CA2585557C - Nouveaux composes pharmaceutiques - Google Patents

Nouveaux composes pharmaceutiques Download PDF

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Publication number
CA2585557C
CA2585557C CA002585557A CA2585557A CA2585557C CA 2585557 C CA2585557 C CA 2585557C CA 002585557 A CA002585557 A CA 002585557A CA 2585557 A CA2585557 A CA 2585557A CA 2585557 C CA2585557 C CA 2585557C
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Canada
Prior art keywords
ethyl
pyrimidin
pyrazolo
amine
ethoxyethyl
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Expired - Fee Related
Application number
CA002585557A
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English (en)
Other versions
CA2585557A1 (fr
Inventor
Brad Alan Acker
Robert Owen Hughes
Eric John Jacobsen
Hwang-Fun Lu
Thomas Edward Rogers
Michael Brent Tollefson
John Keith Walker
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Pharmacia and Upjohn Co LLC
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Pharmacia and Upjohn Co LLC
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Publication of CA2585557A1 publication Critical patent/CA2585557A1/fr
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Publication of CA2585557C publication Critical patent/CA2585557C/fr
Expired - Fee Related legal-status Critical Current
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
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  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
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  • Endocrinology (AREA)
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  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Reproductive Health (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Psychiatry (AREA)
  • Pulmonology (AREA)
  • Addiction (AREA)
  • Pregnancy & Childbirth (AREA)
  • Immunology (AREA)
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CA002585557A 2004-10-28 2005-10-17 Nouveaux composes pharmaceutiques Expired - Fee Related CA2585557C (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US62294104P 2004-10-28 2004-10-28
US60/622,941 2004-10-28
PCT/IB2005/003326 WO2006046135A2 (fr) 2004-10-28 2005-10-17 Nouveaux composes pharmaceutiques

Publications (2)

Publication Number Publication Date
CA2585557A1 CA2585557A1 (fr) 2006-05-04
CA2585557C true CA2585557C (fr) 2009-08-18

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CA002585557A Expired - Fee Related CA2585557C (fr) 2004-10-28 2005-10-17 Nouveaux composes pharmaceutiques

Country Status (4)

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EP (1) EP1809632A2 (fr)
JP (1) JP2008517994A (fr)
CA (1) CA2585557C (fr)
WO (1) WO2006046135A2 (fr)

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BRPI0609225A2 (pt) 2005-05-12 2010-03-09 Pfizer formas cristalinas anidras de n-[1-(2-etoxietil)-5-(n-etil-n-metilamino)-7-(4-metilpiridi n-2-il-amino)-1h-pirazolo[4,3-d]pirimidina-3-carbonil] metanossulfonamida, composição farmacêutica compreendendo as mesmas e uso das mesmas
NL2000291C2 (nl) * 2005-11-10 2009-02-17 Pfizer Prod Inc 1-(1-(2-ethoxyethyl)-3-ethyl-7-(4-methylpyridin-2-ylamino)-1H- pyrazool(4,3-d)pyrimidine-5-yl)piperidine-4-carbonzuur en zouten daarvan.
ES2310144B1 (es) 2007-06-15 2010-01-12 Galenicum Health, S.L. Intermedios para la preparacion de un inhibidor de la fosfodiesterasa tipo 5.
WO2012073143A1 (fr) 2010-12-01 2012-06-07 Pfizer Inc. Inhibiteur de kat ii
EP2809659A1 (fr) 2012-02-03 2014-12-10 Basf Se Composés de pyrimidine fongicides
EA201491667A1 (ru) 2012-03-13 2015-03-31 Басф Се Фунгицидные соединения пиримидина
US9422267B2 (en) 2012-12-26 2016-08-23 Medivation Technologies, Inc. Fused pyrimidine compounds and use thereof
WO2015036059A1 (fr) 2013-09-16 2015-03-19 Basf Se Composés fongicides de pyrimidine
US11554120B2 (en) * 2018-08-03 2023-01-17 Bristol-Myers Squibb Company 1H-pyrazolo[4,3-d]pyrimidine compounds as toll-like receptor 7 (TLR7) agonists and methods and uses therefor
CN115322105A (zh) * 2021-05-11 2022-11-11 江苏润安制药有限公司 一种合成艾拉莫德关键中间体的方法

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WO2006046135A2 (fr) 2006-05-04

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