CA2699414C - Treatment of vasomotor symptoms using flibanserin - Google Patents
Treatment of vasomotor symptoms using flibanserin Download PDFInfo
- Publication number
- CA2699414C CA2699414C CA2699414A CA2699414A CA2699414C CA 2699414 C CA2699414 C CA 2699414C CA 2699414 A CA2699414 A CA 2699414A CA 2699414 A CA2699414 A CA 2699414A CA 2699414 C CA2699414 C CA 2699414C
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- CA
- Canada
- Prior art keywords
- vasomotor symptoms
- flibanserin
- acid
- composition according
- optionally
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US97160507P | 2007-09-12 | 2007-09-12 | |
| US60/971,605 | 2007-09-12 | ||
| PCT/EP2008/062011 WO2009034111A1 (en) | 2007-09-12 | 2008-09-11 | Treatment of vasomotor symptoms |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2699414A1 CA2699414A1 (en) | 2009-03-19 |
| CA2699414C true CA2699414C (en) | 2016-04-05 |
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| Application Number | Title | Priority Date | Filing Date |
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| CA2699414A Expired - Fee Related CA2699414C (en) | 2007-09-12 | 2008-09-11 | Treatment of vasomotor symptoms using flibanserin |
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Families Citing this family (6)
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| US10675280B2 (en) | 2001-10-20 | 2020-06-09 | Sprout Pharmaceuticals, Inc. | Treating sexual desire disorders with flibanserin |
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| PL1912650T3 (pl) | 2005-08-03 | 2018-01-31 | Sprout Pharmaceuticals Inc | Zastosowanie flibanseryny w leczeniu otyłości |
| EP2097389B1 (en) * | 2006-12-20 | 2011-09-14 | Boehringer Ingelheim International GmbH | Sulfated benzimidazolone derivatives having mixed serotonine receptor affinity |
| UY31335A1 (es) * | 2007-09-12 | 2009-04-30 | Tratamiento de sintomas vasomotores | |
| WO2017133337A1 (zh) * | 2016-02-02 | 2017-08-10 | 深圳市塔吉瑞生物医药有限公司 | 一种取代的苯并咪唑酮化合物及包含该化合物的组合物 |
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| PL2021006T3 (pl) * | 2006-05-09 | 2015-12-31 | Sprout Pharmaceuticals Inc | Zastosowanie flibanseryny do leczenia pomenopauzalnych zaburzeń popędu płciowego |
| US20090312242A1 (en) * | 2006-06-30 | 2009-12-17 | Ramiro Castro | Flibanserin for the treatment of urinary incontinence and related diseases |
| WO2008006839A2 (en) * | 2006-07-14 | 2008-01-17 | Boehringer Ingelheim International Gmbh | Combinations of flibanserin with caffeine, process for their preparation and use thereof as medicaments |
| US20090318469A1 (en) | 2006-07-14 | 2009-12-24 | Boehringer Ingelheim International Gmbh | Use of Flibanserin for the Treatment of Sexual Disorders in Females |
| WO2008019996A2 (en) | 2006-08-14 | 2008-02-21 | Boehringer Ingelheim International Gmbh | Formulations of flibanserin and method for manufacturing the same |
| CL2007002214A1 (es) * | 2006-08-14 | 2008-03-07 | Boehringer Ingelheim Int | Composicion farmaceutica en la forma de comprimido, donde al menos la longitud del comprimido en el estado anterior de la aplicacion es al menos 7/12 del diametro pilorico del paciente y despues de ingerirlo en estado alimentado, la longitud del comp |
| MX2009002031A (es) | 2006-08-25 | 2009-03-06 | Boehringer Ingelheim Int | Sistema de liberacion controlada y metodo para fabricarlo. |
| EP2097389B1 (en) | 2006-12-20 | 2011-09-14 | Boehringer Ingelheim International GmbH | Sulfated benzimidazolone derivatives having mixed serotonine receptor affinity |
