CA2658896A1 - Crystalline forms of rapamycin analogs - Google Patents

Crystalline forms of rapamycin analogs Download PDF

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Publication number
CA2658896A1
CA2658896A1 CA002658896A CA2658896A CA2658896A1 CA 2658896 A1 CA2658896 A1 CA 2658896A1 CA 002658896 A CA002658896 A CA 002658896A CA 2658896 A CA2658896 A CA 2658896A CA 2658896 A1 CA2658896 A1 CA 2658896A1
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Canada
Prior art keywords
powder
ray diffraction
diffraction pattern
rapamycin analog
composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002658896A
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English (en)
French (fr)
Inventor
Shekhar Viswanath
Larry Bartelt
Robert Leanna
Michael Rasmussen
Madhup Dhaon
Rodger Henry
Thomas Borchardt
Shuang Chen
Geoff Zhang
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Abbott Laboratories
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Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US11/781,804 external-priority patent/US7812032B2/en
Priority claimed from US11/781,807 external-priority patent/US7820812B2/en
Application filed by Individual filed Critical Individual
Publication of CA2658896A1 publication Critical patent/CA2658896A1/en
Abandoned legal-status Critical Current

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
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CA002658896A 2006-07-25 2007-07-24 Crystalline forms of rapamycin analogs Abandoned CA2658896A1 (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US82031706P 2006-07-25 2006-07-25
US60/820,317 2006-07-25
US11/781,804 US7812032B2 (en) 2006-07-25 2007-07-23 Crystalline forms of rapamycin analogs
US11/781,804 2007-07-23
US11/781,807 US7820812B2 (en) 2006-07-25 2007-07-23 Methods of manufacturing crystalline forms of rapamycin analogs
US11/781,807 2007-07-23
PCT/US2007/074159 WO2008014222A1 (en) 2006-07-25 2007-07-24 Crystalline forms of rapamycin analogs

Publications (1)

Publication Number Publication Date
CA2658896A1 true CA2658896A1 (en) 2008-01-31

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ID=38562825

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002658896A Abandoned CA2658896A1 (en) 2006-07-25 2007-07-24 Crystalline forms of rapamycin analogs

Country Status (10)

Country Link
EP (2) EP2051984A1 (Direct)
JP (1) JP2010500286A (Direct)
KR (1) KR20090035716A (Direct)
AU (1) AU2007276837B2 (Direct)
BR (1) BRPI0714945B8 (Direct)
CA (1) CA2658896A1 (Direct)
IL (1) IL196706A0 (Direct)
MX (1) MX2009001067A (Direct)
NZ (1) NZ574654A (Direct)
WO (1) WO2008014222A1 (Direct)

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US7812032B2 (en) 2006-07-25 2010-10-12 Abbott Laboratories Crystalline forms of rapamycin analogs
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WO2013022458A1 (en) * 2011-08-05 2013-02-14 Boston Scientific Scimed, Inc. Methods of converting amorphous drug substance into crystalline form
US9056152B2 (en) 2011-08-25 2015-06-16 Boston Scientific Scimed, Inc. Medical device with crystalline drug coating
US9439892B2 (en) 2013-05-16 2016-09-13 Surmodics, Inc. Macrolide particulates, methods for preparation, and medical devices associated therewith
WO2014201236A1 (en) * 2013-06-12 2014-12-18 Surmodics, Inc. Solvent methods for preparing crystalline macrolide particulates, compositions, and articles containing particulates
DE102013110294B4 (de) * 2013-09-18 2016-07-07 Innora Gmbh Limus-Depot-Formulierung auf Ballonkathetern
US10098846B2 (en) 2016-03-31 2018-10-16 Surmodics, Inc. Drug-containing particulate composition with cationic agent, associated medical devices, and methods for treatment
EP3554571B1 (en) 2016-12-16 2024-11-13 Surmodics, Inc. Hydrophobic active agent particle coatings and methods for treatment
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