GEP20125574B - Fused pyrimidine derivatives as trpv3 modulators - Google Patents

Fused pyrimidine derivatives as trpv3 modulators

Info

Publication number
GEP20125574B
GEP20125574B GEAP200911911A GEAP2009011911A GEP20125574B GE P20125574 B GEP20125574 B GE P20125574B GE AP200911911 A GEAP200911911 A GE AP200911911A GE AP2009011911 A GEAP2009011911 A GE AP2009011911A GE P20125574 B GEP20125574 B GE P20125574B
Authority
GE
Georgia
Prior art keywords
pyrimidine derivatives
fused pyrimidine
trpv3
trpv3 modulators
modulators
Prior art date
Application number
GEAP200911911A
Other languages
English (en)
Inventor
V S Prasadarao Lingam
Abraham Thomas
Joshi Neelima Khairatkar
Dattaguru Anandrao More
Javed Yusuf Khatik
Vidya Ganapati Kattige
Original Assignee
Glenmark Pharmaceuticals Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glenmark Pharmaceuticals Sa filed Critical Glenmark Pharmaceuticals Sa
Publication of GEP20125574B publication Critical patent/GEP20125574B/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Anesthesiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Psychology (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
GEAP200911911A 2008-01-11 2009-01-07 Fused pyrimidine derivatives as trpv3 modulators GEP20125574B (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN82MU2008 2008-01-11
US2877008P 2008-02-14 2008-02-14
IN548MU2008 2008-03-18
IN798MU2008 2008-04-04
US4827608P 2008-04-28 2008-04-28

Publications (1)

Publication Number Publication Date
GEP20125574B true GEP20125574B (en) 2012-07-10

Family

ID=41056428

Family Applications (1)

Application Number Title Priority Date Filing Date
GEAP200911911A GEP20125574B (en) 2008-01-11 2009-01-07 Fused pyrimidine derivatives as trpv3 modulators

Country Status (10)

Country Link
US (1) US8349846B2 (https=)
EP (1) EP2229388A4 (https=)
JP (1) JP5419894B2 (https=)
AU (1) AU2009220825A1 (https=)
CA (1) CA2724008A1 (https=)
EA (1) EA018133B1 (https=)
GE (1) GEP20125574B (https=)
MX (1) MX2010005769A (https=)
NZ (1) NZ595781A (https=)
WO (1) WO2009109987A2 (https=)

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US8119647B2 (en) * 2008-04-23 2012-02-21 Glenmark Pharmaceuticals S.A. Fused pyrimidineone compounds as TRPV3 modulators
AU2009332651A1 (en) * 2008-12-26 2011-12-01 Glenmark Pharmaceuticals, S.A. Fused imidazole derivatives as TRPV3 antagonist
AR090789A1 (es) * 2012-04-23 2014-12-10 Genentech Inc Intermediarios y procesos para la preparacion de compuestos
JP7638987B2 (ja) 2019-11-25 2025-03-04 アムジエン・インコーポレーテツド デルタ－５デサチュラーゼ阻害剤としての複素環式化合物、及び使用法

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Also Published As

Publication number Publication date
EA201000674A1 (ru) 2011-02-28
EP2229388A2 (en) 2010-09-22
CA2724008A1 (en) 2009-09-11
AU2009220825A2 (en) 2012-04-19
JP5419894B2 (ja) 2014-02-19
WO2009109987A3 (en) 2009-12-17
EA018133B1 (ru) 2013-05-30
MX2010005769A (es) 2010-11-12
WO2009109987A2 (en) 2009-09-11
US8349846B2 (en) 2013-01-08
US20100292254A1 (en) 2010-11-18
NZ595781A (en) 2013-07-26
AU2009220825A1 (en) 2012-01-19
JP2011509288A (ja) 2011-03-24
EP2229388A4 (en) 2012-03-07

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