CA2555313A1 - Heparanase inhibitors and uses thereof - Google Patents
Heparanase inhibitors and uses thereof Download PDFInfo
- Publication number
- CA2555313A1 CA2555313A1 CA002555313A CA2555313A CA2555313A1 CA 2555313 A1 CA2555313 A1 CA 2555313A1 CA 002555313 A CA002555313 A CA 002555313A CA 2555313 A CA2555313 A CA 2555313A CA 2555313 A1 CA2555313 A1 CA 2555313A1
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- Prior art keywords
- alkyl
- nr9r
- group
- aryl
- compound
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- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US54190404P | 2004-02-06 | 2004-02-06 | |
| US06/541,904 | 2004-02-06 | ||
| PCT/IL2005/000149 WO2005074375A2 (en) | 2004-02-06 | 2005-02-06 | Heparanase inhibitors and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2555313A1 true CA2555313A1 (en) | 2005-08-18 |
Family
ID=37074845
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002555313A Abandoned CA2555313A1 (en) | 2004-02-06 | 2005-02-06 | Heparanase inhibitors and uses thereof |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20070185176A1 (enExample) |
| EP (1) | EP1720828A2 (enExample) |
| JP (1) | JP2007525494A (enExample) |
| AU (1) | AU2005211255A1 (enExample) |
| CA (1) | CA2555313A1 (enExample) |
| WO (1) | WO2005074375A2 (enExample) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI20041129A0 (fi) * | 2004-08-30 | 2004-08-30 | Ctt Cancer Targeting Tech Oy | Tioksotiatsolidinoniyhdisteitä lääkkeinä käytettäviksi |
| RU2008131330A (ru) * | 2005-12-30 | 2010-02-10 | Арбор Вита Корпорейшн (Us) | Низкомолекулярные ингибиторы взаимодействия pdz |
| US8633160B2 (en) * | 2005-12-30 | 2014-01-21 | Nono Inc. | Small molecule inhibitors of PDZ interactions |
| KR101426093B1 (ko) | 2006-02-10 | 2014-08-01 | 서미트 코포레이션 피엘씨 | 뒤시엔느 근이영양증의 치료 |
| US7875603B2 (en) * | 2006-09-21 | 2011-01-25 | Nova Southeastern University | Specific inhibitors for vascular endothelial growth factor receptors |
| DK2170396T3 (en) * | 2007-08-03 | 2017-03-13 | Summit Therapeutics Plc | PHARMACEUTICAL COMBINATIONS TO TREAT THE MUSCLE DYROPHY OF DUCHENNES |
| GB0715937D0 (en) * | 2007-08-15 | 2007-09-26 | Vastox Plc | Method of treatment og duchenne muscular dystrophy |
| CN101544846B (zh) * | 2009-05-04 | 2012-07-04 | 泰兴市锦鸡染料有限公司 | 一种活性嫩黄染料及其合成工艺 |
| US8628554B2 (en) | 2010-06-13 | 2014-01-14 | Virender K. Sharma | Intragastric device for treating obesity |
| US9526648B2 (en) | 2010-06-13 | 2016-12-27 | Synerz Medical, Inc. | Intragastric device for treating obesity |
| US10420665B2 (en) | 2010-06-13 | 2019-09-24 | W. L. Gore & Associates, Inc. | Intragastric device for treating obesity |
| US10010439B2 (en) | 2010-06-13 | 2018-07-03 | Synerz Medical, Inc. | Intragastric device for treating obesity |
| BR112013032813A2 (pt) | 2011-06-20 | 2016-08-16 | Du Pont | composto de fórmula, composição e método para o tratamento, controle, prevenção ou proteção dos animais contra a infecção por helmintos |
| WO2013131931A1 (en) * | 2012-03-06 | 2013-09-12 | Compound Handling B.V. | Aminomethylene pyrazolones with therapeutic activity |
| EP2636673A1 (en) * | 2012-03-06 | 2013-09-11 | Compound Handling B.V. | Aminomethylene pyrazolones with therapeutic activity |
| US10779980B2 (en) | 2016-04-27 | 2020-09-22 | Synerz Medical, Inc. | Intragastric device for treating obesity |
| EP3381906A1 (en) * | 2017-03-27 | 2018-10-03 | Leadiant Biosciences SA | Compounds for use as heparanase inhibitors |
| AU2019387370A1 (en) | 2018-11-30 | 2021-06-10 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
| WO2020219753A1 (en) * | 2019-04-24 | 2020-10-29 | University Of Florida Research Foundation, Incorporated | Heparanase compounds and methods of use |
| KR20240035820A (ko) | 2021-07-09 | 2024-03-18 | 플렉시움 인코포레이티드 | Ikzf2를 조절하는 아릴 화합물 및 약학 조성물 |
| CN119174818A (zh) * | 2023-06-21 | 2024-12-24 | 厦门大学 | Otub2抑制剂及其在肿瘤免疫中的应用 |
Family Cites Families (2)
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|---|---|---|---|---|
| AU2002230057A1 (en) * | 2001-01-29 | 2002-08-12 | Insight Strategy And Marketing Ltd | Diphenyl ether derivatives and their uses as heparanase inhibitors |
| WO2002060867A2 (en) * | 2001-01-29 | 2002-08-08 | Insight Strategy And Marketing Ltd | Carbazole derivatives and their uses as heparanase inhibitors |
-
2005
- 2005-02-06 US US10/588,554 patent/US20070185176A1/en not_active Abandoned
- 2005-02-06 AU AU2005211255A patent/AU2005211255A1/en not_active Abandoned
- 2005-02-06 EP EP05703192A patent/EP1720828A2/en not_active Withdrawn
- 2005-02-06 WO PCT/IL2005/000149 patent/WO2005074375A2/en not_active Ceased
- 2005-02-06 CA CA002555313A patent/CA2555313A1/en not_active Abandoned
- 2005-02-06 JP JP2006552017A patent/JP2007525494A/ja not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20070185176A1 (en) | 2007-08-09 |
| JP2007525494A (ja) | 2007-09-06 |
| WO2005074375A3 (en) | 2009-04-23 |
| WO2005074375A2 (en) | 2005-08-18 |
| AU2005211255A1 (en) | 2005-08-18 |
| EP1720828A2 (en) | 2006-11-15 |
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| FZDE | Discontinued |