CA2632149C - Pyrimidine derivatives for the treatment of abnormal cell growth - Google Patents
Pyrimidine derivatives for the treatment of abnormal cell growth Download PDFInfo
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- CA2632149C CA2632149C CA2632149A CA2632149A CA2632149C CA 2632149 C CA2632149 C CA 2632149C CA 2632149 A CA2632149 A CA 2632149A CA 2632149 A CA2632149 A CA 2632149A CA 2632149 C CA2632149 C CA 2632149C
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- A61P35/02—Antineoplastic agents specific for leukemia
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- A—HUMAN NECESSITIES
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US74125205P | 2005-12-01 | 2005-12-01 | |
| US60/741,252 | 2005-12-01 | ||
| PCT/IB2006/003349 WO2007063384A2 (en) | 2005-12-01 | 2006-11-20 | Pyrimidine derivatives for the treatment of abnormal cell growth |
Publications (2)
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| CA2632149A1 CA2632149A1 (en) | 2007-06-07 |
| CA2632149C true CA2632149C (en) | 2011-11-15 |
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|---|---|---|---|
| CA2632149A Active CA2632149C (en) | 2005-12-01 | 2006-11-20 | Pyrimidine derivatives for the treatment of abnormal cell growth |
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| Country | Link |
|---|---|
| US (1) | US8722884B2 (enExample) |
| EP (1) | EP1966192B1 (enExample) |
| JP (2) | JP5134234B2 (enExample) |
| AR (1) | AR057202A1 (enExample) |
| CA (1) | CA2632149C (enExample) |
| TW (1) | TWI374880B (enExample) |
| WO (1) | WO2007063384A2 (enExample) |
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|---|---|---|---|---|
| ES2593486T3 (es) | 2007-04-18 | 2016-12-09 | Pfizer Products Inc. | Derivados de sulfonil amida para el tratamiento del crecimiento celular anómalo |
| EA020807B1 (ru) | 2008-06-17 | 2015-01-30 | Астразенека Аб | Соединения пиридина |
| WO2011018517A1 (en) | 2009-08-14 | 2011-02-17 | Boehringer Ingelheim International Gmbh | Regioselective preparation of 2-amino-5-trifluoromethylpyrimidine derivatives |
| US8933227B2 (en) | 2009-08-14 | 2015-01-13 | Boehringer Ingelheim International Gmbh | Selective synthesis of functionalized pyrimidines |
| US20120244141A1 (en) | 2010-09-28 | 2012-09-27 | Boehringer Ingelheim International Gmbh | Stratification of cancer patients for susceptibility to therapy with PTK2 inhibitors |
| ES2691673T3 (es) | 2011-02-17 | 2018-11-28 | Cancer Therapeutics Crc Pty Limited | Inhibidores de Fak |
| DK2675794T3 (da) | 2011-02-17 | 2019-05-06 | Cancer Therapeutics Crc Pty Ltd | Selektive fak-inhibitorer |
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| JPS5924990B2 (ja) * | 1979-11-21 | 1984-06-13 | 協和醗酵工業株式会社 | 新規なピペリジン誘導体 |
| GB9222700D0 (en) * | 1992-10-29 | 1992-12-09 | Smithkline Beecham Plc | Chemical compounds |
| US5795909A (en) * | 1996-05-22 | 1998-08-18 | Neuromedica, Inc. | DHA-pharmaceutical agent conjugates of taxanes |
| ES2174462T3 (es) * | 1997-07-29 | 2002-11-01 | Upjohn Co | Formulacion autoestimulante para compuestos lipofilos. |
| CH689805A8 (fr) * | 1998-07-02 | 2000-02-29 | Smithkline Beecham Plc | Méthanesulfonate de paroxétine, procédé pour sa préparation et compositions pharmaceutiques le contenant. |
| JP2001261654A (ja) * | 2000-03-21 | 2001-09-26 | Mitsui Chemicals Inc | キノリン誘導体およびそれを有効成分として含有する核内レセプター作動薬 |
| WO2003037344A1 (en) * | 2001-11-02 | 2003-05-08 | Shire Biochem Inc. | Pharmaceutical compositions for the treatment of leukemia comprising dioxolane nucleosides analogs |
| EP1625121B1 (en) * | 2002-12-20 | 2010-02-24 | Pfizer Products Inc. | Pyrimidine derivatives for the treatment of abnormal cell growth |
| UA80767C2 (en) | 2002-12-20 | 2007-10-25 | Pfizer Prod Inc | Pyrimidine derivatives for the treatment of abnormal cell growth |
| US7109337B2 (en) * | 2002-12-20 | 2006-09-19 | Pfizer Inc | Pyrimidine derivatives for the treatment of abnormal cell growth |
| JP2007537235A (ja) | 2004-05-14 | 2007-12-20 | ファイザー・プロダクツ・インク | 異常細胞増殖の治療用ピリミジン誘導体 |
| WO2005111022A1 (en) | 2004-05-14 | 2005-11-24 | Pfizer Products Inc. | Pyrimidines derivatives for the treatment of abnormal cell growth |
| BRPI0510963A (pt) | 2004-05-14 | 2007-11-20 | Pfizer Prod Inc | derivados pirimidina para o tratamento do crescimento anormal de células |
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- 2006-11-20 EP EP06809250A patent/EP1966192B1/en not_active Not-in-force
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| WO2007063384A3 (en) | 2007-10-04 |
| EP1966192A2 (en) | 2008-09-10 |
| JP2007153892A (ja) | 2007-06-21 |
| CA2632149A1 (en) | 2007-06-07 |
| US20110033441A1 (en) | 2011-02-10 |
| EP1966192B1 (en) | 2012-10-17 |
| AR057202A1 (es) | 2007-11-21 |
| JP5134234B2 (ja) | 2013-01-30 |
| WO2007063384A2 (en) | 2007-06-07 |
| US8722884B2 (en) | 2014-05-13 |
| JP2012255038A (ja) | 2012-12-27 |
| TW200730507A (en) | 2007-08-16 |
| TWI374880B (en) | 2012-10-21 |
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