AU2007338793B2 - Heterocyclic compounds and their use in treating inflammation, angiogenesis and cancer - Google Patents
Heterocyclic compounds and their use in treating inflammation, angiogenesis and cancer Download PDFInfo
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- AU2007338793B2 AU2007338793B2 AU2007338793A AU2007338793A AU2007338793B2 AU 2007338793 B2 AU2007338793 B2 AU 2007338793B2 AU 2007338793 A AU2007338793 A AU 2007338793A AU 2007338793 A AU2007338793 A AU 2007338793A AU 2007338793 B2 AU2007338793 B2 AU 2007338793B2
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- compound
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- cycloalkyl
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Classifications
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US87628306P | 2006-12-20 | 2006-12-20 | |
| US60/876,283 | 2006-12-20 | ||
| PCT/US2007/026064 WO2008079292A1 (en) | 2006-12-20 | 2007-12-19 | Heterocyclic compounds and their use in treating inflammation, angiogenesis and cancer |
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| AU2007338793A1 AU2007338793A1 (en) | 2008-07-03 |
| AU2007338793B2 true AU2007338793B2 (en) | 2012-05-03 |
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| AU2007338793A Ceased AU2007338793B2 (en) | 2006-12-20 | 2007-12-19 | Heterocyclic compounds and their use in treating inflammation, angiogenesis and cancer |
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| Country | Link |
|---|---|
| US (1) | US8338455B2 (enExample) |
| EP (1) | EP2118088B1 (enExample) |
| JP (1) | JP5528812B2 (enExample) |
| AU (1) | AU2007338793B2 (enExample) |
| CA (1) | CA2672903C (enExample) |
| ES (1) | ES2387471T3 (enExample) |
| MX (1) | MX2009006543A (enExample) |
| WO (1) | WO2008079292A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104918945A (zh) * | 2012-11-01 | 2015-09-16 | 因赛特公司 | 作为jak抑制剂的三环稠合噻吩衍生物 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK3184526T3 (en) | 2005-12-13 | 2019-01-14 | Incyte Holdings Corp | PYRROLO [2,3-D] PYRIMIDINE DERIVATIVES AS A JANUS-KINASE INHIBITOR |
| EP2740731B1 (en) | 2007-06-13 | 2016-03-23 | Incyte Holdings Corporation | Crystalline salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl)-3-cyclopentylpropanenitrile |
| KR20100093552A (ko) | 2007-11-02 | 2010-08-25 | 버텍스 파마슈티칼스 인코포레이티드 | 단백질 키나제 ｃ-세타로서의 [1ｈ-피라졸로[3,4-ｂ]피리딘-4-일]-페닐 또는 -피리딘-2-일 유도체 |
| CL2009001884A1 (es) * | 2008-10-02 | 2010-05-14 | Incyte Holdings Corp | Uso de 3-ciclopentil-3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)propanonitrilo, inhibidor de janus quinasa, y uso de una composición que lo comprende para el tratamiento del ojo seco. |
| JP5770102B2 (ja) * | 2008-12-19 | 2015-08-26 | ジェネンテック， インコーポレイテッド | 複素環化合物と使用方法 |
| ES2487542T3 (es) * | 2009-05-22 | 2014-08-21 | Incyte Corporation | Derivados de N-(hetero)aril-pirrolidina de pirazol-4-il-pirrolo[2,3-d]pirimidinas y pirrol-3-il-pirrolo[2,3-d]pirimidinas como inhibidores de cinasas Janus |
| WO2010135621A1 (en) * | 2009-05-22 | 2010-11-25 | Incyte Corporation | 3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]octane- or heptane-nitrile as jak inhibitors |
| JP2011057661A (ja) * | 2009-08-14 | 2011-03-24 | Bayer Cropscience Ag | 殺虫性カルボキサミド類 |
| WO2011028685A1 (en) * | 2009-09-01 | 2011-03-10 | Incyte Corporation | Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors |
| SMT201800137T1 (it) | 2010-03-10 | 2018-07-17 | Incyte Holdings Corp | Derivati di piperidin-4-il azetidina come inibitori di jak1 |
| PH12012502296B1 (en) | 2010-05-21 | 2017-10-06 | Incyte Holdings Corp | Topical formulation for a jak inhibitor |
| ES2536415T3 (es) | 2010-11-19 | 2015-05-25 | Incyte Corporation | Pirrolopiridinas y pirrolopirimidinas sustituidas heterocíclicas como inhibidores de JAK |
| SG190839A1 (en) | 2010-11-19 | 2013-07-31 | Incyte Corp | Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as jak inhibitors |
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| MA39987A (fr) | 2014-04-30 | 2017-03-08 | Incyte Corp | Procédés de préparation d'un inhibiteur de jak1 et nouvelles formes associées |
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| SMT202400306T1 (it) | 2018-03-30 | 2024-09-16 | Incyte Corp | Trattamento dell'idrosadenite suppurativa utilizzando inibitori di jak. |
| AU2021255966A1 (en) * | 2020-04-17 | 2022-11-17 | Escient Pharmaceuticals, Inc. | Modulators of mas-related G-protein receptor X4 and related products and methods |
| KR20230022457A (ko) * | 2020-05-08 | 2023-02-15 | 조지아뮨 엘엘씨 | Akt3 조절제 |
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- 2007-12-19 AU AU2007338793A patent/AU2007338793B2/en not_active Ceased
- 2007-12-19 JP JP2009542923A patent/JP5528812B2/ja not_active Expired - Fee Related
- 2007-12-19 MX MX2009006543A patent/MX2009006543A/es active IP Right Grant
- 2007-12-19 US US12/004,156 patent/US8338455B2/en not_active Expired - Fee Related
- 2007-12-19 EP EP07863179A patent/EP2118088B1/en active Active
- 2007-12-19 WO PCT/US2007/026064 patent/WO2008079292A1/en not_active Ceased
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| EP0416581A1 (en) * | 1989-09-05 | 1991-03-13 | G.D. Searle & Co. | Substituted N-benzylpiperidine amides |
| US6372736B1 (en) * | 1998-07-21 | 2002-04-16 | Pfizer Inc | Heterocyclic compounds as inhibitors of rotamase enzymes |
| US20040034028A1 (en) * | 2000-11-23 | 2004-02-19 | Alyx-Caroline Guevel | 4-(biphenylcarbonylamino)piperidine derivatives as mtp inhibitors |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104918945A (zh) * | 2012-11-01 | 2015-09-16 | 因赛特公司 | 作为jak抑制剂的三环稠合噻吩衍生物 |
| CN104918945B (zh) * | 2012-11-01 | 2018-01-05 | 因赛特公司 | 作为jak抑制剂的三环稠合噻吩衍生物 |
| US11851442B2 (en) | 2012-11-01 | 2023-12-26 | Incyte Corporation | Tricyclic fused thiophene derivatives as JAK inhibitors |
Also Published As
| Publication number | Publication date |
|---|---|
| US20080161346A1 (en) | 2008-07-03 |
| MX2009006543A (es) | 2009-06-26 |
| AU2007338793A1 (en) | 2008-07-03 |
| CA2672903C (en) | 2012-10-23 |
| JP5528812B2 (ja) | 2014-06-25 |
| JP2010513523A (ja) | 2010-04-30 |
| US8338455B2 (en) | 2012-12-25 |
| WO2008079292A1 (en) | 2008-07-03 |
| CA2672903A1 (en) | 2008-07-03 |
| ES2387471T3 (es) | 2012-09-24 |
| EP2118088B1 (en) | 2012-05-30 |
| EP2118088A1 (en) | 2009-11-18 |
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