CA2735286C - Fused pyrrolidino-cyclopropane derivatives as selective 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors - Google Patents
Fused pyrrolidino-cyclopropane derivatives as selective 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors Download PDFInfo
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- CA2735286C CA2735286C CA2735286A CA2735286A CA2735286C CA 2735286 C CA2735286 C CA 2735286C CA 2735286 A CA2735286 A CA 2735286A CA 2735286 A CA2735286 A CA 2735286A CA 2735286 C CA2735286 C CA 2735286C
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| Application Number | Priority Date | Filing Date | Title |
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| EP08290822.9 | 2008-09-01 | ||
| EP08290822 | 2008-09-01 | ||
| PCT/EP2009/005654 WO2010022850A1 (en) | 2008-09-01 | 2009-08-05 | Fused pyrrolidino-cyclopropane derivatives as selective 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors |
Publications (2)
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| CA2735286A1 CA2735286A1 (en) | 2010-03-04 |
| CA2735286C true CA2735286C (en) | 2017-12-05 |
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| CA2735286A Active CA2735286C (en) | 2008-09-01 | 2009-08-05 | Fused pyrrolidino-cyclopropane derivatives as selective 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors |
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| US9580422B2 (en) * | 2013-10-22 | 2017-02-28 | Bristol-Myers Squibb Company | Isotopically labeled triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors |
| MA40759A (fr) | 2014-09-26 | 2017-08-01 | Pfizer | Modulateurs de rorc2 de type pyrrolopyridine substitué par un méthyle et trifluorométhyle et leurs procédés d'utilisation |
| EP3235813A1 (en) | 2016-04-19 | 2017-10-25 | Cidqo 2012, S.L. | Aza-tetra-cyclo derivatives |
| CA3243547A1 (en) * | 2021-12-21 | 2023-06-29 | Corcept Therapeutics Inc | INDAZOLE GLUCOCORTICOID RECEPTOR BICYCLIC ANTAGONISTS |
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| US4088652A (en) * | 1975-07-31 | 1978-05-09 | American Cyanamid Company | Acylazabicyclohexanes |
| AU2003287909A1 (en) * | 2003-01-08 | 2004-08-10 | Mibitech Aps | Electro-therapeutic device and method of electro-therapeutic treatment |
| US7700583B2 (en) | 2003-04-11 | 2010-04-20 | High Point Pharmaceuticals, Llc | 11β-hydroxysteroid dehydrogenase type 1 active compounds |
| EP1615698B1 (en) * | 2003-04-11 | 2010-09-29 | High Point Pharmaceuticals, LLC | New amide derivatives and pharmaceutical use thereof |
| WO2006106423A2 (en) * | 2005-04-07 | 2006-10-12 | Pfizer Inc. | Amino sulfonyl derivatives as inhibitors of human 11-.beta.-hydrosysteroid dehydrogenase |
| EP1971614A1 (en) * | 2005-11-14 | 2008-09-24 | Probiodrug AG | Cyclopropyl-fused pyrrolidine derivatives as dipeptidyl peptidase iv inhibitors |
| GB0625198D0 (en) | 2006-12-18 | 2007-01-24 | Glaxo Group Ltd | Chemical compounds |
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| EA020238B1 (ru) | 2014-09-30 |
| BRPI0918288A2 (pt) | 2015-12-22 |
| EP2321317A1 (en) | 2011-05-18 |
| CN102137864B (zh) | 2014-12-31 |
| BRPI0918288B1 (pt) | 2018-11-06 |
| AU2009287118B2 (en) | 2014-02-27 |
| EA201100419A1 (ru) | 2011-10-31 |
| US20110172265A1 (en) | 2011-07-14 |
| JP2012501302A (ja) | 2012-01-19 |
| KR101707580B1 (ko) | 2017-02-16 |
| CA2735286A1 (en) | 2010-03-04 |
| AU2009287118A1 (en) | 2010-03-04 |
| IL211447A (en) | 2014-07-31 |
| US8486964B2 (en) | 2013-07-16 |
| CN102137864A (zh) | 2011-07-27 |
| WO2010022850A1 (en) | 2010-03-04 |
| MX2011002181A (es) | 2011-03-30 |
| IL211447A0 (en) | 2011-05-31 |
| JP5579717B2 (ja) | 2014-08-27 |
| EP2321317B1 (en) | 2014-12-24 |
| AU2009287118B9 (en) | 2014-08-07 |
| AR073224A1 (es) | 2010-10-20 |
| KR20110059749A (ko) | 2011-06-03 |
| ZA201102418B (en) | 2011-12-28 |
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Effective date: 20140801 |