CA2821827A1 - 6-thio-substituted imidazopyrazines for use as mps-1 and tkk inhibitors in the treatment of hyperproliferative disorders - Google Patents
6-thio-substituted imidazopyrazines for use as mps-1 and tkk inhibitors in the treatment of hyperproliferative disorders Download PDFInfo
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- CA2821827A1 CA2821827A1 CA2821827A CA2821827A CA2821827A1 CA 2821827 A1 CA2821827 A1 CA 2821827A1 CA 2821827 A CA2821827 A CA 2821827A CA 2821827 A CA2821827 A CA 2821827A CA 2821827 A1 CA2821827 A1 CA 2821827A1
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- alkyl
- alkoxy
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| PCT/EP2011/072582 WO2012080228A1 (en) | 2010-12-17 | 2011-12-13 | 6-thio-substituted imidazopyrazines for use as mps-1 and tkk inhibitors in the treatment of hyperproliferative disorders |
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| CN102413831B (zh) | 2009-04-29 | 2014-06-04 | 拜耳知识产权有限责任公司 | 取代的咪唑并喹喔啉 |
| TW201107329A (en) | 2009-07-30 | 2011-03-01 | Oncotherapy Science Inc | Fused imidazole derivative having ttk inhibitory action |
| CA2772790C (en) | 2009-09-04 | 2017-06-27 | Benjamin Bader | Substituted aminoquinoxalines as tyrosine threonine kinase inhibitors |
| EP2343294A1 (en) | 2009-11-30 | 2011-07-13 | Bayer Schering Pharma AG | Substituted triazolopyridines |
| EP2343295A1 (en) | 2009-11-30 | 2011-07-13 | Bayer Schering Pharma AG | Triazolopyridine derivates |
| EP2343297A1 (en) | 2009-11-30 | 2011-07-13 | Bayer Schering Pharma AG | Triazolopyridines |
| ES2555261T3 (es) * | 2010-06-01 | 2015-12-30 | Bayer Intellectual Property Gmbh | Imidazopirazinas sustituidas |
| ES2530802T3 (es) * | 2010-12-17 | 2015-03-06 | Bayer Ip Gmbh | Imidazopirazinas 6-tiosustituidas para uso como inhibidores de MPS-1 y TKK en el tratamiento de trastornos hiperproliferativos |
-
2011
- 2011-12-13 ES ES11796994T patent/ES2530802T3/es active Active
- 2011-12-13 JP JP2013543703A patent/JP5964853B2/ja not_active Expired - Fee Related
- 2011-12-13 US US13/995,055 patent/US9212184B2/en not_active Expired - Fee Related
- 2011-12-13 CN CN201180067336.4A patent/CN103403006B/zh not_active Expired - Fee Related
- 2011-12-13 EP EP11796994.9A patent/EP2651947B1/en not_active Not-in-force
- 2011-12-13 WO PCT/EP2011/072582 patent/WO2012080228A1/en not_active Ceased
- 2011-12-13 CA CA2821827A patent/CA2821827A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| JP5964853B2 (ja) | 2016-08-03 |
| EP2651947A1 (en) | 2013-10-23 |
| CN103403006B (zh) | 2015-11-25 |
| ES2530802T3 (es) | 2015-03-06 |
| US20130281460A1 (en) | 2013-10-24 |
| EP2651947B1 (en) | 2014-12-10 |
| JP2013545775A (ja) | 2013-12-26 |
| US9212184B2 (en) | 2015-12-15 |
| CN103403006A (zh) | 2013-11-20 |
| WO2012080228A1 (en) | 2012-06-21 |
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