CA2789606A1 - Analogues peptidiques en tant qu'agonistes des recepteurs opioides - Google Patents

Analogues peptidiques en tant qu'agonistes des recepteurs opioides Download PDF

Info

Publication number
CA2789606A1
CA2789606A1 CA2789606A CA2789606A CA2789606A1 CA 2789606 A1 CA2789606 A1 CA 2789606A1 CA 2789606 A CA2789606 A CA 2789606A CA 2789606 A CA2789606 A CA 2789606A CA 2789606 A1 CA2789606 A1 CA 2789606A1
Authority
CA
Canada
Prior art keywords
compound
pain
formula
preparation
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2789606A
Other languages
English (en)
Inventor
Christopher Gordon Barber
Dafydd Rhys Owen
Lisa Rosemary Thompson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Ltd
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of CA2789606A1 publication Critical patent/CA2789606A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
CA2789606A 2010-02-25 2011-02-11 Analogues peptidiques en tant qu'agonistes des recepteurs opioides Abandoned CA2789606A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US30799310P 2010-02-25 2010-02-25
US61/307,993 2010-02-25
PCT/IB2011/050580 WO2011104649A1 (fr) 2010-02-25 2011-02-11 Analogues peptidiques

Publications (1)

Publication Number Publication Date
CA2789606A1 true CA2789606A1 (fr) 2011-09-01

Family

ID=43778553

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2789606A Abandoned CA2789606A1 (fr) 2010-02-25 2011-02-11 Analogues peptidiques en tant qu'agonistes des recepteurs opioides

Country Status (8)

Country Link
US (2) US20110207654A1 (fr)
EP (1) EP2539358A1 (fr)
JP (1) JP2013520489A (fr)
AR (1) AR080297A1 (fr)
CA (1) CA2789606A1 (fr)
TW (1) TW201138763A (fr)
UY (1) UY33240A (fr)
WO (1) WO2011104649A1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2564366T3 (es) * 2011-07-13 2016-03-22 Pfizer Limited Análogos de encefalina
CN103793181B (zh) * 2012-11-05 2019-05-24 腾讯科技（深圳）有限公司 一种多层关联存储架构的数据同步方法及数据同步系统

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58146507A (ja) * 1982-02-24 1983-09-01 Asai Gerumaniumu Kenkyusho:Kk モルヒネ様作用増強剤
ZA851181B (en) * 1984-02-16 1986-04-30 Searle & Co Substituted tyrosyl alanine dipeptide amides
KR0166088B1 (ko) 1990-01-23 1999-01-15 . 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도
US5376645A (en) 1990-01-23 1994-12-27 University Of Kansas Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof
WO1994011018A1 (fr) * 1992-11-12 1994-05-26 Biomeasure, Inc. Peptides opioides
SE9600769D0 (sv) * 1996-02-28 1996-02-28 Astra Ab Compounds useful as analgesic
SE9701718D0 (sv) * 1997-05-07 1997-05-07 Astra Ab Analgesic peptidomimetic compounds
GB9711643D0 (en) 1997-06-05 1997-07-30 Janssen Pharmaceutica Nv Glass thermoplastic systems
US6114310A (en) 1998-01-23 2000-09-05 Microcide Pharmaceuticals, Inc. Efflux pump inhibitors
ES2357340T3 (es) 2006-10-18 2011-04-25 Pfizer Products Inc. Compuestos de biaril éter urea.
CL2008000835A1 (es) 2007-03-23 2008-10-03 Icagen Inc Pfizer Ltd Compuestos derivados de sulfonamidas, inhibidores de los canales de calcio; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento del dolor, sindrome de intestino irritable, enfermedad de crohn, taquiarritm
WO2008135826A2 (fr) 2007-05-03 2008-11-13 Pfizer Limited Dérivés de la pyridine
US8124610B2 (en) 2007-07-13 2012-02-28 Icagen Inc. Sodium channel inhibitors
PT2385938E (pt) 2009-01-12 2015-06-02 Pfizer Ltd Derivados de sulfonamida

Also Published As

Publication number Publication date
US20120329724A1 (en) 2012-12-27
AR080297A1 (es) 2012-03-28
TW201138763A (en) 2011-11-16
UY33240A (es) 2011-09-30
US20110207654A1 (en) 2011-08-25
WO2011104649A1 (fr) 2011-09-01
US8598123B2 (en) 2013-12-03
JP2013520489A (ja) 2013-06-06
EP2539358A1 (fr) 2013-01-02

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued

Effective date: 20170213