CA2872021C - Glucokinase activator compositions for the treatment of diabetes - Google Patents
Glucokinase activator compositions for the treatment of diabetes Download PDFInfo
- Publication number
- CA2872021C CA2872021C CA2872021A CA2872021A CA2872021C CA 2872021 C CA2872021 C CA 2872021C CA 2872021 A CA2872021 A CA 2872021A CA 2872021 A CA2872021 A CA 2872021A CA 2872021 C CA2872021 C CA 2872021C
- Authority
- CA
- Canada
- Prior art keywords
- insulin
- diabetes
- pharmaceutically acceptable
- glucose
- glucokinase activator
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US201261648110P | 2012-05-17 | 2012-05-17 | |
| US61/648,110 | 2012-05-17 | ||
| PCT/US2013/041076 WO2013173417A2 (en) | 2012-05-17 | 2013-05-15 | Glucokinase activator compositions for the treatment of diabetes |
Publications (2)
| Publication Number | Publication Date |
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| CA2872021A1 CA2872021A1 (en) | 2013-11-21 |
| CA2872021C true CA2872021C (en) | 2022-08-16 |
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| Application Number | Title | Priority Date | Filing Date |
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| CA2872021A Active CA2872021C (en) | 2012-05-17 | 2013-05-15 | Glucokinase activator compositions for the treatment of diabetes |
Country Status (16)
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| EP (1) | EP2849776B1 (en, 2012) |
| JP (1) | JP6234443B2 (en, 2012) |
| KR (2) | KR102371364B1 (en, 2012) |
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| AU (2) | AU2013262895A1 (en, 2012) |
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| MX (1) | MX360304B (en, 2012) |
| SG (2) | SG11201406987UA (en, 2012) |
| WO (1) | WO2013173417A2 (en, 2012) |
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| PL2576524T3 (pl) | 2010-05-26 | 2018-03-30 | Vtv Therapeutics Llc | Zastosowanie metforminy w skojarzeniu z aktywatorem glukokinazy i kompozycje zawierające metforminę i aktywator glukokinazy |
| SG11201406987UA (en) * | 2012-05-17 | 2014-12-30 | Transtech Pharma Llc | Glucokinase activator compositions for the treatment of diabetes |
| KR102408480B1 (ko) | 2018-05-30 | 2022-06-10 | 이삼구 | 당뇨질환의 치료용 조성물 |
| IL279036B2 (en) * | 2018-05-31 | 2025-07-01 | Hua Medicine Shanghai Ltd | Pharmaceutical combination, composition, and combination formulation comprising glucokinase activator and sglt-2 inhibitor and preparation methods and uses thereof |
| MX2020008905A (es) * | 2018-06-12 | 2020-12-03 | Vtv Therapeutics Llc | Usos terapeuticos de activadores de glucoquinasa en combinacion con insulina o analogos de insulinas. |
| CA3169432A1 (en) * | 2020-01-31 | 2021-08-05 | Hua Medicine (Shanghai) Ltd. | Treating treatment-resistant diabetes with glucokinase activator |
| US11872221B2 (en) | 2020-01-31 | 2024-01-16 | Hua Medicine (Shanghai) Ltd. | Treating untreated or treatment-resistant diabetes with glucokinase activator |
| WO2021167840A1 (en) | 2020-02-18 | 2021-08-26 | Vtv Therapeutics Llc | Sulfoxide and sulfone glucokinase activators and methods of use thereof |
| CA3185834A1 (en) * | 2020-06-04 | 2021-12-09 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with hepatic impairment |
| CA3185831A1 (en) * | 2020-06-04 | 2021-12-09 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with renal impairment |
| US11857536B2 (en) | 2020-06-04 | 2024-01-02 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with renal impairment |
| MX2022015525A (es) * | 2020-06-08 | 2023-03-23 | Vtv Therapeutics Llc | Sales o co-cristales del acido {2-[3-ciclohexil-3-(trans-4-propoxi ciclohexil)ureido]tiazol-5-ilsulfanil}acetico y usos de los mismos. |
| WO2021252309A1 (en) * | 2020-06-08 | 2021-12-16 | Vtv Therapeutics Llc | Crystalline forms of {2-[3-cyclohexyl-3-(trans-4-propoxy- cyclohexyl)-ureido]-thiazol-5-ylsulfanyl} -acetic acid and and uses thereof |
| CN115350268B (zh) * | 2022-08-24 | 2025-02-11 | 深圳青澜生物技术有限公司 | 一种用于治疗糖尿病的制剂、微针及其制备工艺 |
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| PL2576524T3 (pl) * | 2010-05-26 | 2018-03-30 | Vtv Therapeutics Llc | Zastosowanie metforminy w skojarzeniu z aktywatorem glukokinazy i kompozycje zawierające metforminę i aktywator glukokinazy |
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| SG11201406987UA (en) | 2012-05-17 | 2014-12-30 | Transtech Pharma Llc | Glucokinase activator compositions for the treatment of diabetes |
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2013
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- 2013-05-15 AU AU2013262895A patent/AU2013262895A1/en not_active Abandoned
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- 2013-05-15 EA EA201492109A patent/EA201492109A1/ru unknown
- 2013-05-15 WO PCT/US2013/041076 patent/WO2013173417A2/en active Application Filing
- 2013-05-15 CN CN201380024802.XA patent/CN104349790A/zh active Pending
- 2013-05-15 CN CN202410499223.0A patent/CN118453592A/zh active Pending
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- 2013-05-15 JP JP2015512779A patent/JP6234443B2/ja active Active
- 2013-05-15 EP EP13726933.8A patent/EP2849776B1/en active Active
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- 2013-05-15 BR BR112014028622A patent/BR112014028622A2/pt not_active Application Discontinuation
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| ES2878001T3 (es) | 2021-11-18 |
| AU2013262895A1 (en) | 2014-11-13 |
| US20200138909A1 (en) | 2020-05-07 |
| SG10201609644UA (en) | 2017-01-27 |
| IN2014DN09554A (en, 2012) | 2015-07-17 |
| WO2013173417A3 (en) | 2014-02-20 |
| SG11201406987UA (en) | 2014-12-30 |
| CN118453592A (zh) | 2024-08-09 |
| MX360304B (es) | 2018-10-29 |
| KR20210027547A (ko) | 2021-03-10 |
| CA2872021A1 (en) | 2013-11-21 |
| JP2015517525A (ja) | 2015-06-22 |
| US20180311314A1 (en) | 2018-11-01 |
| EA201492109A1 (ru) | 2015-07-30 |
| HK1202458A1 (en) | 2015-10-02 |
| JP6234443B2 (ja) | 2017-11-22 |
| AU2017203835B2 (en) | 2018-11-22 |
| MX2014013105A (es) | 2015-04-08 |
| US10980861B2 (en) | 2021-04-20 |
| BR112014028622A2 (pt) | 2017-06-27 |
| EP2849776B1 (en) | 2021-04-21 |
| KR102371364B1 (ko) | 2022-03-07 |
| WO2013173417A2 (en) | 2013-11-21 |
| CN104349790A (zh) | 2015-02-11 |
| US20140066372A1 (en) | 2014-03-06 |
| EP2849776A2 (en) | 2015-03-25 |
| US10588943B2 (en) | 2020-03-17 |
| US10004782B2 (en) | 2018-06-26 |
| IL235484A0 (en) | 2014-12-31 |
| AU2017203835A1 (en) | 2017-06-22 |
| KR20150013838A (ko) | 2015-02-05 |
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