CA2793391A1 - Arylsulfonamide ccr3 antagonists - Google Patents
Arylsulfonamide ccr3 antagonists Download PDFInfo
- Publication number
- CA2793391A1 CA2793391A1 CA2793391A CA2793391A CA2793391A1 CA 2793391 A1 CA2793391 A1 CA 2793391A1 CA 2793391 A CA2793391 A CA 2793391A CA 2793391 A CA2793391 A CA 2793391A CA 2793391 A1 CA2793391 A1 CA 2793391A1
- Authority
- CA
- Canada
- Prior art keywords
- alkyl
- optionally substituted
- halo
- hydrogen
- nr1b
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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- 239000005557 antagonist Substances 0.000 title description 8
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Classifications
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US31497110P | 2010-03-17 | 2010-03-17 | |
| US61/314,971 | 2010-03-17 | ||
| PCT/US2011/028771 WO2011116161A2 (en) | 2010-03-17 | 2011-03-17 | Arylsulfonamide ccr3 antagonists |
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| Publication Number | Publication Date |
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| CA2793391A1 true CA2793391A1 (en) | 2011-09-22 |
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| CA2793391A Abandoned CA2793391A1 (en) | 2010-03-17 | 2011-03-17 | Arylsulfonamide ccr3 antagonists |
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| WO (1) | WO2011116161A2 (enExample) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA05010055A (es) | 2003-03-24 | 2005-11-23 | Actimis Pharmaceuticals Inc | Derivados de 2-fenoxi- y 2-fenil-sulfomamida con actividad antagonista del ccr3, para el tratamiento del asma y otros desordenes inflamatorios o inmunologicos. |
| AU2010239340B2 (en) | 2009-04-22 | 2015-07-02 | Axikin Pharmaceuticals, Inc. | 2,5-disubstituted arylsulfonamide CCR3 antagonists |
| US8946197B2 (en) | 2009-11-16 | 2015-02-03 | Chdi Foundation, Inc. | Transglutaminase TG2 inhibitors, pharmaceutical compositions, and methods of use thereof |
| CA2814011A1 (en) * | 2010-10-11 | 2012-04-19 | Axikin Pharmaceuticals, Inc. | Salts of arylsulfonamide ccr3 antagonists |
| US8889716B2 (en) | 2011-05-10 | 2014-11-18 | Chdi Foundation, Inc. | Transglutaminase TG2 inhibitors, pharmaceutical compositions, and methods of use thereof |
| AU2013312420A1 (en) | 2012-09-07 | 2015-02-26 | Axikin Pharmaceuticals, Inc. | Isotopically enriched arylsulfonamide CCR3 antagonists |
| WO2014075124A1 (en) * | 2012-11-15 | 2014-05-22 | Victoria University | Methods and compositions for the treatment and/or prevention of bowel disorders |
| TWI763668B (zh) * | 2016-05-05 | 2022-05-11 | 美商嘉來克生命科學有限責任公司 | 整合應激途徑之調節劑 |
| CN119490205B (zh) * | 2025-01-14 | 2025-04-22 | 莱州诚源盐化有限公司 | 一种离子膜法氯碱生产专用工业盐的制备方法 |
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-
2011
- 2011-03-17 EP EP11715094.6A patent/EP2547655B1/en not_active Not-in-force
- 2011-03-17 CN CN2011800243474A patent/CN102892754A/zh active Pending
- 2011-03-17 WO PCT/US2011/028771 patent/WO2011116161A2/en not_active Ceased
- 2011-03-17 MX MX2012010714A patent/MX336559B/es unknown
- 2011-03-17 CA CA2793391A patent/CA2793391A1/en not_active Abandoned
- 2011-03-17 AR ARP110100873A patent/AR080770A1/es unknown
- 2011-03-17 US US13/050,831 patent/US8741894B2/en not_active Expired - Fee Related
- 2011-03-17 AU AU2011227232A patent/AU2011227232B2/en not_active Ceased
- 2011-03-17 JP JP2013500199A patent/JP5818873B2/ja not_active Expired - Fee Related
- 2011-03-17 TW TW100109234A patent/TW201134820A/zh unknown
-
2012
- 2012-09-19 IL IL222000A patent/IL222000A0/en unknown
-
2014
- 2014-04-22 US US14/258,906 patent/US20140221428A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| JP5818873B2 (ja) | 2015-11-18 |
| WO2011116161A3 (en) | 2012-04-19 |
| CN102892754A (zh) | 2013-01-23 |
| MX2012010714A (es) | 2013-01-29 |
| AU2011227232A1 (en) | 2012-10-11 |
| WO2011116161A2 (en) | 2011-09-22 |
| AR080770A1 (es) | 2012-05-09 |
| TW201134820A (en) | 2011-10-16 |
| US20110230487A1 (en) | 2011-09-22 |
| US8741894B2 (en) | 2014-06-03 |
| EP2547655B1 (en) | 2016-03-09 |
| AU2011227232B2 (en) | 2015-07-09 |
| EP2547655A2 (en) | 2013-01-23 |
| JP2013522316A (ja) | 2013-06-13 |
| IL222000A0 (en) | 2012-12-02 |
| US20140221428A1 (en) | 2014-08-07 |
| MX336559B (es) | 2016-01-25 |
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