CA2724008A1 - Fused pyrimidine derivatives as trpv3 modulators - Google Patents

Fused pyrimidine derivatives as trpv3 modulators Download PDF

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Publication number
CA2724008A1
CA2724008A1 CA2724008A CA2724008A CA2724008A1 CA 2724008 A1 CA2724008 A1 CA 2724008A1 CA 2724008 A CA2724008 A CA 2724008A CA 2724008 A CA2724008 A CA 2724008A CA 2724008 A1 CA2724008 A1 CA 2724008A1
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CA
Canada
Prior art keywords
substituted
unsubstituted
compound
pyrido
pyrimidin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2724008A
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English (en)
French (fr)
Inventor
Prasada Rao V.S. LINGAM
Abraham Thomas
Dattaguru Anandrao More
Javed Yusuf Khatik
Neelima Khairatkar-Joshi
Vidya Ganapati Kattige
Original Assignee
Glenmark Pharmaceuticals SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glenmark Pharmaceuticals SA filed Critical Glenmark Pharmaceuticals SA
Publication of CA2724008A1 publication Critical patent/CA2724008A1/en
Abandoned legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
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  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Anesthesiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
CA2724008A 2008-01-11 2009-01-07 Fused pyrimidine derivatives as trpv3 modulators Abandoned CA2724008A1 (en)

Applications Claiming Priority (11)

Application Number Priority Date Filing Date Title
IN82MU2008 2008-01-11
IN82/MUM/2008 2008-01-11
US2877008P 2008-02-14 2008-02-14
US61/028,770 2008-02-14
IN548/MUM/2008 2008-03-18
IN548MU2008 2008-03-18
IN798MU2008 2008-04-04
IN798/MUM/2008 2008-04-04
US4827608P 2008-04-28 2008-04-28
US61/048,276 2008-04-28
PCT/IN2009/000025 WO2009109987A2 (en) 2008-01-11 2009-01-07 Fused pyrimidine derivatives as trpv3 modulators

Publications (1)

Publication Number Publication Date
CA2724008A1 true CA2724008A1 (en) 2009-09-11

Family

ID=41056428

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2724008A Abandoned CA2724008A1 (en) 2008-01-11 2009-01-07 Fused pyrimidine derivatives as trpv3 modulators

Country Status (10)

Country Link
US (1) US8349846B2 (https=)
EP (1) EP2229388A4 (https=)
JP (1) JP5419894B2 (https=)
AU (1) AU2009220825A1 (https=)
CA (1) CA2724008A1 (https=)
EA (1) EA018133B1 (https=)
GE (1) GEP20125574B (https=)
MX (1) MX2010005769A (https=)
NZ (1) NZ595781A (https=)
WO (1) WO2009109987A2 (https=)

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US8119647B2 (en) * 2008-04-23 2012-02-21 Glenmark Pharmaceuticals S.A. Fused pyrimidineone compounds as TRPV3 modulators
JP2012514577A (ja) 2008-12-26 2012-06-28 グレンマーク ファーマシューティカルズ， エセ．アー． Ｔｒｐｖ３アンタゴニストとしての縮合イミダゾール誘導体
SG11201406818VA (en) * 2012-04-23 2014-11-27 Genentech Inc Intermediates and processes for preparing compounds
AU2020391161A1 (en) 2019-11-25 2022-06-09 Amgen Inc. Heterocyclic compounds as Delta-5 Desaturase inhibitors and methods of use

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US20100292254A1 (en) 2010-11-18
EP2229388A4 (en) 2012-03-07
AU2009220825A2 (en) 2012-04-19
JP2011509288A (ja) 2011-03-24
EA018133B1 (ru) 2013-05-30
JP5419894B2 (ja) 2014-02-19
NZ595781A (en) 2013-07-26
MX2010005769A (es) 2010-11-12
WO2009109987A3 (en) 2009-12-17
WO2009109987A2 (en) 2009-09-11
EA201000674A1 (ru) 2011-02-28
GEP20125574B (en) 2012-07-10
US8349846B2 (en) 2013-01-08
AU2009220825A1 (en) 2012-01-19
EP2229388A2 (en) 2010-09-22

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