CA2858938C - 2- (pyridin-2yl) - 1, 7 - diaza - spiro [4.4] nonane- 6 - one compound as voltage-gated sodium channels modulator - Google Patents
2- (pyridin-2yl) - 1, 7 - diaza - spiro [4.4] nonane- 6 - one compound as voltage-gated sodium channels modulator Download PDFInfo
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- CA2858938C CA2858938C CA2858938A CA2858938A CA2858938C CA 2858938 C CA2858938 C CA 2858938C CA 2858938 A CA2858938 A CA 2858938A CA 2858938 A CA2858938 A CA 2858938A CA 2858938 C CA2858938 C CA 2858938C
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Landscapes
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| GB1122113.2 | 2011-12-22 | ||
| US61/579,613 | 2011-12-22 | ||
| PCT/GB2012/053233 WO2013093496A1 (en) | 2011-12-22 | 2012-12-21 | 2 - (pyridin- 2yl) - 1, 7 -diaza-spiro [4.4] nonane- 6 -one compound as voltage-gated sodium channels modulator |
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| GB201209015D0 (en) | 2012-05-22 | 2012-07-04 | Convergence Pharmaceuticals | Novel compounds |
| RU2650523C1 (ru) | 2017-07-24 | 2018-04-16 | федеральное государственное автономное образовательное учреждение высшего образования "Казанский (Приволжский) федеральный университет" (ФГАОУ ВО КФУ) | Производное пиридоксина для лечения эпилепсии |
| MX2020003821A (es) * | 2017-10-10 | 2023-01-12 | Biogen Inc | Proceso de elaboración de espiroderivados. |
| KR102349776B1 (ko) | 2017-11-17 | 2022-01-10 | 셀릭스 바이오 프라이빗 리미티드 | 눈 질환의 치료를 위한 조성물 및 방법 |
| CN113563258A (zh) * | 2021-07-29 | 2021-10-29 | 派普医药(江苏)有限公司 | 一种4-溴-2-(二氟甲基)-5-甲基吡啶的制备方法 |
| WO2023044364A1 (en) | 2021-09-15 | 2023-03-23 | Enko Chem, Inc. | Protoporphyrinogen oxidase inhibitors |
| CN118251389A (zh) * | 2021-09-24 | 2024-06-25 | 泽农医药公司 | 作为钠通道活化剂的吡啶基衍生物 |
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| UA57002C2 (uk) | 1995-10-13 | 2003-06-16 | Мерк Фросст Кенада Енд Ко./Мерк Фросст Кенада Енд Сі. | Похідне (метилсульфоніл)феніл-2-(5н)-фуранону, фармацевтична композиція та спосіб лікування |
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| US7505330B2 (en) * | 2006-08-31 | 2009-03-17 | Micron Technology, Inc. | Phase-change random access memory employing read before write for resistance stabilization |
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| JP2010516734A (ja) | 2007-01-24 | 2010-05-20 | グラクソ グループ リミテッド | ３，５−ジアミノ−６−（２，３−ジクロロフェニル）−１，２，４−トリアジンまたはｒ（−）−２，４−ジアミノ−５−（２，３−ジクロロフェニル）−６−フルオロメチルピリミジンを含む医薬組成物 |
| GB0701365D0 (en) | 2007-01-24 | 2007-03-07 | Glaxo Group Ltd | Novel pharmaceutical compositions |
| GB0706630D0 (en) | 2007-04-04 | 2007-05-16 | Glaxo Group Ltd | Novel compounds |
| ES2536694T3 (es) | 2009-09-14 | 2015-05-27 | Convergence Pharmaceuticals Limited | Procedimiento para preparar derivados de alfa-carboxamida |
| MY165579A (en) * | 2009-10-14 | 2018-04-05 | Xenon Pharmaceuticals Inc | Synthetic methods for spiro-oxindole compounds |
| GB201122113D0 (en) * | 2011-12-22 | 2012-02-01 | Convergence Pharmaceuticals | Novel compounds |
