-16
BR112016012833A2 (https=) 2017-08-08
AU2014367781A1 (en) 2016-06-23
CN105792821B (zh) 2018-05-04
MX370898B (es) 2020-01-09
KR20160106053A (ko) 2016-09-09
MX2016007370A (es) 2016-10-03

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Effective date: 20191011