CA2585557A1 - Nouveaux composes pharmaceutiques - Google Patents

Nouveaux composes pharmaceutiques Download PDF

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Publication number
CA2585557A1
CA2585557A1 CA002585557A CA2585557A CA2585557A1 CA 2585557 A1 CA2585557 A1 CA 2585557A1 CA 002585557 A CA002585557 A CA 002585557A CA 2585557 A CA2585557 A CA 2585557A CA 2585557 A1 CA2585557 A1 CA 2585557A1
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Canada
Prior art keywords
inhibitors
pde
pyrazolo
pyrimidine derivatives
derivatives useful
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Granted
Application number
CA002585557A
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English (en)
Other versions
CA2585557C (fr
Inventor
Brad Alan Acker
Robert Owen Hughes
Eric John Jacobsen
Hwang-Fun Lu
Thomas Edward Rogers
Michael Brent Tollefson
John Keith Walker
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Pharmacia and Upjohn Co LLC
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Individual
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Publication of CA2585557C publication Critical patent/CA2585557C/fr
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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CA002585557A 2004-10-28 2005-10-17 Nouveaux composes pharmaceutiques Expired - Fee Related CA2585557C (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US62294104P 2004-10-28 2004-10-28
US60/622,941 2004-10-28
PCT/IB2005/003326 WO2006046135A2 (fr) 2004-10-28 2005-10-17 Nouveaux composes pharmaceutiques

Publications (2)

Publication Number Publication Date
CA2585557A1 true CA2585557A1 (fr) 2006-05-04
CA2585557C CA2585557C (fr) 2009-08-18

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CA002585557A Expired - Fee Related CA2585557C (fr) 2004-10-28 2005-10-17 Nouveaux composes pharmaceutiques

Country Status (4)

Country Link
EP (1) EP1809632A2 (fr)
JP (1) JP2008517994A (fr)
CA (1) CA2585557C (fr)
WO (1) WO2006046135A2 (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2006245416B2 (en) 2005-05-12 2012-02-23 Pfizer Inc. Anhydrous crystalline forms of N-[1-(2-ethoxyethyl)-5-(N-ethyl-N-methylamino)-7-(4-methylpyridin-2-yl-amino)-1H-pyrazolo[4,3-d]pyrimidine-3-carbonyl]methanesulfonamide
NL2000291C2 (nl) 2005-11-10 2009-02-17 Pfizer Prod Inc 1-(1-(2-ethoxyethyl)-3-ethyl-7-(4-methylpyridin-2-ylamino)-1H- pyrazool(4,3-d)pyrimidine-5-yl)piperidine-4-carbonzuur en zouten daarvan.
ES2310144B1 (es) 2007-06-15 2010-01-12 Galenicum Health, S.L. Intermedios para la preparacion de un inhibidor de la fosfodiesterasa tipo 5.
WO2012073143A1 (fr) 2010-12-01 2012-06-07 Pfizer Inc. Inhibiteur de kat ii
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