CA2716334A1 - Inhibitors of human phosphatidyl-inositol 3-kinase delta - Google Patents

Inhibitors of human phosphatidyl-inositol 3-kinase delta Download PDF

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Publication number
CA2716334A1
CA2716334A1 CA2716334A CA2716334A CA2716334A1 CA 2716334 A1 CA2716334 A1 CA 2716334A1 CA 2716334 A CA2716334 A CA 2716334A CA 2716334 A CA2716334 A CA 2716334A CA 2716334 A1 CA2716334 A1 CA 2716334A1
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CA
Canada
Prior art keywords
substituted
unsubstituted
compound
group
4alkylenec
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2716334A
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English (en)
French (fr)
Inventor
Stephen L. White
Fuqiang Ruan
Edward A. Kesicki
Eugene Thorsett
Francine Farouz
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Icos Corp
Original Assignee
Icos Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Icos Corp filed Critical Icos Corp
Publication of CA2716334A1 publication Critical patent/CA2716334A1/en
Abandoned legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Transplantation (AREA)
  • Emergency Medicine (AREA)
  • Communicable Diseases (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Otolaryngology (AREA)
CA2716334A 2007-11-13 2008-11-12 Inhibitors of human phosphatidyl-inositol 3-kinase delta Abandoned CA2716334A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US98772307P 2007-11-13 2007-11-13
US60/987,723 2007-11-13
PCT/US2008/083262 WO2009064802A2 (en) 2007-11-13 2008-11-12 Inhibitors of human phosphatidyl-inositol 3-kinase delta

Publications (1)

Publication Number Publication Date
CA2716334A1 true CA2716334A1 (en) 2009-05-22

Family

ID=40639422

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2716334A Abandoned CA2716334A1 (en) 2007-11-13 2008-11-12 Inhibitors of human phosphatidyl-inositol 3-kinase delta

Country Status (13)

Country Link
US (1) US20110021541A1 (OSRAM)
EP (1) EP2220089A4 (OSRAM)
JP (1) JP2011503193A (OSRAM)
KR (1) KR20100119745A (OSRAM)
CN (1) CN101952292A (OSRAM)
AU (1) AU2008321099A1 (OSRAM)
CA (1) CA2716334A1 (OSRAM)
EA (1) EA201070611A1 (OSRAM)
GE (1) GEP20125635B (OSRAM)
IL (1) IL205747A0 (OSRAM)
NZ (1) NZ585460A (OSRAM)
SG (1) SG185996A1 (OSRAM)
WO (1) WO2009064802A2 (OSRAM)

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