CA2512879A1 - N-cyclohexylaminocarbonyl benzenesulfonamide derivatives - Google Patents
N-cyclohexylaminocarbonyl benzenesulfonamide derivatives Download PDFInfo
- Publication number
- CA2512879A1 CA2512879A1 CA002512879A CA2512879A CA2512879A1 CA 2512879 A1 CA2512879 A1 CA 2512879A1 CA 002512879 A CA002512879 A CA 002512879A CA 2512879 A CA2512879 A CA 2512879A CA 2512879 A1 CA2512879 A1 CA 2512879A1
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- Prior art keywords
- compound
- compounds
- inhibitors
- effective amount
- treating
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- DNIIWANRGRGVRG-UHFFFAOYSA-N 1-(benzenesulfonyl)-3-cyclohexylurea Chemical class C=1C=CC=CC=1S(=O)(=O)NC(=O)NC1CCCCC1 DNIIWANRGRGVRG-UHFFFAOYSA-N 0.000 title claims abstract description 7
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- C—CHEMISTRY; METALLURGY
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
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Landscapes
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- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US44076103P | 2003-01-17 | 2003-01-17 | |
| US60/440,761 | 2003-01-17 | ||
| PCT/US2004/000689 WO2004066963A2 (en) | 2003-01-17 | 2004-01-13 | N-cyclohexylaminocarbonyl benzenesulfonamide derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2512879A1 true CA2512879A1 (en) | 2004-08-12 |
Family
ID=32825142
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002512879A Abandoned CA2512879A1 (en) | 2003-01-17 | 2004-01-13 | N-cyclohexylaminocarbonyl benzenesulfonamide derivatives |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US7319170B2 (en:Method) |
| EP (1) | EP1587535A4 (en:Method) |
| JP (1) | JP2007504285A (en:Method) |
| AU (1) | AU2004207444B2 (en:Method) |
| CA (1) | CA2512879A1 (en:Method) |
| WO (1) | WO2004066963A2 (en:Method) |
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| KR20060056944A (ko) | 2003-07-14 | 2006-05-25 | 아레나 파마슈티칼스, 인크. | 대사 조절제로서 융합된 아릴 및 헤테로아릴 유도체 및이에 관련된 장애의 예방 또는 치료 |
| WO2006057503A1 (en) * | 2004-11-25 | 2006-06-01 | Lg Life Sciences, Ltd. | NOVEL COMPOUNDS AS AGONIST FOR PPARϜ AND PPARα, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME |
| WO2006057505A1 (en) * | 2004-11-25 | 2006-06-01 | Lg Life Sciences, Ltd. | NOVEL COMPOUNDS AS AGONIST FOR PPARϜ AND PPARα, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME |
| MY148521A (en) | 2005-01-10 | 2013-04-30 | Arena Pharm Inc | Substituted pyridinyl and pyrimidinyl derivatives as modulators of metabolism and the treatment of disorders related thereto |
| EP1841422A1 (en) * | 2005-01-18 | 2007-10-10 | Novartis AG | Methods of use of dual ppar agonist compounds and drug delivery devices containing such compounds |
| ATE539743T1 (de) * | 2005-06-27 | 2012-01-15 | Newtree Co Ltd | Verfahren zur prävention und behandlung von ppar- vermittelten zuständen mit macelignan |
| EP1785133A1 (en) * | 2005-11-10 | 2007-05-16 | Laboratoires Fournier S.A. | Use of fenofibrate or a derivative thereof for preventing diabetic retinopathy |
| WO2007058504A1 (en) * | 2005-11-21 | 2007-05-24 | Lg Life Sciences, Ltd. | Novel compounds as agonist for ppar gamma and ppar alpha, method for preparation of the same, and pharmaceutical composition containing the same |
| US20080020014A1 (en) * | 2006-07-19 | 2008-01-24 | Paul Consigny | Implantable devices containing nuclear receptor ligands for the treatment of vascular and related disorders |
| US20080194575A1 (en) * | 2006-10-04 | 2008-08-14 | Naiara Beraza | Treatment for non-alcoholic-steatohepatitis |
| AU2008240158B2 (en) * | 2007-04-11 | 2014-07-10 | Omeros Corporation | Compositions and methods for prophylaxis and treatment of addictions |
| US20160331729A9 (en) * | 2007-04-11 | 2016-11-17 | Omeros Corporation | Compositions and methods for prophylaxis and treatment of addictions |
| US11241420B2 (en) | 2007-04-11 | 2022-02-08 | Omeros Corporation | Compositions and methods for prophylaxis and treatment of addictions |
| MX2007006092A (es) * | 2007-05-21 | 2009-02-25 | World Trade Imp Export Wtie Ag | Composiciones farmaceuticas que comprenden la combinacion de un agente derivado hidrogenado de lipstatina y un agente inhibidor de hmg-coa reductasa. |
| JO2870B1 (en) | 2008-11-13 | 2015-03-15 | ميرك شارب اند دوهم كورب | Amino Tetra Hydro Pirans as Inhibitors of Peptide Dipeptide IV for the Treatment or Prevention of Diabetes |
| WO2010056717A1 (en) | 2008-11-17 | 2010-05-20 | Merck Sharp & Dohme Corp. | Substituted bicyclic amines for the treatment of diabetes |
| WO2011011508A1 (en) | 2009-07-23 | 2011-01-27 | Schering Corporation | Benzo-fused oxazepine compounds as stearoyl-coenzyme a delta-9 desaturase inhibitors |
| WO2011011506A1 (en) | 2009-07-23 | 2011-01-27 | Schering Corporation | Spirocyclic oxazepine compounds as stearoyl-coenzyme a delta-9 desaturase inhibitors |
| US8552022B2 (en) | 2009-08-13 | 2013-10-08 | Merck Sharp & Dohme Corp. | Substituted cyclopropyl compounds, compositions containing such compounds and methods of treatment |
| MX2012002633A (es) | 2009-09-02 | 2012-04-20 | Merck Sharp & Dohme | Aminotetrahidropiranos como inhibidores de la dipeptidil peptidasa iv para el tratamiento prevencion de la diabetes. |
| EP2538783B1 (en) | 2010-02-22 | 2016-06-01 | Merck Sharp & Dohme Corp. | Substituted aminotetrahydrothiopyrans and derivatives thereof as dipeptidyl peptidase-iv inhibitors for the treatment of diabetes |
| EP2571876B1 (en) | 2010-05-21 | 2016-09-07 | Merck Sharp & Dohme Corp. | Substituted seven-membered heterocyclic compounds as dipeptidyl peptidase-iv inhibitors for the treatment of diabetes |
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| US5254589A (en) * | 1991-10-15 | 1993-10-19 | Warner-Lambert Company | Sulfonyl urea and carbamate ACAT inhibitors |
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| WO2001016120A1 (en) * | 1999-08-27 | 2001-03-08 | Eli Lilly And Company | Biaryl-oxa(thia)zole derivatives and their use as ppars modulators |
| AU7115300A (en) * | 1999-09-08 | 2001-04-10 | Glaxo Group Limited | Oxazole ppar antagonists |
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| EP1587535A4 (en) | 2010-02-24 |
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| US7319170B2 (en) | 2008-01-15 |
| WO2004066963A3 (en) | 2004-11-11 |
| AU2004207444A1 (en) | 2004-08-12 |
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