CA2858778A1 - Process for the preparation of 2-phenyl-[1,2,4]triazolo[1,5-a]pyridine derivatives - Google Patents

Process for the preparation of 2-phenyl-[1,2,4]triazolo[1,5-a]pyridine derivatives Download PDF

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Publication number
CA2858778A1
CA2858778A1 CA2858778A CA2858778A CA2858778A1 CA 2858778 A1 CA2858778 A1 CA 2858778A1 CA 2858778 A CA2858778 A CA 2858778A CA 2858778 A CA2858778 A CA 2858778A CA 2858778 A1 CA2858778 A1 CA 2858778A1
Authority
CA
Canada
Prior art keywords
pyridine
triazolo
mmol
formula
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2858778A
Other languages
English (en)
French (fr)
Inventor
Bjoern Bartels
Serena Maria FANTASIA
Alexander Flohr
Kurt Puentener
Shaoning Wang
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of CA2858778A1 publication Critical patent/CA2858778A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
CA2858778A 2012-02-09 2013-02-07 Process for the preparation of 2-phenyl-[1,2,4]triazolo[1,5-a]pyridine derivatives Abandoned CA2858778A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP12154786 2012-02-09
EP12154786.3 2012-02-09
PCT/EP2013/052362 WO2013117610A1 (en) 2012-02-09 2013-02-07 Process for the preparation of 2-phenyl-[1,2,4]triazolo[1,5-a]pyridine derivatives

Publications (1)

Publication Number Publication Date
CA2858778A1 true CA2858778A1 (en) 2013-08-15

Family

ID=47664298

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2858778A Abandoned CA2858778A1 (en) 2012-02-09 2013-02-07 Process for the preparation of 2-phenyl-[1,2,4]triazolo[1,5-a]pyridine derivatives

Country Status (11)

Country Link
US (1) US9115130B2 (en:Method)
EP (1) EP2812330B1 (en:Method)
JP (1) JP6122034B2 (en:Method)
KR (1) KR20140128998A (en:Method)
CN (1) CN104093718B (en:Method)
BR (1) BR112014016427A8 (en:Method)
CA (1) CA2858778A1 (en:Method)
ES (1) ES2558618T3 (en:Method)
MX (1) MX348447B (en:Method)
RU (1) RU2620379C2 (en:Method)
WO (1) WO2013117610A1 (en:Method)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20170032329A (ko) 2014-07-30 2017-03-22 모찌다 세이야쿠 가부시끼가이샤 피라졸 유도체의 제조 방법
JP6568855B2 (ja) * 2014-07-30 2019-08-28 持田製薬株式会社 ピラゾール誘導体の製造方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4358454A (en) * 1982-01-08 1982-11-09 Schering Corporation 1,3,4-Triazolo[1,5-a]pyridines
JP4101755B2 (ja) * 2001-10-08 2008-06-18 エフ．ホフマン−ラ ロシュ アーゲー ８−アミノ−〔１，２，４〕トリアゾロ〔１，５−ａ〕ピリジン−６−カルボン酸アミド
JP2011032225A (ja) * 2009-08-03 2011-02-17 Gifu Ichi １，２，４−トリアゾール誘導体の製造方法
US8349824B2 (en) * 2010-12-07 2013-01-08 Hoffmann-La Roche Inc. Triazolopyridine compounds

Also Published As

Publication number Publication date
US9115130B2 (en) 2015-08-25
RU2620379C2 (ru) 2017-05-25
EP2812330A1 (en) 2014-12-17
WO2013117610A1 (en) 2013-08-15
US20140350259A1 (en) 2014-11-27
MX348447B (es) 2017-06-13
BR112014016427A8 (pt) 2017-07-04
RU2014134278A (ru) 2016-03-27
BR112014016427A2 (pt) 2017-06-13
CN104093718B (zh) 2016-05-04
JP2015511235A (ja) 2015-04-16
KR20140128998A (ko) 2014-11-06
JP6122034B2 (ja) 2017-04-26
CN104093718A (zh) 2014-10-08
MX2014008814A (es) 2014-10-24
ES2558618T3 (es) 2016-02-05
EP2812330B1 (en) 2015-12-02
HK1197244A1 (zh) 2015-01-09

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Legal Events

Date Code Title Description
EEER Examination request

Effective date: 20180206

FZDE Discontinued

Effective date: 20200831