CA2672903C - Heterocyclic compounds and their use in treating inflammation, angiogenesis and cancer - Google Patents
Heterocyclic compounds and their use in treating inflammation, angiogenesis and cancer Download PDFInfo
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- CA2672903C CA2672903C CA2672903A CA2672903A CA2672903C CA 2672903 C CA2672903 C CA 2672903C CA 2672903 A CA2672903 A CA 2672903A CA 2672903 A CA2672903 A CA 2672903A CA 2672903 C CA2672903 C CA 2672903C
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Classifications
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US87628306P | 2006-12-20 | 2006-12-20 | |
| US60/876,283 | 2006-12-20 | ||
| PCT/US2007/026064 WO2008079292A1 (en) | 2006-12-20 | 2007-12-19 | Heterocyclic compounds and their use in treating inflammation, angiogenesis and cancer |
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| CA2672903A1 CA2672903A1 (en) | 2008-07-03 |
| CA2672903C true CA2672903C (en) | 2012-10-23 |
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| CA2672903A Expired - Fee Related CA2672903C (en) | 2006-12-20 | 2007-12-19 | Heterocyclic compounds and their use in treating inflammation, angiogenesis and cancer |
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| US (1) | US8338455B2 (enExample) |
| EP (1) | EP2118088B1 (enExample) |
| JP (1) | JP5528812B2 (enExample) |
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| MX (1) | MX2009006543A (enExample) |
| WO (1) | WO2008079292A1 (enExample) |
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| DK3184526T3 (en) | 2005-12-13 | 2019-01-14 | Incyte Holdings Corp | PYRROLO [2,3-D] PYRIMIDINE DERIVATIVES AS A JANUS-KINASE INHIBITOR |
| EP2740731B1 (en) | 2007-06-13 | 2016-03-23 | Incyte Holdings Corporation | Crystalline salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl)-3-cyclopentylpropanenitrile |
| KR20100093552A (ko) | 2007-11-02 | 2010-08-25 | 버텍스 파마슈티칼스 인코포레이티드 | 단백질 키나제 ｃ-세타로서의 [1ｈ-피라졸로[3,4-ｂ]피리딘-4-일]-페닐 또는 -피리딘-2-일 유도체 |
| CL2009001884A1 (es) * | 2008-10-02 | 2010-05-14 | Incyte Holdings Corp | Uso de 3-ciclopentil-3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)propanonitrilo, inhibidor de janus quinasa, y uso de una composición que lo comprende para el tratamiento del ojo seco. |
| JP5770102B2 (ja) * | 2008-12-19 | 2015-08-26 | ジェネンテック， インコーポレイテッド | 複素環化合物と使用方法 |
| ES2487542T3 (es) * | 2009-05-22 | 2014-08-21 | Incyte Corporation | Derivados de N-(hetero)aril-pirrolidina de pirazol-4-il-pirrolo[2,3-d]pirimidinas y pirrol-3-il-pirrolo[2,3-d]pirimidinas como inhibidores de cinasas Janus |
| WO2010135621A1 (en) * | 2009-05-22 | 2010-11-25 | Incyte Corporation | 3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]octane- or heptane-nitrile as jak inhibitors |
| JP2011057661A (ja) * | 2009-08-14 | 2011-03-24 | Bayer Cropscience Ag | 殺虫性カルボキサミド類 |
| WO2011028685A1 (en) * | 2009-09-01 | 2011-03-10 | Incyte Corporation | Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors |
| SMT201800137T1 (it) | 2010-03-10 | 2018-07-17 | Incyte Holdings Corp | Derivati di piperidin-4-il azetidina come inibitori di jak1 |
| PH12012502296B1 (en) | 2010-05-21 | 2017-10-06 | Incyte Holdings Corp | Topical formulation for a jak inhibitor |
| ES2536415T3 (es) | 2010-11-19 | 2015-05-25 | Incyte Corporation | Pirrolopiridinas y pirrolopirimidinas sustituidas heterocíclicas como inhibidores de JAK |
| SG190839A1 (en) | 2010-11-19 | 2013-07-31 | Incyte Corp | Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as jak inhibitors |
| JP2014520151A (ja) | 2011-06-20 | 2014-08-21 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | 蠕虫感染を処置するためのヘテロ環式化合物 |
| WO2012177606A1 (en) | 2011-06-20 | 2012-12-27 | Incyte Corporation | Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as jak inhibitors |
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| IE903196A1 (en) * | 1989-09-05 | 1991-03-13 | Searle & Co | Substituted n-benzylpiperidine amides |
| EP0860433B1 (en) | 1995-11-07 | 2002-07-03 | Kirin Beer Kabushiki Kaisha | Quinoline derivatives and quinazoline derivatives inhibiting autophosphorylation of growth factor receptor originating in platelet and pharmaceutical compositions containing the same |
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| PL199802B1 (pl) | 1999-02-10 | 2008-10-31 | Astrazeneca Ab | Pochodne chinazoliny, sposoby ich wytwarzania, ich kompozycje farmaceutyczne i ich zastosowania |
| HUP0202682A3 (en) | 1999-09-10 | 2003-03-28 | Merck & Co Inc | Tyrosine kinase inhibitors, pharmaceutical compositions containing them and their use |
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- 2007-12-19 AU AU2007338793A patent/AU2007338793B2/en not_active Ceased
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| US20080161346A1 (en) | 2008-07-03 |
| MX2009006543A (es) | 2009-06-26 |
| AU2007338793A1 (en) | 2008-07-03 |
| AU2007338793B2 (en) | 2012-05-03 |
| JP5528812B2 (ja) | 2014-06-25 |
| JP2010513523A (ja) | 2010-04-30 |
| US8338455B2 (en) | 2012-12-25 |
| WO2008079292A1 (en) | 2008-07-03 |
| CA2672903A1 (en) | 2008-07-03 |
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| EP2118088B1 (en) | 2012-05-30 |
| EP2118088A1 (en) | 2009-11-18 |
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