UY33240A - ?análogos de péptidos?. - Google Patents

?análogos de péptidos?.

Info

Publication number
UY33240A
UY33240A UY0001033240A UY33240A UY33240A UY 33240 A UY33240 A UY 33240A UY 0001033240 A UY0001033240 A UY 0001033240A UY 33240 A UY33240 A UY 33240A UY 33240 A UY33240 A UY 33240A
Authority
UY
Uruguay
Prior art keywords
analogs
peptides
substituents
medicine
compounds
Prior art date
Application number
UY0001033240A
Other languages
English (en)
Inventor
Christopher Gordon Barber
Dafydd Rhys Owen
Lisa Rosemary Thompson
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of UY33240A publication Critical patent/UY33240A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pain & Pain Management (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a compuestos de Fórmula (I). y a sus sales farmacéuticamente aceptables, en la que los sustituyentes son como se han descrito en el presente documento, y su uso en medicina, en particular como agonistas opioides.
UY0001033240A 2010-02-25 2011-02-24 ?análogos de péptidos?. UY33240A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US30799310P 2010-02-25 2010-02-25

Publications (1)

Publication Number Publication Date
UY33240A true UY33240A (es) 2011-09-30

Family

ID=43778553

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001033240A UY33240A (es) 2010-02-25 2011-02-24 ?análogos de péptidos?.

Country Status (8)

Country Link
US (2) US20110207654A1 (es)
EP (1) EP2539358A1 (es)
JP (1) JP2013520489A (es)
AR (1) AR080297A1 (es)
CA (1) CA2789606A1 (es)
TW (1) TW201138763A (es)
UY (1) UY33240A (es)
WO (1) WO2011104649A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013008123A1 (en) * 2011-07-13 2013-01-17 Pfizer Limited Enkephalin analogues
CN103793181B (zh) * 2012-11-05 2019-05-24 腾讯科技（深圳）有限公司 一种多层关联存储架构的数据同步方法及数据同步系统

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58146507A (ja) * 1982-02-24 1983-09-01 Asai Gerumaniumu Kenkyusho:Kk モルヒネ様作用増強剤
ES8606404A1 (es) * 1984-02-16 1986-04-16 Searle & Co Amidas dipeptidas analgesicas o antihipertensivas
US5376645A (en) 1990-01-23 1994-12-27 University Of Kansas Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof
KR0166088B1 (ko) 1990-01-23 1999-01-15 . 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도
JPH07503485A (ja) * 1992-11-12 1995-04-13 バイオメジャー　インコーポレイテッド オピオイドペプチド
SE9600769D0 (sv) * 1996-02-28 1996-02-28 Astra Ab Compounds useful as analgesic
SE9701718D0 (sv) * 1997-05-07 1997-05-07 Astra Ab Analgesic peptidomimetic compounds
GB9711643D0 (en) 1997-06-05 1997-07-30 Janssen Pharmaceutica Nv Glass thermoplastic systems
US6114310A (en) 1998-01-23 2000-09-05 Microcide Pharmaceuticals, Inc. Efflux pump inhibitors
DE602007011793D1 (de) 2006-10-18 2011-02-17 Pfizer Prod Inc Biaryl-ether-harnstoffverbindungen
US8357711B2 (en) 2007-03-23 2013-01-22 Pfizer Limited Heterocyclic sulfonamides as inhibitors of ion channels
EA015952B1 (ru) 2007-05-03 2011-12-30 Пфайзер Лимитед 2-пиридинкарбоксамидные производные в качестве модуляторов натриевых каналов
EP2173743A2 (en) 2007-07-13 2010-04-14 Icagen, Inc. Sodium channel inhibitors
GEP20135992B (en) 2009-01-12 2013-12-25 Icagen Inc Sulfonamide derivatives

Also Published As

Publication number Publication date
CA2789606A1 (en) 2011-09-01
TW201138763A (en) 2011-11-16
EP2539358A1 (en) 2013-01-02
WO2011104649A1 (en) 2011-09-01
US8598123B2 (en) 2013-12-03
US20120329724A1 (en) 2012-12-27
AR080297A1 (es) 2012-03-28
JP2013520489A (ja) 2013-06-06
US20110207654A1 (en) 2011-08-25

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Legal Events

Date Code Title Description
DESI Application deemed to be withdrawn

Effective date: 20121113