CA2591313A1 - Procedes de preparation de composes indazole - Google Patents
Procedes de preparation de composes indazole Download PDFInfo
- Publication number
- CA2591313A1 CA2591313A1 CA002591313A CA2591313A CA2591313A1 CA 2591313 A1 CA2591313 A1 CA 2591313A1 CA 002591313 A CA002591313 A CA 002591313A CA 2591313 A CA2591313 A CA 2591313A CA 2591313 A1 CA2591313 A1 CA 2591313A1
- Authority
- CA
- Canada
- Prior art keywords
- formula
- compound
- alkyl
- aryl
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US62471904P | 2004-11-02 | 2004-11-02 | |
US60/624,719 | 2004-11-02 | ||
US62480104P | 2004-12-14 | 2004-12-14 | |
US60/624,801 | 2004-12-14 | ||
PCT/IB2005/003348 WO2006048761A2 (fr) | 2004-11-02 | 2005-10-21 | Procedes de preparation de composes indazole |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2591313A1 true CA2591313A1 (fr) | 2006-05-11 |
Family
ID=35456957
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002591313A Abandoned CA2591313A1 (fr) | 2004-11-02 | 2005-10-21 | Procedes de preparation de composes indazole |
Country Status (9)
Country | Link |
---|---|
EP (1) | EP1814859A2 (fr) |
KR (1) | KR20070085727A (fr) |
AU (1) | AU2005300241A1 (fr) |
CA (1) | CA2591313A1 (fr) |
IL (1) | IL183605A0 (fr) |
MX (1) | MX2007006554A (fr) |
RU (1) | RU2007120635A (fr) |
TW (1) | TW200630345A (fr) |
WO (1) | WO2006048761A2 (fr) |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2136284A1 (en) * | 1971-02-08 | 1972-08-31 | Diamond Shamrock Corp., Cleveland, Ohio (V.StA.) | Herbicidal pyrrolidinyl-carboxanilides - from arylisocyanates and pyrrolidines in organic solvents |
PE20010306A1 (es) * | 1999-07-02 | 2001-03-29 | Agouron Pharma | Compuestos de indazol y composiciones farmaceuticas que los contienen utiles para la inhibicion de proteina kinasa |
-
2005
- 2005-10-21 KR KR1020077012588A patent/KR20070085727A/ko not_active Application Discontinuation
- 2005-10-21 RU RU2007120635/04A patent/RU2007120635A/ru not_active Application Discontinuation
- 2005-10-21 CA CA002591313A patent/CA2591313A1/fr not_active Abandoned
- 2005-10-21 EP EP05797459A patent/EP1814859A2/fr not_active Withdrawn
- 2005-10-21 MX MX2007006554A patent/MX2007006554A/es unknown
- 2005-10-21 WO PCT/IB2005/003348 patent/WO2006048761A2/fr active Application Filing
- 2005-10-21 AU AU2005300241A patent/AU2005300241A1/en not_active Abandoned
- 2005-11-01 TW TW094138277A patent/TW200630345A/zh unknown
-
2007
- 2007-05-31 IL IL183605A patent/IL183605A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
IL183605A0 (en) | 2007-09-20 |
WO2006048761A3 (fr) | 2006-06-22 |
TW200630345A (en) | 2006-09-01 |
AU2005300241A1 (en) | 2006-05-11 |
MX2007006554A (es) | 2007-06-19 |
WO2006048761A2 (fr) | 2006-05-11 |
KR20070085727A (ko) | 2007-08-27 |
EP1814859A2 (fr) | 2007-08-08 |
RU2007120635A (ru) | 2008-12-10 |
AU2005300241A2 (en) | 2006-05-11 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EEER | Examination request | ||
FZDE | Discontinued |