CA2718608A1 - Solid forms of an anti-hiv phosphoindole compound - Google Patents

Solid forms of an anti-hiv phosphoindole compound Download PDF

Info

Publication number
CA2718608A1
CA2718608A1 CA2718608A CA2718608A CA2718608A1 CA 2718608 A1 CA2718608 A1 CA 2718608A1 CA 2718608 A CA2718608 A CA 2718608A CA 2718608 A CA2718608 A CA 2718608A CA 2718608 A1 CA2718608 A1 CA 2718608A1
Authority
CA
Canada
Prior art keywords
crystal form
viii
exhibits
ray powder
powder diffraction
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2718608A
Other languages
English (en)
French (fr)
Inventor
Adel M. Moussa
Mike H. O'neill
Xiaohong Sheng
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Idenix Pharmaceuticals LLC
Original Assignee
Idenix Pharmaceuticals LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idenix Pharmaceuticals LLC filed Critical Idenix Pharmaceuticals LLC
Publication of CA2718608A1 publication Critical patent/CA2718608A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/572—Five-membered rings
    • C07F9/5728—Five-membered rings condensed with carbocyclic rings or carbocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CA2718608A 2008-03-27 2009-03-27 Solid forms of an anti-hiv phosphoindole compound Abandoned CA2718608A1 (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US7234908P 2008-03-27 2008-03-27
US61/072,349 2008-03-27
US4384108P 2008-04-10 2008-04-10
US61/043,841 2008-04-10
US15586909P 2009-02-26 2009-02-26
US61/155,869 2009-02-26
PCT/US2009/038479 WO2009120914A1 (en) 2008-03-27 2009-03-27 Solid forms of an anti-hiv phosphoindole compound

Publications (1)

Publication Number Publication Date
CA2718608A1 true CA2718608A1 (en) 2009-10-01

Family

ID=40791117

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2718608A Abandoned CA2718608A1 (en) 2008-03-27 2009-03-27 Solid forms of an anti-hiv phosphoindole compound

Country Status (9)

Country Link
US (1) US8470870B2 (enExample)
EP (1) EP2276771A1 (enExample)
JP (1) JP2011515498A (enExample)
AU (1) AU2009228150A1 (enExample)
BR (1) BRPI0910241A2 (enExample)
CA (1) CA2718608A1 (enExample)
MX (1) MX2010010455A (enExample)
TW (1) TW200946541A (enExample)
WO (1) WO2009120914A1 (enExample)

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CN105939723B (zh) 2013-12-17 2020-02-28 珍白斯凯尔有限公司 前列腺癌治疗用组合物
KR102413243B1 (ko) 2014-12-23 2022-06-27 주식회사 젬백스앤카엘 안질환 치료 펩티드 및 이를 포함하는 안질환 치료용 조성물
JP6751097B2 (ja) 2015-02-27 2020-09-02 ジェムバックス アンド カエル カンパニー，リミティド 聴力損傷予防用ペプチド及びそれを含む組成物
CN107847551B (zh) 2015-07-02 2022-02-08 珍白斯凯尔有限公司 具有抗病毒作用的肽和包含其的组合物
CN109328068A (zh) 2016-04-07 2019-02-12 珍白斯凯尔有限公司 具有增加端粒酶活性和延长端粒的效果的肽以及包含该肽的组合物

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Also Published As

Publication number Publication date
MX2010010455A (es) 2011-03-21
US20110039803A1 (en) 2011-02-17
TW200946541A (en) 2009-11-16
EP2276771A1 (en) 2011-01-26
AU2009228150A1 (en) 2009-10-01
US8470870B2 (en) 2013-06-25
BRPI0910241A2 (pt) 2015-09-29
JP2011515498A (ja) 2011-05-19
WO2009120914A1 (en) 2009-10-01

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Legal Events

Date Code Title Description
EEER Examination request

Effective date: 20140319

FZDE Discontinued

Effective date: 20160329

FZDE Discontinued

Effective date: 20160329