| GB201209015D0 (en) | 2012-05-22 | 2012-07-04 | Convergence Pharmaceuticals | Novel compounds |
-
2011
- 2011-12-22 GB GBGB1122113.2A patent/GB201122113D0/en not_active Ceased
-
2012
- 2012-12-21 KR KR1020147019965A patent/KR20140113692A/ko not_active Withdrawn
- 2012-12-21 CA CA2858938A patent/CA2858938C/en active Active
- 2012-12-21 WO PCT/GB2012/053234 patent/WO2013093497A1/en active Application Filing
- 2012-12-21 AU AU2012356386A patent/AU2012356386A1/en not_active Abandoned
- 2012-12-21 SG SG11201403356YA patent/SG11201403356YA/en unknown
- 2012-12-21 JP JP2014548201A patent/JP2015502394A/ja active Pending
- 2012-12-21 CN CN201280070485.0A patent/CN104271581B/zh not_active Expired - Fee Related
- 2012-12-21 BR BR112014014940A patent/BR112014014940A2/pt not_active Application Discontinuation
- 2012-12-21 WO PCT/GB2012/053233 patent/WO2013093496A1/en active Application Filing
- 2012-12-21 EA EA201491251A patent/EA026500B1/ru unknown
- 2012-12-21 ES ES12810416.3T patent/ES2581327T3/es active Active
- 2012-12-21 EP EP12810417.1A patent/EP2794612B1/en not_active Not-in-force
- 2012-12-21 HK HK15103930.0A patent/HK1203492A1/xx unknown
- 2012-12-21 IN IN1469MUN2014 patent/IN2014MN01469A/en unknown
- 2012-12-21 HK HK15104075.3A patent/HK1203501A1/xx unknown
- 2012-12-21 US US14/365,372 patent/US9376436B2/en not_active Expired - Fee Related
- 2012-12-21 JP JP2014548202A patent/JP2015502395A/ja active Pending
- 2012-12-21 EP EP12810416.3A patent/EP2797922B1/en not_active Not-in-force
- 2012-12-21 US US14/365,391 patent/US9303032B2/en not_active Expired - Fee Related
- 2012-12-21 MX MX2014007637A patent/MX2014007637A/es unknown
-
2014
- 2014-06-10 ZA ZA2014/04269A patent/ZA201404269B/en unknown
- 2014-06-18 IL IL233215A patent/IL233215A0/en unknown
-
2016
- 2016-02-25 US US15/053,445 patent/US20160185758A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN104271581A (zh) | 2015-01-07 |
| US20150225400A1 (en) | 2015-08-13 |
| WO2013093497A1 (en) | 2013-06-27 |
| IL233215A0 (en) | 2014-08-31 |
| EA026500B1 (ru) | 2017-04-28 |
| MX2014007637A (es) | 2014-09-26 |
| US9303032B2 (en) | 2016-04-05 |
| US9376436B2 (en) | 2016-06-28 |
| EP2797922B1 (en) | 2016-04-06 |
| ES2581327T3 (es) | 2016-09-05 |
| IN2014MN01469A (forum.php) | 2015-04-17 |
| KR20140113692A (ko) | 2014-09-24 |
| HK1203492A1 (en) | 2015-10-30 |
| US20160185758A1 (en) | 2016-06-30 |
| BR112014014940A2 (pt) | 2017-06-13 |
| CA2858938A1 (en) | 2013-06-27 |
| EA201491251A1 (ru) | 2014-11-28 |
| AU2012356386A1 (en) | 2014-07-10 |
| US20140350040A1 (en) | 2014-11-27 |
| CN104271581B (zh) | 2016-08-31 |
| GB201122113D0 (en) | 2012-02-01 |
| JP2015502395A (ja) | 2015-01-22 |
| ZA201404269B (en) | 2016-06-29 |
| WO2013093496A1 (en) | 2013-06-27 |
| EP2797922A1 (en) | 2014-11-05 |
| HK1203501A1 (en) | 2015-10-30 |
| SG11201403356YA (en) | 2014-07-30 |
| JP2015502394A (ja) | 2015-01-22 |
| EP2794612B1 (en) | 2016-04-06 |
| EP2794612A1 (en) | 2014-10-29 |
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