| JP2010522714A (ja) | 2007-03-28 | 2010-07-08 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 新規な医薬組成物 |
| UY31335A1 (es) * | 2007-09-12 | 2009-04-30 | Tratamiento de sintomas vasomotores |
-
2008
- 2008-09-10 UY UY31335A patent/UY31335A1/es not_active Application Discontinuation
- 2008-09-10 CL CL2008002693A patent/CL2008002693A1/es unknown
- 2008-09-10 PE PE2008001580A patent/PE20091188A1/es not_active Application Discontinuation
- 2008-09-11 JP JP2010524478A patent/JP2010539130A/ja active Pending
- 2008-09-11 KR KR1020107005191A patent/KR20100059848A/ko not_active Withdrawn
- 2008-09-11 MX MX2010002032A patent/MX2010002032A/es not_active Application Discontinuation
- 2008-09-11 WO PCT/EP2008/062011 patent/WO2009034111A1/en not_active Ceased
- 2008-09-11 EA EA201000433A patent/EA201000433A1/ru unknown
- 2008-09-11 EP EP08803978.9A patent/EP2200614B1/en active Active
- 2008-09-11 AR ARP080103952A patent/AR068416A1/es unknown
- 2008-09-11 CA CA2699414A patent/CA2699414C/en not_active Expired - Fee Related
- 2008-09-11 US US12/675,231 patent/US20110136825A1/en not_active Abandoned
- 2008-09-11 AU AU2008297104A patent/AU2008297104A1/en not_active Abandoned
- 2008-09-11 BR BRPI0816791A patent/BRPI0816791A2/pt not_active IP Right Cessation
- 2008-09-11 TW TW097134893A patent/TW200927118A/zh unknown
- 2008-09-11 CN CN2008801069327A patent/CN101801380B/zh not_active Expired - Fee Related
- 2008-09-11 NZ NZ584183A patent/NZ584183A/en not_active IP Right Cessation
- 2008-09-11 ES ES08803978.9T patent/ES2444707T3/es active Active
-
2010
- 2010-01-19 ZA ZA201000384A patent/ZA201000384B/xx unknown
- 2010-03-11 TN TNP2010000108A patent/TN2010000108A1/fr unknown
- 2010-03-12 CO CO10029659A patent/CO6260073A2/es not_active Application Discontinuation
- 2010-04-08 MA MA32746A patent/MA31757B1/fr unknown
-
2013
- 2013-03-20 US US13/847,683 patent/US20140005203A1/en not_active Abandoned
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2014
- 2014-12-26 US US14/583,275 patent/US10166230B2/en active Active
-
2017
- 2017-08-25 US US15/686,665 patent/US9949969B2/en not_active Expired - Fee Related
-
2018
- 2018-11-26 US US16/200,004 patent/US10596170B2/en not_active Expired - Fee Related
-
2020
- 2020-03-05 US US16/810,273 patent/US20200253962A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| JP2010539130A (ja) | 2010-12-16 |
| EA201000433A1 (ru) | 2010-10-29 |
| US10596170B2 (en) | 2020-03-24 |
| US20110136825A1 (en) | 2011-06-09 |
| CN101801380B (zh) | 2013-05-08 |
| US20140005203A1 (en) | 2014-01-02 |
| TW200927118A (en) | 2009-07-01 |
| US10166230B2 (en) | 2019-01-01 |
| ES2444707T3 (es) | 2014-02-26 |
| US20180071283A1 (en) | 2018-03-15 |
| EP2200614B1 (en) | 2013-11-27 |
| CL2008002693A1 (es) | 2009-10-16 |
| US20190091219A1 (en) | 2019-03-28 |
| CA2699414A1 (en) | 2009-03-19 |
| AU2008297104A1 (en) | 2009-03-19 |
| WO2009034111A1 (en) | 2009-03-19 |
| CN101801380A (zh) | 2010-08-11 |
| AR068416A1 (es) | 2009-11-18 |
| UY31335A1 (es) | 2009-04-30 |
| US9949969B2 (en) | 2018-04-24 |
| US20150250783A1 (en) | 2015-09-10 |
| ZA201000384B (en) | 2010-09-29 |
| MA31757B1 (fr) | 2010-10-01 |
| KR20100059848A (ko) | 2010-06-04 |
| MX2010002032A (es) | 2010-03-15 |
| TN2010000108A1 (fr) | 2011-09-26 |
| CO6260073A2 (es) | 2011-03-22 |
| NZ584183A (en) | 2012-05-25 |
| BRPI0816791A2 (pt) | 2019-09-24 |
| EP2200614A1 (en) | 2010-06-30 |
| PE20091188A1 (es) | 2009-08-31 |
| US20200253962A1 (en) | 2020-08-13 |
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